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N,2,2,6,6-pentamethyl-N-[1-(pyrazine-2-carbonyl)piperidin-4-yl]piperidin-4-amine
N,N,4-trimethyl-6-(2,4,6-trimethylphenyl)pyrimidin-2-amine
2-(furan-3-carbonyl)-7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-6-one
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-1,6-dimethyl-4-oxo-1,4-dihydroquinoline-3-carboxamide
5-chloro-N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-6-oxo-1,6-dihydropyridine-3-carboxamide
{[(3S,4R)-1-(5-ethylthiophene-3-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl}dimethylamine
4,4-difluoro-N-[3-(methylsulfamoyl)phenyl]piperidine-1-carboxamide
N-({3,5-dimethoxy-4-[2-(1-methylpyrrolidin-2-yl)ethoxy]phenyl}methyl)-4-methoxy-N-[(3S)-2-oxoazepan-3-yl]benzene-1-sulfonamide
N6-benzyl-N5-methyl-N5-(pyridin-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
2-({[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl](methyl)amino}methyl)benzonitrile
ethyl 4-{5-cyclopropyl-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}piperazine-1-carboxylate
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-[3-(3-fluorophenyl)-1H-pyrazol-4-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-{4-[(3-chlorophenyl)methyl]piperazin-1-yl}-2-[methyl(piperidin-4-yl)amino]ethan-1-one
methyl 4-methoxy-3-[({2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}carbamoyl)amino]benzoate
2-[2-(propan-2-yl)-1H-imidazol-1-yl]-1-[3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]propan-1-one
(2S)-2-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]pyrrolidine-1-carboxamide
1-(2,1,3-benzoxadiazol-4-ylmethyl)-N-[4-(furan-2-yl)phenyl]piperidine-3-carboxamide
3-{1-[(3-chloropyridin-4-yl)methyl]piperidin-3-yl}-N-(4-fluoro-2-methylphenyl)propanamide
2-[(4aR,7aS)-6,6-dioxo-4-[4-(1H-1,2,4-triazol-1-yl)butanoyl]-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
N-[4-(2-{[(2,3-dimethylphenyl)methyl]amino}acetamido)phenyl]-N-methylacetamide
6-[(2-fluorophenyl)methyl]-N-[(1-phenylcyclopentyl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
N-(2-ethylphenyl)-3-({2-[(prop-2-en-1-yl)amino]phenyl}formamido)propanamide
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-1-(propan-2-yl)piperidine-3-carboxamide
3-(dimethyl-1,2-oxazol-4-yl)-1-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]urea
3-(5-fluoro-1H-1,3-benzodiazol-2-yl)-1-{3-[(methylsulfanyl)methyl]piperidin-1-yl}propan-1-one
3-[({1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperidin-3-yl}oxy)methyl]pyridine
1-[1-(propan-2-yl)piperidin-4-yl]-N-(pyridin-4-ylmethyl)piperidine-3-carboxamide
4-[1-(3,4-dimethoxyphenyl)cyclopentanecarbonyl]-1,4-oxazepan-6-ol
N-benzyl-3-(1H-imidazol-2-yl)-N-methylimidazo[1,2-a]pyridine-2-carboxamide
N'-(2,4-dimethylphenyl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]propanediamide
2-methyl-N-[3-(methylsulfanyl)propyl]imidazo[1,2-a]pyrimidine-3-carboxamide
1-{4-[(4,4-difluoropiperidin-1-yl)methyl]-2-methoxyphenoxy}-3-[methyl(propan-2-yl)amino]propan-2-ol
7-[5-(pyrrolidin-2-yl)thiophene-2-carbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-3-[(3S,4R)-4-(morpholin-4-yl)-1-(naphthalen-1-ylmethyl)piperidin-3-yl]propan-1-one
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-2-(3,5-dimethyl-1H-pyrazol-1-yl)acetamide
[1-(dimethyl-1,3-thiazol-4-yl)ethyl](methyl)({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)amine
1-{[4-(propan-2-yl)pyrimidin-2-yl]amino}-3-(pyrrolidin-1-yl)propan-2-ol
N-(1-{1-[(2-ethoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-phenylpropanamide
N-phenyl-1-[3-(thiophen-3-yl)-1H-pyrazole-5-carbonyl]piperidin-3-amine
2-ethoxy-6-{[3-(2-hydroxyethyl)-4-(3-phenylpropyl)piperazin-1-yl]methyl}phenol
2-{[4-hydroxy-4-(pyridin-3-yl)piperidin-1-yl]methyl}-3,5-dimethoxybenzoic acid
N-[(2,4-dimethoxyphenyl)methyl]-3-[1-(1H-pyrrole-2-carbonyl)piperidin-3-yl]propanamide
5-(4-methoxy-3,5-dimethylphenyl)pyrimidin-2-amine
methyl 6-({[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}amino)pyridine-3-carboxylate
6-(difluoromethyl)-2-[4-({ethyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
6-[3-(4-methoxy-2-methylbenzoyl)piperidin-1-yl]-9H-purin-2-amine
4-{4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-6-methylpyrimidine
1-ethyl-2-{4-[1-(2-methoxyethyl)-1,2,3,6-tetrahydropyridin-4-yl]-1H-pyrazol-1-yl}-1H-1,3-benzodiazole
N-[2-(3-{[methyl(quinolin-8-ylmethyl)amino]methyl}phenoxy)ethyl]cyclohexanecarboxamide
5-[4-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]-1-(3-phenylpropyl)piperidin-2-one