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1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine
N-{1-[1-(2,1,3-benzoxadiazol-5-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2,2-dimethylpropanamide
2-(furan-2-yl)-1-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]azepane
N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
3-[(3R,4S)-1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
1-(4-{[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]methyl}phenyl)-1H-1,2,4-triazole
8-(oxan-4-yl)-1-(2-phenylethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{[1-butyl-2-(4-methylpentanesulfonyl)-1H-imidazol-5-yl]methyl}-1,4-diazepan-5-one
methyl 4-{[3-(2-hydroxyethyl)-4-(3-methylbut-2-en-1-yl)piperazin-1-yl]methyl}benzoate
N-ethyl-N-[2-(4-fluorophenoxy)ethyl]-2,4-dimethylpyrimidine-5-carboxamide
5-(4-methylpiperidin-1-yl)-1-(prop-2-en-1-yl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
ethyl (4aR,6R,8aS)-6-(morpholin-4-yl)-2-(pyrazin-2-yl)-decahydroisoquinoline-8a-carboxylate
N-[(3R,4S)-1-[(4-cyanophenyl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]-2-hydroxyacetamide
1-(4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzoyl)piperidin-3-ol
2,3,6-trimethyl-4-[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]quinoline
1-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-2-(methoxymethyl)piperidine
2-(3-hydroxypropyl)-9-(1,3-thiazol-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-{1-benzyl-4-[(4-methoxy-3-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
2-cyclopropyl-4-(4-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidine-1-carbonyl}piperidin-1-yl)-2,3-dihydro-1H-isoindole-1,3-dione
ethyl 4-benzyl-1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxylate
1-{3-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidine-1-carbonyl]phenyl}pyrrolidin-2-one
(cyclopropylmethyl)({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)(oxolan-2-ylmethyl)amine
4-{[4-methoxy-2-methyl-5-(propan-2-yl)phenyl]methyl}-1-phenylpiperazin-2-one
2-(4-{[2-(furan-2-yl)phenyl]methyl}-1-methylpiperazin-2-yl)ethan-1-ol
N-(3,4-dimethoxyphenyl)-1-(6-methylpyridine-2-carbonyl)piperidin-3-amine
2-({4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}methyl)-N-[2-(1,3-thiazol-4-yl)ethyl]-1,3-oxazole-4-carboxamide
2-methoxy-N-[3-(4-{[2-(thiophen-2-yl)ethyl]amino}piperidin-1-yl)phenyl]benzamide
4-[4-(4-ethylpiperazin-1-yl)piperidin-1-yl]-N-(1-phenylethyl)benzamide
2-{4-[(5-ethylfuran-2-yl)methyl]-1-(2-phenylethyl)piperazin-2-yl}ethan-1-ol
N-(2-{3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}ethyl)acetamide
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-3-(4H-1,2,4-triazol-4-yl)benzamide
N-{[1-(1-carbamoylethyl)-1,2,3,6-tetrahydropyridin-4-yl]methyl}adamantane-1-carboxamide
1-(4-{[3-(3-fluoro-4-methoxybenzoyl)piperidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
2-chloro-5-acetamido-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}benzamide
8-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one
1-[4-(dimethylamino)-5-fluoropyrimidin-2-yl]-4-(pyridin-3-yl)piperidin-4-ol
1-[(3-methoxyphenyl)methyl]-4-({4-[(thiophen-2-ylmethyl)amino]quinazolin-2-yl}methyl)piperazin-2-one
6-[1-benzyl-3-(pyrrolidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-2,3,4,5-tetrahydropyridazin-3-one
1-methyl-4-{[4-phenyl-5-(thiophen-3-yl)-1H-imidazol-1-yl]methyl}pyrrolidin-2-one
3-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-3-methyl-1-{4-[(trifluoromethyl)sulfanyl]phenyl}urea
{3-[(2-fluorophenyl)methyl]-1-[3-(methylsulfanyl)propyl]piperidin-3-yl}methanol
N-cyclopropyl-N-[(2-methoxyphenyl)methyl]-5-phenyl-1,2-oxazole-3-carboxamide
5-[(4-fluorophenyl)methyl]-5-{1-[2-(2-methylphenyl)acetyl]piperidin-4-yl}-3-(oxolan-3-yl)imidazolidine-2,4-dione
6-(1-benzothiophen-3-yl)-2-{4-[3-(hydroxymethyl)piperidin-1-yl]piperidin-1-yl}-N-(propan-2-yl)pyridine-3-carboxamide
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-[2-(pyridin-2-ylsulfanyl)acetamido]acetic acid
3-[3-({[2-(4-hydroxypiperidin-1-yl)ethyl]amino}methyl)-1H-indol-1-yl]propanamide
N'-cyclooctyl-N-methyl-N-[1-(methylcarbamoyl)propan-2-yl]butanediamide
3-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-6-methylpyridazine
7-(1,3-benzothiazol-2-yl)-4-[2-(1H-pyrazol-1-yl)ethyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-[2-(2-methoxyphenyl)ethyl]-5-(1-methyl-1H-imidazol-2-yl)-4-phenyl-1H-imidazole