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8-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)-5-fluorophenyl]methyl}-1,3-dioxa-8-azaspiro[4.5]decan-2-one
1-[2-(1H-1,3-benzodiazol-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]-2-(1H-pyrazol-1-yl)butan-1-one
methyl N-(1-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}ethyl)carbamate
3-[(2R,3R,6R)-5-[4-(dimethylamino)benzoyl]-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)-1-(2,2-diethylcyclopropanecarbonyl)piperidine
3-[(1-cyclopentylpyrrolidin-3-yl)methyl]benzamide
1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-3-(1H-pyrazol-5-yl)piperidine
5-methyl-3-[2-(morpholin-4-yl)ethyl]-5-[1-(4-phenylbenzoyl)piperidin-4-yl]imidazolidine-2,4-dione
1-cycloheptanecarbonyl-4-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]piperidine
5-(azocan-1-yl)-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole
ethyl 1-[(2,4-dimethylphenyl)carbamoyl]-4-(2-phenylethyl)piperidine-4-carboxylate
N-(isoquinolin-5-ylmethyl)-N-methyl-1-(2-methyl-6-propylpyrimidin-4-yl)piperidin-4-amine
1-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pentane-1,2-dione
9-[2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)acetyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(2-methylpyrimidin-4-yl)-4-(quinolin-6-yloxy)piperidine-4-carboxylic acid
2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(1,2-oxazol-3-ylmethyl)acetamide
4-{[3-(2-hydroxyethyl)-4-(3-methylbut-2-en-1-yl)piperazin-1-yl]methyl}-2,6-dimethylphenol
(2R,3R)-3-{methyl[3-(2-methylphenoxy)propyl]amino}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
3-({4-[1-(1-methyl-1H-pyrazole-5-carbonyl)pyrrolidin-3-yl]piperidin-1-yl}methyl)pyridine
4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)-N-(4-ethylphenyl)piperidine-1-carboxamide
2-cyclohexyl-5-{[3-(methanesulfonylmethyl)piperidin-1-yl]methyl}pyrimidine
N-(cyclopropylmethyl)-6-(3-methoxyphenyl)-N-propylimidazo[2,1-b][1,3]thiazole-3-carboxamide
3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]-1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidine
(4aR,6R,8aS)-8a-(methoxymethyl)-2-[2-(methylsulfanyl)pyrimidin-4-yl]-6-(morpholin-4-yl)-decahydroisoquinoline
(2S,4S)-4-[(4-fluorophenyl)sulfanyl]-N-(2-methyl-1,3-benzothiazol-5-yl)-1-(propan-2-yl)pyrrolidine-2-carboxamide
5-(morpholin-4-ylmethyl)-N-[1-(thiophen-2-yl)butyl]furan-3-carboxamide
1-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-methylpentane-1,4-dione
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N,2,3,5-tetramethylpyrazolo[1,5-a]pyrimidin-7-amine
2-({[(4-fluorophenyl)methyl](pyridin-4-ylmethyl)amino}methyl)-6-methylpyridin-3-ol
7-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
5-methoxy-3-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-1H-indole-2-carboxamide
1-(4-benzylpiperazin-1-yl)-3-{1-[(3-fluorophenyl)methyl]piperidin-3-yl}propan-1-one
(3aS,6aS)-2-acetyl-5-[(2,4-dichlorophenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}piperidine-3-carbonitrile
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-[2-(benzenesulfonyl)ethyl]-1-(4-fluorophenyl)-3-methyl-1H-1,2,4-triazole
N-cyclopentyl-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)-2H-1,3-benzodioxole-5-carboxamide
(3S,4R)-N,N-dimethyl-1-(6-phenylpyridazin-3-yl)-4-propylpyrrolidin-3-amine
2-{4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-3-carbonitrile
3-[3-ethyl-5-(1-methyl-2-oxo-1,2-dihydropyridin-3-yl)-1H-1,2,4-triazol-1-yl]-4-fluorobenzene-1-sulfonamide
N-[1-(cyclohex-1-en-1-yl)ethyl]-3-(2-methoxyphenyl)-1H-pyrazole-5-carboxamide
2-{[5-(4-cyanophenyl)-4-(2-methoxyphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-[(2R,3R)-2-methoxy-1'-(quinoxalin-5-ylmethyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenylacetamide
N-(1-ethyl-5-oxopyrrolidin-3-yl)-2-[(quinolin-6-yloxy)methyl]-1,3-oxazole-4-carboxamide
3-{[1-(2-methoxybutanoyl)piperidin-4-yl]methyl}-1-methyl-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[2-(3-methoxyphenoxy)ethyl]-2-azaspiro[4.4]nonan-3-one
{3-[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3-oxopropyl}urea
3-[4-(5-ethyl-2-methylpyrimidin-4-yl)phenyl]propanoic acid
4-{3-[(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]propoxy}benzamide