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2,3-dimethyl-6-[2-(piperidin-1-ylmethyl)-1,4-oxazepane-4-carbonyl]quinoxaline
2-({[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}amino)pyridine-3-carbonitrile
N-[(3S,5S)-5-(diethylcarbamoyl)-1-(oxan-4-yl)pyrrolidin-3-yl]-2-oxo-2,3-dihydro-1H-imidazole-4-carboxamide
1-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
N-[(2S)-1-methoxypropan-2-yl]-4-{[(3R)-3-methylpiperazin-1-yl]sulfonyl}benzamide
2-methoxy-4-[3-(pyridin-2-yl)azetidin-1-yl]pyridine-3-carbonitrile
N-{[5-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-3-yl]methyl}-1-benzylpyrrolidin-3-amine
5-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)-1-cyclopentylpiperidin-2-one
(1R,7S)-3-tert-butyl-6-[3-(morpholin-4-yl)azetidine-1-carbonyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
7-[2-(1-methyl-1H-indol-3-yl)acetyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
1-[(1S,5R)-6-(4-fluoro-3-methylbenzoyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
4-methyl-7-(4H-1,2,4-triazol-4-yl)-2H-chromen-2-one
1-benzyl-N-(1-methoxypropan-2-yl)-2-methyl-5-(2-methylpropanamido)-1H-1,3-benzodiazole-7-carboxamide
4-{4-[3-(4-hydroxyphenyl)-1H-pyrazole-5-carbonyl]piperazin-1-yl}benzonitrile
1-(3,5-dimethyl-1-benzofuran-2-carbonyl)-4-(4-methoxybenzoyl)piperazine
N-{[2-(4-acetylpiperazin-1-yl)-5,8-dimethoxyquinolin-3-yl]methyl}-2-fluoro-N-(oxolan-2-ylmethyl)benzamide
3-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]-1-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperidine
N-[1-({[3-(1H-indazol-1-yl)propyl]carbamoyl}methyl)-1H-pyrazol-4-yl]-3-phenoxypropanamide
3-(1-{6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidine-3-carbonyl)pyridine
2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}acetamide
4-{[4-(4-methoxyphenoxy)piperidin-1-yl]methyl}-2-(propan-2-yl)pyrimidine
N-(2,1,3-benzothiadiazol-5-ylmethyl)-1-(2-methoxyacetyl)piperidine-3-carboxamide
3-{2-oxo-2-[4-(1H-1,2,4-triazole-3-carbonyl)piperazin-1-yl]ethyl}-3,4-dihydroquinazolin-4-one
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]pyrazin-2-amine
8-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
3-benzoyl-9-[(1-propyl-1H-imidazol-2-yl)methyl]-3,9-diazaspiro[5.5]undecane
methyl 5-[(cyclohex-3-en-1-ylmethyl)amino]-3-(2-methoxyacetamido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-6-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-(1H-1,3-benzodiazol-1-yl)-1-{2-[(2-chlorophenyl)methyl]morpholin-4-yl}ethan-1-one
N-[2-(2-oxo-1,3-oxazolidin-3-yl)phenyl]-4-(pyrimidin-2-yloxy)piperidine-1-carboxamide
1-({[(3-{3-[cyclohexyl(methyl)amino]-2-hydroxypropoxy}phenyl)methyl]amino}methyl)cyclohexan-1-ol
3-[4-(4-methoxybenzoyl)piperazine-1-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
[(2,4-dimethoxy-3-methylphenyl)methyl](methyl)[2-(oxan-4-yl)ethyl]amine
(3R,4R)-4-(4-hydroxypiperidin-1-yl)-1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-3-ol
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]quinoxaline-6-carboxamide
4-({4-[(3,5-dimethylphenyl)methyl]-3-oxopiperazin-1-yl}methyl)-1-methyl-1H-pyrrole-2-carbonitrile
1'-(2-chloro-4-fluorobenzoyl)-5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
methyl 3-[3-(cyclopentylcarbamoyl)-1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propanoate
1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-amine
N-(3-methoxypropyl)-2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
3-(piperazine-1-sulfonyl)-N-[3-(1H-1,2,4-triazol-1-yl)propyl]benzamide
methyl 9-(2,3-dihydro-1H-inden-2-yloxy)-7-oxo-3-(quinolin-2-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(2E)-3-(3-fluorophenyl)-1-{4-[3-({methyl[2-(1H-1,2,4-triazol-1-yl)ethyl]amino}methyl)phenoxy]piperidin-1-yl}prop-2-en-1-one
8-methoxy-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(2-methylpropyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-(pyrimidin-2-yl)piperazine-2-carboxylic acid
N-{[4-(4-fluorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}naphthalene-1-carboxamide
1-[4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-2-(1H-indazol-1-yl)ethan-1-one
3-[2-(3-benzoylpiperidin-1-yl)-2-oxoethyl]-3-(2-fluorophenyl)-1-(2-methoxyethyl)pyrrolidine-2,5-dione
2-{4-[(2-phenyl-1,3-thiazol-5-yl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
2-chloro-4-[5-(piperidin-1-ylmethyl)pyridin-2-yl]benzamide