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2-methyl-N-{[8-({4-[methyl(phenyl)amino]phenyl}methyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}propanamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
6-[2-(4-chlorophenoxy)acetyl]-N-[(6-methylpyridin-2-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
(2R,3R,6R)-5-[(4-methoxypyridin-2-yl)methyl]-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
5-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-3-propyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
4-[3-(1-ethyl-1H-pyrazol-3-yl)phenyl]-6-methyl-2-(propan-2-yl)pyrimidine
N-(2-hydroxyethyl)-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-propyl-1,3-oxazole-4-carboxamide
(4aS,8aR)-6-(pyridine-2-carbonyl)-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
7-(4-fluorophenyl)-2-{imidazo[1,2-a]pyridin-3-ylmethyl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
4-[(4-ethoxyphenyl)methyl]-3-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]piperazin-2-one
N-(2H-1,3-benzodioxol-5-yl)-5-[1-(propan-2-yl)pyrrolidin-2-yl]thiophene-2-carboxamide
N-[2-(3-methoxypropanoyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]-3-(4-methylphenyl)propanamide
ethyl 3-(2-phenylethyl)-1-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperidine-3-carboxylate
2-amino-6-methyl-N-[(4-methylphenyl)(pyridin-4-yl)methyl]pyrimidine-4-carboxamide
N-cyclopropyl-5-(quinolin-8-yl)thiophene-2-carboxamide
2-methoxyethyl 2-(3-fluorophenyl)piperidine-1-carboxylate
2-ethyl-6-methyl-4-oxo-N-[2-(pyridin-2-yl)ethyl]-1-(thiophen-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
2-[3-(5-fluoro-2-methoxybenzoyl)piperidine-1-carbonyl]-N,N-dimethylaniline
1-(3,5-dimethylfuran-2-carbonyl)-4-(pyridin-3-yl)piperazine
1-{2-phenylimidazo[1,2-a]pyridine-6-carbonyl}-4-(trifluoromethyl)piperidine
1-{3-[2-(1-ethyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]propyl}-3,5-dimethyl-1H-1,2,4-triazole
1-benzyl-5-acetamido-N-(2-{imidazo[1,2-a]pyrimidin-2-yl}ethyl)-2-methyl-1H-1,3-benzodiazole-7-carboxamide
N-{4-chloro-3-[(3R)-3-hydroxypyrrolidine-1-carbonyl]phenyl}acetamide
N-(3-hydroxypropyl)-2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}-N-(propan-2-yl)acetamide
4-chloro-2-methyl-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)benzamide
1-[(4-ethylphenyl)methyl]-5-(oxolan-3-yl)-1H-1,2,4-triazole
(3aR,6aR)-2-{2-[4-(dimethylamino)phenyl]acetyl}-5-(2-methoxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[4-(2-aminopyrimidin-4-yl)piperidin-1-yl]-2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]ethan-1-one
ethyl 4-(cyclopropylmethyl)-1-{[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}piperidine-4-carboxylate
1-methyl-4-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
2-{4-[(5-chloro-2,3-dimethoxyphenyl)methyl]-1-[(2-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
5-cyclopropyl-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-1,3,4-oxadiazol-2-amine
3-(3-methylbutyl)-8-(pent-4-enoyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[3-(3-fluorophenyl)phenyl]-1-{[5-(hydroxymethyl)furan-2-yl]methyl}piperidine-4-carboxamide
(5S,9aS,9bS)-2-(2-methoxyphenyl)-5-[(E)-2-(2-methoxyphenyl)ethenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-(3-hydroxyazetidin-1-yl)-4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]butan-1-one
N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-2-oxo-6-phenyl-1,2-dihydropyridine-3-carboxamide
N5-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N5,N6,N6-trimethyl-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
(3S,5R)-1-[(3,4-dimethoxyphenyl)methyl]-N3-[(1-ethylpyrrolidin-2-yl)methyl]-N5-(4-fluorophenyl)piperidine-3,5-dicarboxamide
2-amino-4-cyclopropyl-6-(4-fluorophenyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
1-cyclopentyl-N3-methyl-N5-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-N3-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
4-propyl-5-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]pyrimidine
1-(carbamoylmethyl)-N-{2-hydroxy-2-[4-(trifluoromethyl)phenyl]ethyl}piperidine-4-carboxamide
1-[2-(4-methoxyphenoxymethyl)-1,3-oxazole-4-carbonyl]-4-(4-methylphenyl)piperazine
1-[(3R,4S)-3-amino-4-phenylpyrrolidin-1-yl]-2-(azocan-1-yl)ethan-1-one
3-fluoro-4-methoxy-N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}benzamide
1-(4-{1-oxa-7-azaspiro[3.5]nonane-7-carbonyl}phenyl)pyrrolidin-2-one
5-benzamido-1-cyclopentyl-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-1H-1,3-benzodiazole-7-carboxamide
2-methoxy-1-[4-(4-methoxyphenoxy)piperidin-1-yl]ethan-1-one
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)pyrimidin-2-amine