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4-(4-{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}piperazin-1-yl)quinazoline
(1R,5S,8S)-3-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-8-methoxy-3-azabicyclo[3.2.1]octane
1-{[(3-fluorophenyl)methyl]carbamoyl}-3-(3-methoxypropyl)piperidine-3-carboxylic acid
1-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-2-(5-methyl-1,2-oxazol-3-yl)piperidine
5-{[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
3-(4-chloro-2-methylbenzoyl)-1-(1,3-thiazole-5-carbonyl)piperidine
N-[2-(5-methylfuran-2-yl)ethyl]-6-oxo-1-(2-phenylethyl)piperidine-3-carboxamide
1-{[2-(3-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(piperidine-1-carbonyl)piperidine
N-{3-[2-(2-oxo-1,3-oxazolidin-3-yl)acetamido]phenyl}-3-phenylpropanamide
N-(2-methoxyethyl)-6-[2-(2-methoxyphenyl)pyrrolidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
N-[2-(3-fluorophenyl)ethyl]-6-phenylimidazo[2,1-b][1,3]thiazole-3-carboxamide
N-[(2R,3R)-1'-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]-2-(2-methoxyethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
3-[1-(1,4-dithiepan-6-yl)piperidin-4-yl]-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
1-{4-[(3-hydroxy-2,2-dimethylpropyl)amino]-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
5-cyclopropanecarbonyl-1'-[3-(methylsulfanyl)butyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-benzyl-3-({[2-(dimethyl-1,3-thiazol-2-yl)ethyl]amino}methyl)-N-methylimidazo[1,2-a]pyridine-2-carboxamide
2-(4-{[3-(naphthalen-1-yl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)pyrimidine
1-propyl-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}piperidin-4-amine
5-(oxolan-2-yl)-N-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)thiophene-2-carboxamide
(3S,4S)-1-(6-ethylpyrimidin-4-yl)-4-(naphthalen-2-yl)piperidin-3-ol
N-(1-ethyl-1H-1,2,3-triazol-4-yl)-4-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]piperazine-1-carboxamide
6-cyclobutyl-2-(4-{[(prop-2-en-1-yl)(pyridin-4-ylmethyl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
N-methyl-4-(4-{[3-(trifluoromethyl)phenyl]methyl}piperazine-1-carbonyl)pyridin-2-amine
2-[2-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1H-1,3-benzodiazole
1-[2-(2H-1,3-benzodioxol-5-ylmethyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-methyl-N-[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]piperidine-3-carboxamide
(1s,4s)-4-[1-(2H-1,3-benzodioxol-5-yl)-3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]cyclohexan-1-ol
N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)-5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carboxamide
(3aS,6aR)-5-[6-methyl-2-(propan-2-yl)pyrimidin-4-yl]-3-[2-(piperidin-1-yl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
4-[3-(1H-pyrazol-1-ylmethyl)benzoyl]-2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane
N-[(4-methoxynaphthalen-1-yl)methyl]-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-N-(propan-2-yl)propanamide
ethyl 2-[(3S,4R)-3-acetamido-4-(propan-2-yl)pyrrolidin-1-yl]-1,3-oxazole-4-carboxylate
6-[1-(dimethylamino)propan-2-yl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
N-[2-(cyclohex-1-en-1-yl)ethyl]-6-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-6-azaspiro[2.5]octane-1-carboxamide
N,5-dimethyl-N-(thiophen-3-ylmethyl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-2,4-dimethyl-1,3-thiazole-5-carboxamide
3-(2-aminoethyl)-4-[(1R)-1-(4-fluorophenyl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-(3-hydroxybenzoyl)pyrrolidine-3-carboxylic acid
5-ethoxy-N-(4-pentanamidophenyl)furan-2-carboxamide
8-(2-amino-2-methylpropanoyl)-2-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-3-one
methyl 5-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
2-ethoxy-4-[(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)methyl]phenol
3-fluoro-N-[1-(1-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]benzamide
3-{[3-(trifluoromethyl)-1,2,4-oxadiazol-5-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-methyl-3-phenyl-1-(5-propyl-1,2-oxazole-3-carbonyl)piperidine
2-[(4-chlorophenyl)methyl]-N-[(2S)-1-hydroxypropan-2-yl]benzamide
[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]({[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl})methylamine
N-(4-chloro-2-fluorophenyl)-2-{[2-(pyrrolidine-1-sulfonyl)ethyl]amino}acetamide
2-amino-6-cyclopropyl-4-[2-(2,2,2-trifluoroethoxy)pyridin-3-yl]pyridine-3-carbonitrile
4-{1-ethyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1,5-dimethyl-1H-pyrazole
3-({[(2-aminopyrimidin-5-yl)methyl](methyl)amino}methyl)-3-hydroxy-1-[(3-methoxyphenyl)methyl]piperidin-2-one