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4-hydroxy-2-(3-methylphenyl)-N-{1-oxaspiro[4.4]nonan-3-yl}pyrimidine-5-carboxamide
1-(1,5,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-methyl-4-{5-[1-(thiophen-3-ylmethyl)-1H-imidazol-2-yl]thiophen-2-yl}but-3-yn-2-ol
1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-N-(prop-2-en-1-yl)piperidine-3-carboxamide
1-cyclopropyl-6-oxo-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]piperidine-3-carboxamide
1-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methoxyethan-1-one
2-({2-[5-(1H-pyrazol-3-yl)thiophen-2-yl]-1H-imidazol-1-yl}methyl)pyridine
3-{4-[(3-methylpyridin-2-yl)methyl]piperazine-1-carbonyl}-4,5,6,7-tetrahydro-1-benzofuran-4-one
5,6-dimethyl-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]thieno[2,3-d]pyrimidin-4-amine
6-methoxy-3-({2-[5-(propan-2-yl)-1,2-oxazol-3-yl]pyrrolidin-1-yl}methyl)-1,2-dihydroquinolin-2-one
2-methyl-1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-4-(2-methylphenyl)piperazine
[(3,5-dimethyl-1-benzofuran-2-yl)methyl](methyl)[1-(pyrazin-2-yl)propan-2-yl]amine
N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)-5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carboxamide
3-{[(9H-fluoren-9-yl)amino]methyl}pyrrolidin-3-ol
3-(cyclopropylmethyl)-1-(2-methoxy-6-methylphenyl)-3-(2-methoxyethyl)urea
9-[1-(hydroxymethyl)cyclopropanecarbonyl]-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-[2-(piperidine-1-carbonyl)phenoxy]piperidine
2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-[2-(3-methoxyphenyl)ethyl]acetamide
4-(4-methyl-1,3-thiazole-5-carbonyl)-2-{[3-(trifluoromethyl)phenyl]methyl}morpholine
(2S)-1-{6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carbonyl}pyrrolidine-2-carboxamide
2-(cyclopropylmethyl)-9-(5-fluoro-2-methoxybenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
5-(4-methoxy-3,5-dimethylphenyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
2-methoxy-N-[1-(1-{spiro[2.3]hexane-1-carbonyl}piperidin-4-yl)-1H-pyrazol-5-yl]benzamide
5-[4-(benzyloxy)piperidine-1-carbonyl]-1-[2-(morpholin-4-yl)ethyl]piperidin-2-one
1-[2-(3-benzyl-1,2,4-oxadiazol-5-yl)ethyl]-3-(1-ethyl-1H-1,2,3-triazol-4-yl)urea
methyl 5-{[(2-chloro-6-fluorophenyl)methyl]amino}-3-(furan-3-amido)-1-(2-methylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-{1-[(2,6-difluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-2-methyl-4-(2-methylphenyl)piperazine
(2S,4S,5R)-4-[(2-carboxyethyl)carbamoyl]-1,2-dimethyl-5-(2-methylphenyl)pyrrolidine-2-carboxylic acid
1-[2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]-1,4-diazepan-5-one
N-(7-{2-azabicyclo[2.2.1]heptane-2-carbonyl}-1-ethyl-2-(2-fluorophenyl)-1H-1,3-benzodiazol-5-yl)acetamide
N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-9H-purin-6-amine
1-[3-(3-methyl-2,5-dioxoimidazolidin-1-yl)phenyl]-3-{2-[(trifluoromethyl)sulfanyl]ethyl}urea
(2S,4R)-4-amino-N,N-diethyl-1-{[1-(propan-2-yl)-1H-1,3-benzodiazol-2-yl]methyl}pyrrolidine-2-carboxamide
1-(2,2-dimethylpropyl)-4'-[2-(ethylsulfanyl)ethyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-{4-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]-N-{2-[4-(trifluoromethyl)phenyl]ethyl}propanamide
(1R,5S)-6-methyl-7-oxo-N-[1-(thiophen-2-ylmethyl)-1H-pyrazol-5-yl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
1-(2,3-dimethylphenyl)-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}piperidin-4-amine
6-methyl-2-{[2-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)ethyl]amino}-3,4-dihydropyrimidin-4-one
1-[2-(6-chloro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-3-(3-methyl-1H-pyrazol-1-yl)propan-1-one
3-[(3R,4S)-3-(2-methyl-1,3-thiazole-4-amido)-4-(propan-2-yl)pyrrolidin-1-yl]propanoic acid
2-{[methyl({[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl})amino]methyl}quinolin-8-ol
3-(1,2-oxazinan-2-yl)-1-[4-(oxolane-2-carbonyl)piperazin-1-yl]propan-1-one
N-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]quinoline-2-carboxamide
1-methyl-N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
N-[1-(1H-indol-2-yl)ethyl]-N,1-dimethyl-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
N,6-dimethyl-N-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}imidazo[1,2-a]pyridine-2-carboxamide
1-{3-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]phenyl}ethan-1-one
6-{4-[1-(2-phenylethyl)pyrrolidin-3-yl]piperidine-1-carbonyl}-2,3-dihydropyridazin-3-one
4-(1-ethyl-1H-imidazol-2-yl)-1-[3-(3-methylphenyl)-1H-pyrazole-4-carbonyl]piperidine