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(1S,2R)-N2-tert-butyl-N1-[2-(diethylamino)ethyl]-N1-methylcyclohexane-1,2-dicarboxamide
[(2,4-difluoro-3-methoxyphenyl)methyl](2-methoxyethyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
4-(furan-3-yl)-6-methyl-N-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
1-(azocan-1-yl)-3-[2-methoxy-5-({[2-(methylsulfanyl)ethyl]amino}methyl)phenoxy]propan-2-ol
2-cyclopentyl-N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}acetamide
4,5-dimethyl-2-(1H-pyrrol-1-yl)-N-(4H-1,2,4-triazol-4-yl)thiophene-3-carboxamide
4-{[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl}morpholine
N-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]cyclopropanesulfonamide
4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]-1-(2-phenylethyl)piperidine
(2S,4S)-4-amino-1-[2-(phenylformamido)acetyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
3-{1-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]piperidin-3-yl}benzoic acid
2-(3,4-dichlorophenyl)-4-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)morpholine
N-[(2-methylphenyl)methyl]-2-{2-[2-(morpholin-4-yl)ethyl]piperidin-1-yl}acetamide
2-acetyl-8-(4-carbamoyl-1,3-thiazol-2-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-ethyl-3-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-[2-(1H-pyrazol-1-yl)ethyl]benzamide
N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
2-{4-[(4-fluorophenyl)methyl]-1-(3-methylbutyl)piperazin-2-yl}ethan-1-ol
N-ethyl-N-[2-hydroxy-2-(3-hydroxyphenyl)ethyl]-1-methyl-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
4,6-dimethyl-N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}pyrimidin-2-amine
N-(5-chloro-2-methoxyphenyl)-3-[1-(cyclopent-1-ene-1-carbonyl)piperidin-3-yl]propanamide
7,7-dimethyl-2-(oxan-4-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-ethyl-N-{2-[(pyridin-3-yl)amino]ethyl}piperidine-2-carboxamide
1-(2-hydroxypyridine-3-carbonyl)-3-(2-methoxyethyl)piperidine-3-carboxylic acid
3-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-5,5-dimethyl-1,3-oxazolidine-2,4-dione
N-[(1S,2R)-2-(cyclooctylamino)cyclobutyl]benzenesulfonamide
6-[(3-methoxyphenyl)methoxy]-1-(2-phenylethyl)-4-[3-(pyrazin-2-yl)propanoyl]-1,4-diazepan-2-one
(3aS,6aR)-3-[2-(4-methoxyphenyl)ethyl]-5-[(5-methylthiophen-2-yl)methyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-cyclopentyl-2-{[1-(morpholin-4-ylmethyl)cyclohexyl]amino}propanamide
N-{2-hydroxy-2-[3-(trifluoromethyl)phenyl]ethyl}-2-methylimidazo[1,2-a]pyridine-6-carboxamide
N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-6-oxo-1-(3-phenylpropyl)piperidine-3-carboxamide
1-{[2-(azepane-1-carbonyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl}piperidin-4-ol
5-{[3-cyclopropyl-1-(2-methoxyphenyl)-1H-1,2,4-triazol-5-yl]methyl}-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
2,6-dimethyl-5-(2-{5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-oxoethyl)-3,4-dihydropyrimidin-4-one
ethyl 1-[2-(2,3-dihydro-1H-inden-1-yl)acetamido]cyclobutane-1-carboxylate
N-[1-(pyrazin-2-yl)piperidin-3-yl]-1H-indazole-3-carboxamide
4-{1-benzyl-5-[(5-methylfuran-2-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}morpholine
5-[5-(furan-2-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]-2-(propylsulfanyl)pyrimidine
1-methyl-5-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
5-{[2-(2-phenylethyl)piperidin-1-yl]sulfonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
5-[4-(adamantan-1-yl)piperazin-1-yl]-3-(morpholine-4-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazole
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(5-methylthiophene-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[2-(2,3-dihydro-1-benzofuran-5-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]-3-methoxypropanamide
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-3-(2-oxopyrrolidin-1-yl)-N-(pyridin-3-ylmethyl)propanamide
(3S,9aR)-3-[(2S)-butan-2-yl]-8-(quinolin-8-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
ethyl 1-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
4-ethyl-1-methyl-3-{1-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
[(1-tert-butyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl](ethyl){[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-[2-(2-methyl-1H-indol-3-yl)ethyl]-6-oxo-1-(pyridin-2-ylmethyl)piperidine-3-carboxamide
2-{3-[4-(2-methylphenyl)-3-oxopiperazin-1-yl]-3-oxopropyl}-2,3-dihydro-1H-isoindol-1-one