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methyl({[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}){[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}amine
[1-(3,6,7-trimethyl-1-benzofuran-2-carbonyl)piperidin-2-yl]methanol
3-{4-[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidin-1-yl]-4-oxobutyl}-3,4-dihydroquinazolin-4-one
1-[3-(4-methoxyphenyl)-1H-pyrazole-5-carbonyl]azocane
[(3R,4R)-1-(4-methoxy-2-methylbenzoyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
methyl 3-[(3S,4R)-4-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)-1-[(5-methylfuran-2-yl)methyl]piperidin-3-yl]propanoate
3-cyano-N-[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]benzamide
5-phenyl-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
N-{5H,6H,7H,8H,9H,10H,11H-cycloocta[b]indol-2-ylmethyl}-2-(2,4-dioxoimidazolidin-1-yl)acetamide
(3R,4R)-N-benzyl-4-hydroxy-4-(2-methoxyethyl)-N,3-dimethylpiperidine-1-sulfonamide
7-(1-benzothiophen-3-yl)-4-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-{4-[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]phenoxy}acetic acid
2-{[4-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]methyl}-8-methoxyquinoline
5-{2-methyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-5-oxopentanamide
4-({4-[methyl(2-phenylethyl)amino]-6-oxo-1,6-dihydropyridazin-1-yl}methyl)benzamide
[1-(1,3-benzothiazol-2-yl)-3-[(4-fluorophenyl)methyl]piperidin-3-yl]methanol
(2S)-2-amino-1-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-3-(1H-imidazol-4-yl)propan-1-one
3-[3-(3-ethylphenoxy)azetidine-1-carbonyl]-N,N-dimethylaniline
1-[2-(3,4-dihydro-2H-1,4-benzoxazin-4-yl)-2-oxoethyl]-4-phenylpyrrolidin-2-one
1-phenyl-2-[2-(quinolin-2-yl)-1H-imidazol-1-yl]ethan-1-ol
N-ethyl-1-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}-N-(pyridin-4-ylmethyl)piperidin-3-amine
1-[2-amino-6-methyl-5-(prop-2-en-1-yl)pyrimidin-4-yl]-3-(hydroxymethyl)pyrrolidin-3-ol
5-{2-[1-(2-hydroxyethyl)-3-(phenoxymethyl)-1H-1,2,4-triazol-5-yl]ethyl}-4,6-dimethylpyrimidin-2-ol
(2H-1,3-benzodioxol-5-ylmethyl)(methyl)[(5-{[(2-methylphenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)methyl]amine
3-(aminomethyl)-4-(4-chlorophenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}({[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl})amine
N-(dicyclopropylmethyl)-2-(4-fluorophenoxymethyl)-N-methyl-1,3-oxazole-4-carboxamide
{1-[7-(1H-imidazol-4-ylmethyl)-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]piperidin-3-yl}methanol
N-{4-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]-4-oxobutyl}acetamide
N-(1-{1-[(4-acetamidophenyl)methyl]piperidin-4-yl}-2-(2-fluorophenyl)ethyl)-N,2-dimethylfuran-3-carboxamide
N-benzyl-1-{2-[(2,5-dimethoxyphenyl)formamido]ethyl}-N-methyl-1H-1,2,3-triazole-4-carboxamide
2-({2-[2-(dimethylamino)ethoxy]-3-methoxyphenyl}methyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
4-phenyl-1-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}azepane
N-ethyl-2-[1-(3-methylbutyl)-3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-4'-yl]propanamide
2-methyl-5-{4-[2-(2-oxopiperidin-1-yl)acetyl]piperazin-1-yl}-2,3-dihydropyridazin-3-one
6-{[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-2,4-dimethyl-5H,6H-furo[2,3-d]pyrimidine
3-(3,4-difluorophenyl)-N-[1-(2-phenylethyl)piperidin-3-yl]propanamide
N-({2-[4-(2-methoxyphenyl)piperazin-1-yl]pyridin-3-yl}methyl)cyclopropanecarboxamide
N-(2-methoxyethyl)-3-({1-[(3-methyl-1H-indol-2-yl)methyl]piperidin-4-yl}oxy)benzamide
2-(6-methoxynaphthalen-2-yl)-4-[(1-methyl-1H-imidazol-4-yl)sulfonyl]morpholine
6-methyl-2-{[2-({5-phenyl-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-yl}amino)ethyl]amino}-3,4-dihydropyrimidin-4-one
3-butyl-1-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)urea
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-[1-(4-methylphenyl)cyclopropanecarbonyl]pyrrolidin-3-yl]methanol
4-{[2-(3-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
3-(diphenylmethyl)-N-methyl-N-(thiophen-3-ylmethyl)-1,2-oxazole-5-carboxamide
N-[2-(2-methylphenyl)ethyl]-4-propylpyrimidine-5-carboxamide
2-{3-[(2-chlorophenyl)methoxy]phenyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]piperidine-1-sulfonamide
4-(4-chlorophenyl)-N-[(3R,4R)-4-(4-methylpiperazin-1-yl)oxolan-3-yl]butanamide
2-(1H-pyrazol-1-yl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]benzamide