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3-chloro-5-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl}-1,2-dihydropyridin-2-one
4-[2-(3,5-dimethyl-1H-pyrazol-4-yl)pyridine-4-carbonyl]morpholine
N-{[3-(oxolan-3-ylmethoxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)-2-(trifluoromethyl)benzene-1-sulfonamide
1-(4-benzylpiperazin-1-yl)-3-[1-(oxan-4-yl)piperidin-3-yl]propan-1-one
2-[4-(1,4-diazepane-1-carbonyl)phenoxy]-1-(piperidin-1-yl)ethan-1-one
1-(1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}pyrrolidin-3-yl)-3,5-dimethyl-1H-pyrazole
1-[2-(morpholin-4-yl)ethyl]-N-[1-(pyridin-4-yl)propyl]-1H-1,2,3-triazole-4-carboxamide
6-methoxy-N,1-dimethyl-N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-1H-indole-2-carboxamide
N-{1-[(2-chlorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-ethoxybenzamide
4-(2,5-dihydro-1H-pyrrol-1-ylmethyl)-N-[4-(hydroxymethyl)phenyl]benzamide
N-(2-{4-[1-(2-fluorophenyl)-1H-1,2,4-triazol-5-yl]phenoxy}ethyl)acetamide
1-[3-(1H-pyrazol-1-yl)propyl]-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
(3R,9aR)-3-[(1S)-1-hydroxyethyl]-8-(2-methoxybenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-[2-(dimethylamino)ethyl]-9-[2-(2,5-dimethylphenyl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
N-(2-{1-[(2-methylphenyl)methyl]piperidin-3-yl}ethyl)cyclopropanesulfonamide
(3aS,6aS)-2-(2-aminopyrimidin-4-yl)-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[5-({[(2-chlorophenyl)methyl]amino}methyl)-2-methoxyphenoxy]-3-(4-methyl-1,4-diazepan-1-yl)propan-2-ol
4-(1H-pyrazol-3-yl)-1-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)piperidine
(3S,4S)-4-({[(2-phenylphenyl)methyl]amino}methyl)piperidin-3-ol
ethyl[(1-methyl-1H-pyrazol-4-yl)methyl][(1-propyl-1H-imidazol-2-yl)methyl]amine
(1S,5R)-3-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(trifluoromethyl)pyridine
methyl 4-[2-(methylamino)pyridine-4-carbonyl]piperazine-1-carboxylate
2-(2-fluorophenyl)-N-methyl-N-{2-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}acetamide
4-(4-{[2-(2-fluorophenyl)ethyl]amino}piperidin-1-yl)-N,N-dimethylbenzamide
N-{[3-(3-methylbutyl)-3H-imidazo[4,5-b]pyridin-2-yl]methyl}morpholine-2-carboxamide
N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-N'-(4-methylphenyl)propanediamide
2-cyclopentyl-8-(2-methyl-6-oxo-1,6-dihydropyrimidine-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[3-(1H-imidazol-1-yl)propyl]-1-methyl-2-oxo-N-(pyridin-4-ylmethyl)-1,2-dihydropyridine-3-carboxamide
N-{6-methoxy-2-oxo-4-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-1,2,3,4-tetrahydroquinolin-7-yl}methanesulfonamide
3-[(3S,5S,9S)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]-1-(3-fluorophenyl)urea
methyl (2S,4R)-4-(dimethylamino)-1-{8-methylimidazo[1,2-a]pyridine-2-carbonyl}pyrrolidine-2-carboxylate
2-methyl-3-[3-(2-methylphenoxy)azetidine-1-carbonyl]-4,5,6,7-tetrahydro-1H-indol-4-one
9-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-1,4-diazepan-1-yl)ethan-1-one
2-(4-{2-methylpyrido[2,3-d]pyrimidin-4-yl}piperazin-1-yl)-1,3-benzoxazole
1-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}-3-(1-propyl-1H-1,2,4-triazol-3-yl)urea
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-(1H-pyrazol-1-yl)propanamide
methyl 3-({[3-(1H-imidazol-2-yl)propyl]carbamoyl}amino)-4-methylbenzoate
2-methyl-6-({8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}methyl)phenol
N-[2-(2-chlorophenoxy)ethyl]-6-cyanopyridine-3-carboxamide
2-ethyl-4-{[4-(thian-4-yl)piperazin-1-yl]methyl}pyrimidine
1-{4-[2-(3,4-dimethylpiperazin-1-yl)-2-oxoethoxy]phenyl}propan-1-one
methyl 4-{[1-(2-methoxyethyl)-2,4-dioxo-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-8-yl]methyl}benzoate
1-{4-[(2-fluorophenyl)methyl]piperidin-1-yl}-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propan-1-one
N-[2-(4-methoxyphenyl)ethyl]-1-methyl-N-[(1-methylpiperidin-4-yl)methyl]-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
(3R,4R)-4-(azepan-1-yl)-1-{[4-(pyrimidin-2-yloxy)phenyl]methyl}piperidin-3-ol
N-(1H-1,3-benzodiazol-2-ylmethyl)-2-[4-(2-methylquinolin-4-yl)-2-(morpholin-4-ylmethyl)phenoxy]acetamide
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)pyridine-2-carboxamide
N,2,4-trimethyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1,3-thiazole-5-carboxamide