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4-methyl-2-(1-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}piperidin-4-yl)-1H-1,3-benzodiazole
methyl 6-{2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}pyrazine-2-carboxylate
(2-{4-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-ylmethyl]phenoxy}ethyl)dimethylamine
N-(1H-1,3-benzodiazol-2-ylmethyl)-1-(cyclohexylmethyl)-N-methyl-6-oxopiperidine-3-carboxamide
3-[(1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}pyrrolidin-3-yl)methyl]benzamide
2-[4-(1-benzothiophen-2-ylmethyl)-1-cyclopentylpiperazin-2-yl]ethan-1-ol
methyl (2S)-1-{[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}pyrrolidine-2-carboxylate
N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-3-(1-methylpiperidin-2-yl)propanamide
N-(3-methyl-1,2,4-thiadiazol-5-yl)-4-(pyridin-4-yl)-1,4-diazepane-1-carboxamide
N-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]-3-fluoropyridine-4-carboxamide
4-{[(3-hydroxypyrrolidin-3-yl)methyl]amino}-N-phenylpiperidine-1-carboxamide
5-({2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}methyl)-2-methoxybenzoic acid
2-ethyl-8-[3-(2-hydroxyphenyl)-1H-pyrazole-5-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
N-[3-(dimethylamino)-2,2-dimethylpropyl]-5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carboxamide
[(5-tert-butyl-1H-pyrazol-3-yl)methyl][(3-methylthiophen-2-yl)methyl](pyridin-2-ylmethyl)amine
1-(2,3-dihydro-1H-inden-2-yl)-N-(4-methoxyphenyl)piperidin-3-amine
N-({1-[(2-fluorophenyl)methyl]-2-(propane-2-sulfonyl)-1H-imidazol-5-yl}methyl)-N-methyloxolan-3-amine
(2R,3R)-3-(1,4-oxazepan-4-yl)-1'-(pyridin-2-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-[3-oxo-4-(pent-4-en-1-yl)-3,4-dihydro-2H-1,4-benzoxazin-2-yl]acetic acid
5-butyl-1'-(1-methyl-1H-pyrazole-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-(1-benzofuran-2-yl)-2-{5-methyl-4-[4-(propan-2-yl)piperazine-1-carbonyl]-1H-pyrazol-1-yl}pyrimidine
methyl (2S,3S)-2-{[1-benzyl-5-(cyclopropylcarbamoyl)-4-oxo-1,4-dihydropyridin-3-yl]formamido}-3-methylpentanoate
1-(3-phenylpropyl)-N-[2-(pyridin-3-yloxy)phenyl]piperidine-3-carboxamide
5-chloro-3-(4-cyclobutanecarbonyl-1,4-diazepane-1-carbonyl)-4,6-dimethyl-1,2-dihydropyridin-2-one
N-[2-({thieno[2,3-d]pyrimidin-4-yl}amino)ethyl]pyridine-3-carboxamide
N-({2-[benzyl(methyl)amino]-2,3-dihydro-1H-inden-2-yl}methyl)but-2-ynamide
N-methyl-5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1H-pyrazole-3-carboxamide
(3S,4R)-4-(hydroxymethyl)-1-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-ol
2-(4-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1-(3-methylbut-2-en-1-yl)piperazin-2-yl)ethan-1-ol
(1R,3S)-3-(2-aminoethoxy)-7-[1-(2-fluorophenyl)piperidin-4-yl]-7-azaspiro[3.5]nonan-1-ol
1-{2-[(2-chlorophenyl)methyl]morpholin-4-yl}-3-(1-methylcyclopropyl)propan-1-one
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-{[(2,5-dimethylphenyl)methyl]amino}-1-(propan-2-yl)pyrrolidine-2-carboxamide
{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)(2-phenylethyl)amine
6-methyl-4-oxo-N-[2-(3-propoxyphenyl)ethyl]-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
1-(1-benzofuran-2-ylmethyl)azepan-3-amine
5-[2-oxo-2-(4-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidin-1-yl)ethyl]imidazolidine-2,4-dione
N-{[(2S)-1-ethylpyrrolidin-2-yl]methyl}-2-(pyridin-3-yl)pyrimidine-5-carboxamide
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(pyridin-2-ylmethyl)acetamide
N-(1-{7-[(2,3-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-methoxypropanamide
N-benzyl-1-cyclopentyl-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-(5,6-dimethylpyrazin-2-yl)pyrrolidin-3-yl]oxane-4-carboxamide
[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl](ethyl)(oxan-2-ylmethyl)amine
N,N-diethyl-2-[9-methoxy-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetamide
8-{3-fluoro-5-methylimidazo[1,2-a]pyridine-2-carbonyl}-1-oxa-8-azaspiro[4.5]decane
N-{1-[1-(3-amino-1H-1,2,4-triazole-5-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
2-({2,7-dimethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)-N-methylethane-1-sulfonamide
N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
2-(methylamino)-1-(2-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl)ethan-1-one
(3S,4R)-1-[2-(2-methyl-1H-1,3-benzodiazol-5-yl)acetyl]-4-phenylpyrrolidine-3-carboxylic acid
2,5-dimethyl-3-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]pyrazine