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5-chloro-4-{1-[(2-chlorophenyl)methyl]-3-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1,3-dimethyl-1H-pyrazole
4-(2-methylphenoxy)-1-(oxolane-3-carbonyl)piperidine
N-[1-(1-{[4-ethoxy-3-(hydroxymethyl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]cyclopropanecarboxamide
N-(1-hydroxypropan-2-yl)-1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}piperidine-4-carboxamide
4-acetyl-N-{[7-fluoro-5-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
2-(2H-1,3-benzodioxol-5-yl)-N-[(2-{2-[(dimethylsulfamoyl)amino]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]acetamide
4-hydroxy-4-(methanesulfonamidomethyl)-N-(3-methoxyphenyl)azepane-1-carboxamide
4-[4-(1-benzofuran-5-carbonyl)piperazin-1-yl]quinazoline
dimethyl[2-(2-{1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperidin-3-yl}-1H-imidazol-1-yl)ethyl]amine
N3-(cyclohexylmethyl)-1-(2-methoxyethyl)-4-oxo-N5-[1-(thiophen-2-yl)propyl]-1,4-dihydropyridine-3,5-dicarboxamide
N,N-dimethyl-4-{4-[(3-methylpyridin-2-yl)methyl]piperazine-1-carbonyl}piperidine-1-carboxamide
1-methyl-6-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}-3-(2-phenylethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-(1-methyl-1H-1,2,3-triazol-4-yl)-3-({2-[5-(propan-2-yl)-1,2-oxazol-3-yl]pyrrolidin-1-yl}methyl)benzamide
6-ethyl-N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-2-oxo-1,2-dihydropyridine-4-carboxamide
(2S)-2-({[3-(1H-pyrazol-1-yl)phenyl]methyl}amino)propanamide
2-{4-[2-(trifluoromethyl)phenyl]-4H-1,2,4-triazol-3-yl}ethan-1-amine
1-({1-[4-hydroxy-2-(pyridin-3-yl)pyrimidine-5-carbonyl]piperidin-3-yl}methyl)pyrrolidin-2-one
1-[3-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)-3-oxopropyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
N,3-dimethyl-5-propyl-N-(1H-pyrazol-5-ylmethyl)-1-benzofuran-2-carboxamide
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-1-phenyl-1H-1,2,3-triazole-4-carboxamide
2-(pyrrolidin-1-ylmethyl)-1-[(2,4,6-trimethoxyphenyl)methyl]piperidine
(1R,3S)-7-(2-methoxybenzenesulfonyl)-7-azaspiro[3.5]nonane-1,3-diol
1-{4-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]phenyl}-3-(2-methylpropyl)-3-(thiophen-2-ylmethyl)urea
(1S,5R)-6-{[4-(1H-imidazol-1-yl)phenyl]methyl}-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
4-({3-[5-(2-fluorophenyl)-2-(pyridin-3-yl)pyrimidin-4-yl]piperidin-1-yl}methyl)phenol
1-(dimethyl-1,3-thiazole-5-carbonyl)-4-(2-methoxybenzoyl)piperazine
N-(2,3-dihydro-1H-inden-2-yl)-4-hydroxy-2-(pyridin-3-yl)pyrimidine-5-carboxamide
(3R,4S)-1-[(2-butyl-1H-imidazol-4-yl)methyl]-4-cyclopropylpyrrolidin-3-amine
(3R,4R)-4-(azepan-1-yl)-1-cycloheptylpiperidin-3-ol
1-{[5-(4-methoxyphenyl)furan-2-yl]methyl}-3-(5-methyl-1,2,4-oxadiazol-3-yl)piperidine
methyl 1-{3-[4-({[(1-ethyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]-2-hydroxypropyl}piperidine-4-carboxylate
4-{[(1,4-dioxan-2-ylmethyl)carbamoyl]amino}-N-(2-phenylethyl)benzamide
1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-4-[1-(pyridin-3-yl)propan-2-yl]piperazine
ethyl 4-(2-{4-[2-(phenylsulfanyl)acetamido]-1H-pyrazol-1-yl}acetyl)piperazine-1-carboxylate
(2S,4S)-N,1-diethyl-4-[3-(3-hydroxy-3-methylbutyl)benzamido]pyrrolidine-2-carboxamide
1-[(2-chlorophenyl)methyl]-N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
5-{1-[(2,4-dimethylphenyl)methyl]-4-hydroxypiperidin-4-yl}-N-(oxolan-2-ylmethyl)-1-benzofuran-2-carboxamide
5-(3-chloropyridin-2-yl)-1,2,3,4-tetrahydroisoquinoline
N-benzyl-3-{[ethyl(2-methylprop-2-en-1-yl)amino]methyl}-N-methylimidazo[1,2-a]pyridine-2-carboxamide
1-[5-(naphthalen-2-yl)-1,2,4-triazin-3-yl]-4-(pyrimidin-2-yl)-1,4-diazepane
N-[(3-methyl-1-benzofuran-2-yl)methyl]-2-(pyrrolidin-3-yl)benzamide
1-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}-3-(1-oxo-2,3-dihydro-1H-inden-5-yl)urea
(1S,5R)-6-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-(2-methoxyethyl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
6-(4-methoxy-2-methylbenzoyl)-2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]propanamide
4-[(1R,5S)-3,8-diazabicyclo[3.2.1]octane-8-carbonyl]-2,3,6-trimethylquinoline
1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N-{[4-(2-methylpropyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}-1-phenylcyclohexane-1-carboxamide
9-(5-ethyl-2-methylpyrimidin-4-yl)-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one