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2-benzyl-9-(6-methyl-4-oxo-4H-pyran-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
5-{[(2,1,3-benzoxadiazol-5-ylmethyl)(methyl)amino]methyl}-2-methoxybenzoic acid
1-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethan-1-one
(3R,5S)-1-[(3,4-dimethoxyphenyl)methyl]-N3-(4-fluorophenyl)-N5-[(2-methoxyphenyl)methyl]piperidine-3,5-dicarboxamide
N-{[7-chloro-2-(3-methylphenyl)quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]thiophene-2-carboxamide
N-({4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-3-(3,5-dimethyl-1H-pyrazol-1-yl)benzamide
3-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-{[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1,4-diazepane-1-carbaldehyde
2-{1-[1-(propan-2-yl)piperidin-4-yl]-4-(quinolin-8-ylmethyl)piperazin-2-yl}ethan-1-ol
1-(3-methoxyphenyl)-3-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]urea
2-butyl-8-(2-hydroxypyridine-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
(1-{[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}piperidin-3-yl)methanol
(3S,5R)-1-(5-methylthiophene-3-carbonyl)-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxylic acid
2-[(4aR,6R,8aS)-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinolin-2-yl]pyridine-4-carbonitrile
(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)({[7-(methylsulfanyl)-2-(thiophen-2-yl)quinolin-3-yl]methyl})amine
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-[1-(3-methylpyridin-2-yl)propan-2-yl]acetamide
5-(morpholine-4-carbonyl)-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
3-{5-[(2,5-dimethylphenyl)methyl]-1,2,4-oxadiazol-3-yl}pyridazine
1-benzyl-3-(2-methylphenyl)-3-{2-oxo-2-[4-(propan-2-yl)piperazin-1-yl]ethyl}pyrrolidine-2,5-dione
1-[(3S,4R)-1-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxy-N-[3-(2-methyl-1H-imidazol-1-yl)propyl]benzamide
2-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-3-methylpyridine
1-{2-[2-(aminomethyl)piperidin-1-yl]-2-oxoethyl}-3-methoxy-1,2-dihydropyridin-2-one
3-(3-fluorophenyl)-4-[2-(2-phenyl-1H-imidazol-1-yl)acetyl]piperazin-2-one
7-(4-methylpyrimidine-5-carbonyl)-1-oxa-7-azaspiro[3.5]nonane
methyl 4-({4-[(3,5-dimethylphenyl)methyl]-3-oxopiperazin-1-yl}methyl)-1H-pyrazole-3-carboxylate
2-(cyclopropylmethyl)-9-(3-hydroxy-4-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
5-{[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1-(2-methoxyethyl)-1H-imidazole
2-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-ethyl-N-methylacetamide
N2-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}pyrrolidine-1,2-dicarboxamide
N-[2-(2,5-dimethylphenoxy)ethyl]-N-methyl-2-[(4S)-2-oxo-4-(propan-2-yl)-1,3-oxazolidin-3-yl]acetamide
1-(2-methoxyphenyl)-4-[2-(3-methoxyphenyl)azetidine-1-carbonyl]-1H-pyrazole
1-(1,3-diethyl-6-methyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)-3-(1-hydroxy-3-methylbutan-2-yl)urea
[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]({[4-(methylsulfanyl)phenyl]methyl})propylamine
4-(4-methylpyridin-3-yl)-1H-indole
(4aR,8aR)-2-cyclobutanecarbonyl-7-[(3,4-dichlorophenyl)methyl]-decahydro-2,7-naphthyridin-4a-ol
N-benzyl-1-(2-cyclohexylethyl)-N-[(4-methyl-1,3-thiazol-5-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
5-benzyl-1-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-4-phenyl-1H-imidazole
1-{3-[2-methyl-6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}pentan-1-one
1-cyclopentyl-5-{4-[(3-methoxyphenyl)methyl]piperazine-1-carbonyl}piperidin-2-one
N-[(2-aminopyrimidin-5-yl)methyl]-2-(3-fluorophenoxymethyl)-N-methyl-1,3-oxazole-4-carboxamide
N-methyl-N-{2-phenyl-1-[1-(thiolan-3-yl)piperidin-4-yl]ethyl}thiophene-2-carboxamide
1-(furan-2-yl)-2-[3-(1-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]ethane-1,2-dione
N,N-dimethyl-2-(1-phenyl-1H-pyrazol-4-yl)quinoline-4-carboxamide
3-(quinolin-6-ylmethyl)-3H,4H-thieno[2,3-d]pyrimidin-4-one
N-methyl-N-{[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}thian-4-amine
1-(azocan-1-yl)-3-[2-methoxy-5-({[2-(pyrazin-2-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
N-(9H-fluoren-9-yl)-4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carboxamide
3-(2-fluorophenyl)-1-{3-[4-(hydroxymethyl)piperidin-1-yl]piperidin-1-yl}propan-1-one
1-[3-(dimethylamino)propyl]-3-(2-ethoxyethyl)-2-oxo-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid