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1-[(6-methylpyridin-2-yl)methyl]-4-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]piperazine
4-[(4-ethoxyphenyl)methyl]-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N,N-diethyl-2-{[4-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-2-oxo-1-(2-phenylethyl)-1,4-diazepan-6-yl]oxy}acetamide
3-(1,3-benzothiazol-5-yl)-1-methyl-1-[1-(pyridin-3-yl)pentyl]urea
N-{1-[5-(ethylsulfanyl)-4-methyl-4H-1,2,4-triazol-3-yl]ethyl}-2,4-dimethoxybenzamide
N-[1-({[phenyl(pyridin-4-yl)methyl]carbamoyl}methyl)-1H-pyrazol-4-yl]-2-(phenylsulfanyl)acetamide
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N-methyl-2-(phenylamino)pyrimidine-5-carboxamide
5-methoxy-4-oxo-N-(2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)-4H-pyran-2-carboxamide
2-[1-(2,2-dimethylpropyl)-4-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl]ethan-1-ol
4-(2-hydroxybutyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2-(methylamino)pyrimidine-5-carboxamide
3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-N-{1-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}propanamide
2-{methyl[1-(pyrimidin-4-yl)ethyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
N-[(2R,3R)-1'-(3-methoxybenzoyl)-2-(pyridin-4-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
6-({3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}methyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-[(2,3,4-trimethoxyphenyl)methyl]piperazine
3-ethyl-3-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-1-[3-(2-oxo-1,3-oxazolidin-3-yl)phenyl]urea
N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2-[1-(3-methylbut-2-en-1-yl)-3-oxopiperazin-2-yl]acetamide
5-({1-[(4-fluorophenyl)methyl]-3-hydroxy-2-oxopiperidin-3-yl}methyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonitrile
N-[2-(4-chlorophenyl)-2-(pyrrolidin-1-yl)ethyl]-2,6-dimethylpyridine-4-carboxamide
1-ethyl-3-[(3-methoxyphenyl)methyl]-8-[1-(pyridin-3-yl)propan-2-yl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(2-{1-[1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}ethyl)pyrrolidin-2-one
3-[2-(4-hydroxy-1-methylpiperidin-4-yl)ethyl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
N-(4-{[methyl({[1-(2-methylpropyl)pyrrolidin-3-yl]methyl})carbamoyl]methoxy}phenyl)propanamide
2-amino-N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-4-methyl-1,3-thiazole-5-carboxamide
N-(dimethyl-1H-1,2,4-triazol-5-yl)-3-({[(1,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)benzamide
N-(2-hydroxybutyl)-1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}piperidine-4-carboxamide
(2S)-2-({[(3-fluoro-4-methylphenyl)carbamoyl]methyl}amino)-3-methylbutanamide
1-[(3S,4R)-1-{[5-(2-cyanophenyl)furan-2-yl]methyl}-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
(3aS,6aS)-2-[(5-chlorofuran-2-yl)methyl]-5-cyclopentanecarbonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(3-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-5-yl)-3-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine-1-carboxamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-3-[4-(2-fluorophenyl)piperazine-1-carbonyl]-6-methyl-2-propyl-1,4-dihydropyridin-4-one
3-(4-methyl-1,3-thiazol-5-yl)-1-[4-(pyrimidin-2-yloxy)piperidin-1-yl]propan-1-one
(3R,4R)-4-amino-1-({2-[(2-chloro-6-fluorophenyl)methoxy]phenyl}methyl)piperidin-3-ol
2-(2,5-dioxo-1-propylimidazolidin-4-yl)-N-[(2-methyl-1H-1,3-benzodiazol-6-yl)methyl]acetamide
6-[(3R,4R)-3-{[ethyl(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]pyrazine-2-carboxylic acid
[3-(cyclopropylmethyl)-1-{5-[(4-methylpiperazin-1-yl)methyl]pyridin-2-yl}piperidin-3-yl]methanol
N-{1-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]ethyl}-2,6-dimethylaniline
2-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrole-1-carbonyl]-6-chloro-3-fluoroimidazo[1,2-a]pyridine
1-[6-(oxan-2-ylmethyl)-1,2,3,4-tetrahydroquinolin-1-yl]ethan-1-one
(3S,4R)-1-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
N,N-dimethyl-3-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrazin-2-amine
(2S,4R)-4-{[(4-chlorophenyl)methyl]amino}-N-(2-methoxyethyl)-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
5-({imidazo[2,1-b][1,3]thiazol-6-ylmethyl}amino)-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
N-[(3S,4R)-1-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
N-cyclopropyl-N-{[2-(dimethylamino)-7-methylquinolin-3-yl]methyl}-2,2-diphenylacetamide
methyl 3-benzamido-1-(furan-2-ylmethyl)-5-({[3-(2-hydroxyethoxy)phenyl]methyl}amino)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-[(3-methylphenyl)methyl]piperidine
2-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
4-{[4-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)phenyl]methyl}-1λ6-thiomorpholine-1,1-dione