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(4aS,8aR)-1-(2-methylpropyl)-6-[4-(1H-1,2,4-triazol-1-yl)butanoyl]-decahydro-1,6-naphthyridin-2-one
2-(3,5-difluorophenyl)-1-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]ethan-1-one
N-{[2-(4-chlorophenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)furan-2-carboxamide
(2E)-3-(2-chlorophenyl)-N-{[4-(4-methoxyphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}prop-2-enamide
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-4-hydroxy-2-(4-methylphenyl)pyrimidine-5-carboxamide
4-{4-[1-(piperidin-1-yl)ethyl]phenyl}-1H-pyrazole-3-carbonitrile
5-{[1-(3-methylbutyl)-1H-1,3-benzodiazol-2-yl]methyl}-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
2-{2-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-1-yl}pyridine
(3S,4R)-1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
methyl (2S)-1-[3-(3,5-difluorobenzoyl)-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl]pyrrolidine-2-carboxylate
1-(furan-2-ylmethyl)-4-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-1,4-diazepan-6-ol
3-[3-(dimethylamino)propyl]-8-[(2-methoxyphenyl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-(1-ethoxy-2-methylpropan-2-yl)-1-[2-(2-methoxyphenoxy)phenyl]urea
(4S,4aS,8aS)-1-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-4-phenyl-decahydroquinolin-4-ol
N-{[7-chloro-2-(3-methylphenyl)quinolin-3-yl]methyl}-2,3-dimethoxy-N-(2-methoxyethyl)benzamide
4-({1-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]pyrrolidin-3-yl}methyl)benzoic acid
N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-N'-(2-methylphenyl)propanediamide
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(1-methyl-1H-pyrazole-5-carbonyl)piperidine-4-carboxamide
ethyl 1-(furan-2-ylmethyl)-4-(2-phenylethyl)piperidine-4-carboxylate
{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[3-(1H-pyrazol-1-yl)phenyl]methyl}amine
8-(2-hydroxypropanoyl)-3-{2-[4-(propan-2-yl)piperazin-1-yl]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(2H-1,2,3-benzotriazol-2-yl)-1-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}ethan-1-one
1-(2-methyl-4-phenylpiperazin-1-yl)-2-(pyridin-4-ylsulfanyl)ethan-1-one
N-{1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-2-(3-methyl-1,2-oxazol-5-yl)acetamide
3-(oxolan-3-yl)-5-{1,3,6-trimethyl-1H-pyrazolo[3,4-b]pyridin-4-yl}-1,2,4-oxadiazole
4-[3-(cyclopropylmethyl)-1-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-1,2,4-triazol-5-yl]-N-methyl-1,3-thiazol-2-amine
3-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-1-(6-fluoropyridin-3-yl)urea
(4aS,8aR)-1-(4-hydroxybutyl)-6-(5-methyl-1,3-benzoxazol-2-yl)-decahydro-1,6-naphthyridin-2-one
3-[1-({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-2-yl]pyridine
N-{[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
N-butyl-N-[(4-fluorophenyl)methyl]-1,5-dimethyl-1H-pyrrole-2-carboxamide
1-[4-(furan-2-ylmethoxy)phenyl]-3-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}urea
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-N'-(2-ethoxyphenyl)propanediamide
N-methyl-2-(morpholin-4-yl)-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]pyrimidine-5-carboxamide
3-[(4-butyl-1H-1,2,3-triazol-1-yl)methyl]-1-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}piperidine
N-[(2-ethoxyphenyl)methyl]-N-(2-hydroxyethyl)-N'-(4-methylphenyl)propanediamide
N-[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]-2-(dimethyl-1,2-oxazol-4-yl)acetamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]piperidin-3-ol
(1R,5S,6R)-3-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-3-azabicyclo[3.1.0]hexane-6-carboxylic acid
3-cyclohexyl-1-[3-(5-methyl-2-{[2-(morpholin-4-yl)ethyl]sulfanyl}pyrimidin-4-yl)piperidin-1-yl]propan-1-one
2-methyl-N-(naphthalen-1-yl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
N-{1-[4-(piperidin-3-yl)benzoyl]piperidin-4-yl}methanesulfonamide
4-benzyl-1-{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}piperidine
4-[(3S,5R)-3-(hydroxymethyl)-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidine-1-carbonyl]benzonitrile
N-[(5-fluoro-2-methylphenyl)methyl]-4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}benzamide
4-(4-fluorophenyl)-2-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}phenol
4-{2-[(1R,5S)-6-azabicyclo[3.2.1]octan-6-yl]-2-oxoethyl}-1-methyl-2,3,4,5-tetrahydro-1H-1,4-benzodiazepine-2,5-dione
N-[(1-methanesulfonylpiperidin-3-yl)methyl]-4-(propan-2-yl)-1,3-thiazole-2-carboxamide
1-[4-(5-methylpyridin-2-yl)-4-(pyrrolidin-1-ylmethyl)piperidin-1-yl]ethan-1-one
4-[4-cyclohexyl-3-oxo-6-(pyridin-2-ylmethoxy)-1,4-diazepane-1-carbonyl]-2-methyl-1,2-dihydrophthalazin-1-one