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1-{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine
2,3-dimethyl-7-{[5-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
1-cyclobutanecarbonyl-N-[(dimethyl-1,3-thiazol-5-yl)methyl]piperidine-4-carboxamide
3-[4-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
N-[(1S,2S)-1-amino-2,3-dihydro-1H-inden-2-yl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
2-{[4-(2-methoxy-5-methylphenyl)-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
2-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrol-2-yl]-4-(3,3,3-trifluoropropyl)pyrimidine
[1-(3-phenylprop-2-yn-1-yl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl]methanol
N-[(3S,4R)-1-[2-(5-methyl-1H-pyrazol-1-yl)acetyl]-4-(4-methylphenyl)pyrrolidin-3-yl]cyclopropanecarboxamide
(1H-1,3-benzodiazol-2-ylmethyl)(methyl){[(1R,5S,6R)-3-(morpholine-4-carbonyl)-3-azabicyclo[3.1.0]hexan-6-yl]methyl}amine
5-[(quinolin-6-yloxy)methyl]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1,2-oxazole-3-carboxamide
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-1-[4-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]ethan-1-one
4-methyl-N-{[1-(3-methylphenyl)pyrrolidin-3-yl]methyl}pyrimidin-2-amine
2-ethyl-8-(2-ethyl-4-methyl-1,3-thiazole-5-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
2-(3-chloro-4-hydroxyphenyl)-N-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}acetamide
(5S,9aS,9bS)-5-[4-ethoxy-3-(hydroxymethyl)phenyl]-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-cyclopropyl-1-[(1s,4s)-4-{[(2,4-dimethoxyphenyl)methyl]amino}cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
methyl 6-({4-[2-(methylsulfanyl)pyrimidin-4-yl]piperazin-1-yl}methyl)pyridine-2-carboxylate
{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}({2-[4-(propan-2-yloxy)phenyl]ethyl})amine
1-[(4-fluorophenyl)methyl]-N-(oxolan-2-ylmethyl)-N-(pyridin-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-(morpholin-4-yl)-3-(1-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-yl)propan-1-one
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-1-[(3,4-dimethoxyphenyl)methyl]-N5-(2-methylpropyl)piperidine-3,5-dicarboxamide
(1H-1,3-benzodiazol-2-ylmethyl)(butyl)(furan-2-ylmethyl)amine
5-({3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}methyl)pyrimidin-2-amine
N-[1-(1-benzothiophen-2-ylmethyl)piperidin-4-yl]methanesulfonamide
2-(dimethyl-1,3-thiazol-5-yl)-N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)acetamide
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-5-(3,4-dimethylphenoxymethyl)-N-methyl-1,2-oxazole-3-carboxamide
4-[3-(3-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]butanamide
3-[1-(cyclopentylmethyl)piperidin-3-yl]-N-[(2,4-dimethoxyphenyl)methyl]propanamide
4-(cyclopropylmethyl)-1-(1-methyl-1H-indazole-3-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
2-(2,4-dioxoimidazolidin-1-yl)-N-[2-methyl-1-(5-methyl-1H-1,3-benzodiazol-2-yl)propyl]acetamide
9-[2-(benzyloxy)ethyl]-3-oxa-9-azaspiro[5.5]undecane
3-methyl-7-(pyridin-2-ylmethyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
N-[2-(2-methoxyphenyl)ethyl]-2-propyl-1,3-thiazole-4-carboxamide
5-methanesulfonyl-N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-(piperidin-3-yl)pyrimidin-2-amine
3-[3-(3-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1H-indazole
butyl[(4-chloro-1-methyl-1H-pyrazol-3-yl)methyl](furan-2-ylmethyl)amine
3-[({[5-(4-methoxyphenyl)-1,2-oxazol-3-yl]methyl}amino)methyl]pyrrolidin-3-ol
1-(1-{1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-3-yl)propan-1-one
7-(pyridin-2-yl)-4-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(1R,3s,6r,8S)-4-(2-ethylpyrimidine-5-carbonyl)-4-azatricyclo[4.3.1.13,8]undecane
N-cyclopentyl-5-(methoxymethyl)-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)furan-2-carboxamide
N-{[5-chloro-7-(1H-indol-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(2-oxoimidazolidin-1-yl)benzamide
N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
2,4-difluoro-N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methylbenzamide
5-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-ylmethyl}-2-(propylsulfanyl)pyrimidine
5-(4-methylphenyl)-N-[1-(pyridin-4-yl)propyl]-1H-pyrazole-3-carboxamide
ethyl 5-[(4-carbamoylpiperidin-1-yl)methyl]-1-(4-methylphenyl)-1H-pyrazole-4-carboxylate
2-amino-8-(5-ethylfuran-2-yl)-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
N-(1-{7-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-2-carboxamide