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3-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-[(1R)-1-(4-methoxyphenyl)ethyl]benzamide
N-({4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-1,3-dimethyl-1H-pyrazole-5-carboxamide
(2S)-2-[2-(5-methylfuran-2-yl)-1H-imidazol-1-yl]propanamide
8-fluoro-N-[2-(N-methylmethanesulfonamido)ethyl]quinoline-2-carboxamide
4-{4-[6-(cyclopentylamino)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperazin-1-yl}phenol
N-(furan-2-ylmethyl)-3-(2-hydroxyphenyl)-N-(pyridin-2-ylmethyl)-1H-pyrazole-5-carboxamide
3-[1-(1-ethyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(cyclobutylmethyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-methyl-4-(4-methylphthalazin-1-yl)phenol
5-cyclobutyl-N-{[5-(2,6-difluorophenyl)-1,2,4-oxadiazol-3-yl]methyl}-1,3,4-oxadiazol-2-amine
5-(3-{[4-(pentan-2-yl)-1H-1,2,3-triazol-1-yl]methyl}phenyl)-1H-1,2,3,4-tetrazole
8-(5-carboxypyridin-2-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-amino-4-cyclopropyl-6-(4-methanesulfonylphenyl)pyridine-3-carbonitrile
2-{[3-({2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}carbamoyl)phenyl]amino}acetic acid
9-(5,6-dimethylpyrimidin-4-yl)-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
N4-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-5,6,7,8-tetrahydroquinazoline-2,4-diamine
5-(dimethylamino)-2-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2,3-dihydropyridazin-3-one
4-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-1H-pyrazole-3-carbonitrile
methyl[(2-methyl-1,3-oxazol-4-yl)methyl]{[3-(methylsulfanyl)phenyl]methyl}amine
N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)-3-(1H-pyrazol-1-yl)propanamide
N,N,1-trimethyl-2-oxo-1,2-dihydrospiro[indole-3,4'-piperidine]-1'-sulfonamide
5-(furan-2-carbonyl)-3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N-{[7-(5-acetyl-2-fluorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(2,5-dioxoimidazolidin-4-yl)acetamide
4-acetamido-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-methylbenzamide
N-tert-butyl-2-[(2-methyl-5-propylpyrimidin-4-yl)amino]acetamide
2-ethyl-9-(1-ethyl-1H-pyrazole-3-carbonyl)-4-phenyl-2,9-diazaspiro[5.5]undecane
9-(1-methyl-5-oxopyrrolidine-3-carbonyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
{1-[(3-chloropyridin-4-yl)methyl]-3-(2-methylpropyl)piperidin-3-yl}methanol
3-(4-chlorophenyl)-6-[5-ethyl-3-(oxan-4-yl)-1H-1,2,4-triazol-1-yl]pyridazine
1-{[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]amino}propan-2-ol
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-2-(2-fluorophenoxymethyl)-N-methyl-1,3-oxazole-4-carboxamide
(2S,4R)-N-(8-chloroquinolin-5-yl)-4-(dimethylamino)-2-(hydroxymethyl)pyrrolidine-1-carboxamide
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
N-[(4-acetamidophenyl)methyl]-2-{[1-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}acetamide
methyl 4-[(7-{[4-hydroxy-4-(pyridin-3-yl)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)methyl]benzoate
N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
7-methyl-2-{[2-(propylamino)pyrimidin-5-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(3-ethoxy-2-hydroxypropyl)amine
6-(2-hydroxyethyl)-N-[1-(2-methoxyphenyl)propan-2-yl]-N-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide
methyl 3-[(3,4-dimethoxyphenyl)methyl]-7-oxo-9-[2-(thiophen-3-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4-[2-oxo-2-(2-phenylmorpholin-4-yl)ethyl]-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
2-cyclopentyl-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
8-[(1R,9aR)-octahydro-1H-quinolizin-1-ylmethoxy]quinoline-2-carboxamide
1-({4-[(4-ethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)-4-(pyridin-3-yl)piperidin-4-ol
8-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-cyclopropyl-N-({3-[(1-methoxypropan-2-yl)oxy]phenyl}methyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-8-(4-methyl-1H-pyrrole-2-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(2,3-dihydro-1H-inden-2-yl)-N-methyl-N-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}piperidin-3-amine
N-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxamide
1-(3-fluorophenyl)-3-{1-[1-(1H-pyrrole-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea