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2-methyl-6-{1-[4-(propan-2-yloxy)benzoyl]piperidin-3-yl}pyrimidin-4-ol
5-chloro-3-methyl-N-{2-[3-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]propyl}-1H-indole-2-carboxamide
N-(1-{7-[(2,4-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)pyridine-2-carboxamide
2-{5-[(dimethylamino)methyl]-1-(2,3-dimethylphenyl)-1H-1,2,4-triazol-3-yl}acetamide
N-{[2-(3-chlorophenyl)-7-fluoroquinolin-3-yl]methyl}-2-oxo-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
2-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
3-{2-oxo-2-[4-(pyridin-4-yl)piperazin-1-yl]ethyl}-4-(3-phenylpropyl)piperazin-2-one
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-(dimethylamino)-N-methyl-2-(4-methylphenyl)acetamide
1-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine
{[2-methoxy-5-(6-methyl-1H-1,3-benzodiazol-2-yl)phenyl]methyl}dimethylamine
N-[2-(1-methanesulfonylpiperidin-2-yl)ethyl]-6-methylimidazo[1,2-a]pyridine-2-carboxamide
(3aS,6aS)-2-[2-(dimethylamino)acetyl]-5-(3-methoxypyrazin-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[2-(3-fluorophenyl)piperidine-1-carbonyl]-4-methylpiperazine
2-(3-fluorophenyl)-1-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidine
1-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-2-phenoxyethan-1-one
1-(2-cyclohexylethyl)-3-hydroxy-3-{[(pyridin-4-ylmethyl)amino]methyl}piperidin-2-one
(3R,5S)-N-methyl-5-(pyrrolidine-1-carbonyl)-N-(quinoxalin-2-ylmethyl)piperidine-3-carboxamide
4-{[5-(2,2-dimethyloxan-4-yl)-1,2,4-oxadiazol-3-yl]methyl}-1-propylpiperidine
1-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-3-(1-methyl-1H-imidazol-2-yl)piperidine
3-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-9-methoxy-N-[(2-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
ethyl 3-{[(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)carbamoyl]amino}propanoate
8-cyclopropanecarbonyl-2-[3-(1H-pyrazol-1-yl)propanoyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-{3-[(diethylamino)methyl]phenyl}-3-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)urea
N-[1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetamide
4-({5-[1-(cyclopropanesulfonyl)piperidin-3-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)morpholine
3-(3-methoxybenzoyl)-1-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidine
N-({2-[(dimethylamino)methyl]phenyl}methyl)-N,2,5-trimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
2-(3,4-dichlorophenyl)-4-(4-propylpyrimidine-5-carbonyl)morpholine
N-[1-(butan-2-yl)-1H-pyrazol-5-yl]-2-(3,4,5-trimethoxyphenyl)acetamide
2-[5-(1-phenylmethanesulfonylpyrrolidin-2-yl)-1,2,4-oxadiazol-3-yl]pyridine
2-({[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}amino)pyridine-3-carbonitrile
3-[4-(2-methoxyquinolin-3-yl)-1H-pyrazol-1-yl]propanamide
4-(hydroxymethyl)-1-{[2-(2-phenylethoxy)phenyl]methyl}azepan-4-ol
N-cyclopropyl-3-{5-[2-(2-oxo-1,2-dihydropyridin-1-yl)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
6-[(diethylamino)methyl]-N-[(6-methylpyridin-2-yl)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
3-cyclopentyl-N-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}propanamide
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N-methyl-4-(piperidin-1-ylmethyl)benzamide
3-{3-[2-(5-chlorothiophen-2-yl)-1H-imidazol-1-yl]propyl}pyridine
1-ethyl-4-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
1-{1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-4-yl}-2-[2-(2-methoxyphenyl)ethyl]-1H-1,3-benzodiazole
1-(4-{[3-(2,2-dimethylpiperazine-1-carbonyl)-1,2-oxazol-5-yl]methoxy}phenyl)ethan-1-one
5-oxo-1-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}pyrrolidine-3-carboxylic acid
(4aS,7aR)-1-(2,6-dimethylpyrimidine-4-carbonyl)-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-methyl-3-[3-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-4-phenylpyridine
5-(5-chloro-2-oxo-1,2-dihydropyridine-3-carbonyl)-1-(cyclopropylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-{[8-(1-oxo-1,2-dihydroisoquinoline-4-carbonyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}acetamide
8-butanoyl-3-{2-[cyclohexyl(methyl)amino]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-{[2-(4-methoxyphenyl)ethyl]amino}-1-(3-methylpiperidin-1-yl)propan-1-one
[(3-chloro-4,5-dimethoxyphenyl)methyl]({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)methylamine
8-[2-(1H-1,2,4-triazol-1-yl)benzoyl]-1-oxa-8-azaspiro[4.5]decane