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methyl 3-(2-methoxybenzamido)-5-{[2-(3-methoxyphenyl)acetamido]methyl}benzoate
1-(2-methyl-1,3-benzothiazol-5-yl)-3-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}urea
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-2-methoxy-N-methyl-2-phenylacetamide
1-{2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-1H-1,3-benzodiazole-5-carbonyl}piperidine-4-carbonitrile
N-[2-(dimethylamino)ethyl]-N-{[7-fluoro-2-(2-methylphenyl)quinolin-3-yl]methyl}-1,3-dimethyl-1H-pyrazole-5-carboxamide
2-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine-4-carboxamide
(4aS,8aR)-6-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]-1-(2-methylpropyl)-decahydro-1,6-naphthyridin-2-one
2-[2,2-bis(prop-2-en-1-yl)pyrrolidine-1-carbonyl]-1H-imidazole
methyl 4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
butyl 4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxylate
N,N-dimethyl-4-{4-methyl-5-[(4-methylpiperazin-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine-1-carboxamide
8-chloro-2-(furan-2-yl)-4-(2-methyl-1,4-oxazepane-4-carbonyl)quinoline
methyl 4-[4-(2-chloro-4-{[2-(dimethylamino)ethyl]carbamoyl}phenoxy)piperidin-1-yl]pentanoate
(3R,4S)-4-[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]oxolan-3-ol
N-[2-hydroxy-3-(3-methoxyphenoxy)propyl]-2-methyl-1,3-benzothiazole-6-carboxamide
methyl 3-(4-fluorobenzenesulfonamido)-5-{[(4-methyl-1H-imidazol-2-yl)formamido]methyl}benzoate
1-cyclopentyl-N3,N3-diethyl-4-oxo-N5-{[3-(trifluoromethyl)phenyl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
3-(azocan-1-yl)-N-cyclopropyl-N-(1-methylpiperidin-4-yl)propanamide
5-methoxy-2-{[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]methyl}-4H-pyran-4-one
N-cyclopropyl-4-methoxy-3-({[(2-methyl-1,3-thiazol-4-yl)methyl]carbamoyl}amino)benzamide
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(3-methylphenyl)methyl]piperidine
N,1,4,6-tetramethyl-2-oxo-N-[(1-phenylpyrrolidin-3-yl)methyl]-1,2-dihydropyridine-3-carboxamide
N-(3-{4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-oxopropyl)acetamide
N-{[2-(benzyloxy)phenyl]methyl}-1-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
7-(2-chloro-6-fluorobenzoyl)-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-(2-fluoro-3-methylphenyl)-2-[4-(2-methoxyethoxy)piperidin-1-yl]acetic acid
ethyl 1-{7-acetamido-1-[2-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazole-5-carbonyl}piperidine-3-carboxylate
1-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
(1S,2S,9R)-11-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
1-[6-(4-methylphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]azocane
N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
1-(diethylamino)-3-[5-({[(3-fluorophenyl)methyl]amino}methyl)-2-methoxyphenoxy]propan-2-ol
1-amino-N-[(3R,4S)-1-(3-methylpyrazin-2-yl)-4-(propan-2-yl)pyrrolidin-3-yl]cyclopropane-1-carboxamide
(2R,3R)-3-amino-1'-(4-methoxybenzoyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
1-{[2-(2,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(methoxymethyl)piperidine
N-{2-[3-(hydroxymethyl)piperidin-1-yl]ethyl}-5-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
N-{2-[ethyl(methyl)amino]butyl}-2-(4-fluorophenyl)imidazo[1,2-a]pyridine-6-carboxamide
N-[2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]-5-methyl-1,3,4-oxadiazol-2-amine
{1-[(1-hexylpiperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}methanol
1-(2-{[2-methyl-6-(piperidin-3-yl)pyrimidin-4-yl]amino}ethyl)piperidin-4-ol
(2S)-2-[(2-amino-5-butyl-6-methylpyrimidin-4-yl)amino]-3-hydroxypropanamide
7-(6-tert-butyl-2-oxo-2,3-dihydropyrimidine-4-carbonyl)-2,7-diazaspiro[4.4]nonane-1,3-dione
1-[(6-chloropyridin-3-yl)methyl]-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
[(3,4-dimethoxyphenyl)methyl](methyl){[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}amine
2-(3-methoxypropyl)-9-{[3-(methylsulfanyl)phenyl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
5-(4-methoxyphenyl)-3-[3-(morpholin-4-ylmethyl)piperidin-1-yl]-1,2,4-triazine
4-ethyl-6-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine
[(1-cyclopentylpiperidin-4-yl)methyl][(4-methoxyphenyl)methyl](pyridin-3-ylmethyl)amine
1-(4-chlorophenyl)-N-{[7-(6-methoxypyridazin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclobutane-1-carboxamide