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3-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-4-(2H-1,3-benzodioxol-5-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(2S,4S)-4-amino-N-methyl-1-[(3R)-3-phenylbutanoyl]pyrrolidine-2-carboxamide
methyl 3-(2,6-difluorobenzoyl)-7-oxo-9-(3-phenylpropoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
5-{[4-(methylsulfanyl)phenyl]methyl}-5-{3-oxo-3-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]propyl}pyrrolidin-2-one
(2S)-N-[4-(difluoromethoxy)-3-ethoxyphenyl]-2-(methoxymethyl)pyrrolidine-1-carboxamide
5-[4-(2,2-dimethylpropanoyl)piperazin-1-yl]-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
1-(1,4-dithiepan-6-yl)-3-[3-(propan-2-yloxy)benzoyl]piperidine
2-methoxy-N-[4-methyl-3-({[(5-methyl-1,2-oxazol-3-yl)methyl]carbamoyl}amino)phenyl]acetamide
5-methoxy-3-({2-[2-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}methyl)-1H-indazole
(2S,4R)-4-amino-1-{[2-(benzyloxy)phenyl]methyl}-N-ethylpyrrolidine-2-carboxamide
3-ethyl-5-(1-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1H-imidazol-2-yl)-1,2-oxazole
3-(2,6-dimethylhept-5-en-1-yl)-9-methoxy-N-[(2-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
(1R,5R)-6-[2-(4-fluorophenoxy)ethyl]-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane
1-[2-(dimethylamino)-2-(4-methylphenyl)ethyl]-3-(4-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)urea
N-{1-[7-(2,2-diphenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]-2-methylpropyl}methanesulfonamide
ethyl 4-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]piperazine-1-carboxylate
(2S,3R)-2-amino-3-hydroxy-1-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}butan-1-one
7-[4-(3,5-dimethyl-1H-pyrazol-1-yl)butanoyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
4-amino-2-{4-[(4-ethyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}pyrimidine-5-carbonitrile
1-(2-carbamoylethyl)-N-[4-(2-fluorophenoxy)phenyl]piperidine-4-carboxamide
1-(3,5-dimethyl-1-benzofuran-2-carbonyl)-2-(3-methoxyphenyl)pyrrolidine
1-[(2-methyl-1H-indol-3-yl)methyl]-4-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidin-4-ol
1-{4-[(4-chloro-2-fluorophenyl)methyl]-6-hydroxy-1,4-diazepan-1-yl}ethan-1-one
(1R,3S,5S)-8-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]-8-azabicyclo[3.2.1]octan-3-ol
(3S,4S)-4-cyclopropyl-1-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]pyrrolidine-3-carboxylic acid
(3S,5R)-1-[(2-methoxyphenyl)methyl]-5-[(pyridin-4-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(3-methyl-1,2-oxazole-5-carbonyl)piperidine
1-{1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carbonyl}azocane
2-(3-{[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]methyl}phenoxy)ethan-1-ol
2-[(1,3-benzothiazol-2-yl)amino]-1-{1-oxa-8-azaspiro[4.5]decan-8-yl}ethan-1-one
1-[(3-cyclohexyl-1,2-oxazol-5-yl)methyl]azepan-3-amine
1-{1-[6-(azepan-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperidin-4-yl}piperidin-3-ol
2-[7-(2-methoxyethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-5,6-dimethylpyridine-3-carbonitrile
N-[3-(4-fluorophenyl)-3-(furan-2-yl)propyl]-4-hydroxy-2-methylpyrimidine-5-carboxamide
ethyl 1-[(4-hydroxy-3,5-dimethoxyphenyl)methyl]-3-(2-phenoxyethyl)piperidine-3-carboxylate
[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]({[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
2-[(2-fluorophenyl)methyl]-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
4-[2-(1-{[3-(hydroxymethyl)-4-methoxyphenyl]methyl}piperidin-2-yl)ethyl]phenol
1-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)-3-ethylurea
N-[(1-methylpiperidin-3-yl)methyl]-3-(2-oxopiperidin-1-yl)-N-(2-phenylethyl)propanamide
N-ethyl-5-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine-1-carbonyl}pyrimidin-2-amine
3-fluoro-5-[4-(1-hydroxy-3-phenylpropyl)piperidine-1-carbonyl]benzonitrile
3-{1-[2-(dimethyl-1,3-thiazol-5-yl)acetyl]piperidin-3-yl}-N-[(3-methoxyphenyl)methyl]propanamide
N,1-dimethyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
ethyl 2-{[4-(4-cyclohexyl-1H-1,2,3-triazol-1-yl)piperidine-1-carbonyl]amino}acetate
1-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-3-(3-methoxybenzoyl)piperidine
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(pyridazine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-(azepan-1-yl)-3-{5-[(2,5-dimethoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl}propan-1-one
1-[7-(5-chloro-2-methoxyphenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(3,4,5-trimethoxyphenyl)ethan-1-one