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(1R,5R)-6-(cyclopropylmethyl)-3-(5-methyl-1,3,4-oxadiazol-2-yl)-3,6-diazabicyclo[3.2.2]nonane
2-{2-[1-(methoxymethyl)cyclobutanecarbonyl]-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-1-yl}pyridine
methyl (1R,3S,3aR,6aS)-5-ethyl-1-[(4-hydroxyphenyl)methyl]-3-(1H-imidazol-2-yl)-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
5-({1-[methyl(pyridin-3-ylmethyl)amino]hex-5-en-2-yl}oxy)pyridine-2-carbonitrile
5,7-dimethyl-N-{[1-(morpholin-4-yl)cyclopentyl]methyl}pyrido[2,3-d]pyrimidin-4-amine
(3R,4S)-4-({[7-methoxy-2-(thiophen-2-yl)quinolin-3-yl]methyl}(methyl)amino)oxolan-3-ol
4-(1-{[5-(3,4,5-trimethoxyphenyl)-1,2,4-triazin-3-yl]amino}ethyl)hepta-1,6-dien-4-ol
(1S,5R)-3-(1H-1,3-benzodiazole-5-carbonyl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
[(2S,6S)-4-(2-fluoro-4-methylbenzoyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
(2,1,3-benzothiadiazol-5-ylmethyl)(methyl){[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}amine
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-2-[4-(propane-1-sulfonyl)morpholin-3-yl]acetamide
2-(dimethyl-1,3-thiazol-5-yl)-N-[2-(pyridin-3-ylformamido)ethyl]acetamide
N-[(3-methoxyphenyl)methyl]-3-[1-(3-phenoxypropanoyl)piperidin-3-yl]propanamide
N-[(1-cyclopropanecarbonylpiperidin-3-yl)methyl]-6-methylpyridine-3-carboxamide
1-[4-(4-methylphenoxy)piperidin-1-yl]-2-(morpholin-4-yl)ethan-1-one
5-(3-methylfuran-2-carbonyl)-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
(1S,5R)-3-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-({4-phenyl-5-[5-(1H-pyrazol-5-yl)furan-2-yl]-1H-imidazol-1-yl}methyl)piperidine
4-[1-({1-[4-(propan-2-yl)phenyl]-1H-pyrazol-4-yl}methyl)piperidin-4-yl]pyrimidin-2-amine
3-ethyl-4-methyl-N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]-1H-pyrazole-5-carboxamide
3-[(oxan-3-yl)sulfamoyl]-N-[2-(1H-pyrazol-1-yl)ethyl]benzamide
N-ethyl-N-[(3S,4R)-4-hydroxyoxolan-3-yl]-3,5,7-trimethyl-1H-indole-2-carboxamide
N4-[(5-ethylpyridin-2-yl)methyl]-N4,5-dimethylpyrimidine-2,4-diamine
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
N-cyclopropyl-4-hydroxy-2-(2-methyl-1,3-thiazol-4-yl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]pyrimidine-5-carboxamide
N-[1-(2-methanesulfonylethyl)piperidin-4-yl]-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
1-(4-fluorophenyl)-6,6-dimethyl-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
N-(6-cyanopyridin-3-yl)-4-(pyrimidin-2-yloxy)piperidine-1-carboxamide
3-(2,2-dimethyloxan-4-yl)-3-ethyl-1-[3-(2-methoxyethoxy)phenyl]urea
N-phenyl-1-(2,4,5-trimethylbenzoyl)piperidin-3-amine
1-(4-methylphenyl)-3-{[1-(pyridin-4-ylmethyl)piperidin-3-yl]methyl}urea
2-[(4-{5-[(cyclohexylmethyl)sulfanyl]-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]-6-methylpyridine
1-(1-{1-butyl-3-[(4-methoxyphenyl)methyl]-1H-1,2,4-triazol-5-yl}ethyl)-4-methylpiperazine
5-methyl-4-(1-methyl-1H-pyrazol-5-yl)-2-(4-phenylpiperidin-1-yl)pyrimidine
N-propyl-N-(pyridin-4-ylmethyl)pyridine-3-carboxamide
2-{4-[2-(oxolan-3-yl)-1H-imidazol-1-yl]phenyl}-1H-1,3-benzodiazole
2-chloro-N-({1-[2-(pyrrolidin-1-yl)benzoyl]piperidin-3-yl}methyl)benzamide
N3-[1-(2-chlorophenyl)ethyl]-N5-methyl-4-oxo-1-(3-phenylpropyl)-1,4-dihydropyridine-3,5-dicarboxamide
4-benzyl-3-{1-[(2-methyl-1,3-oxazol-4-yl)methyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
2-{[6-amino-2-(butylsulfanyl)pyrimidin-4-yl](methyl)amino}ethan-1-ol
2-{2-[2-(2,4-dimethoxyphenyl)-1H-imidazol-1-yl]ethyl}pyridine
ethyl 1-(cyclopropylmethyl)-5-[(4-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
methyl (1R,3S,3aR,6aS)-1-benzyl-5-methyl-4,6-dioxo-3-(pyridin-3-yl)-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
(3aR,6aR)-2-[2-(4-chlorophenyl)acetyl]-5-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[2-(dimethylamino)ethyl]-3-(3-hydroxy-3-methylbutyl)-N-methylbenzamide
N-{[2-cyclopropylmethanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}-N,1-dimethylpiperidin-4-amine
N-[(3-chlorophenyl)methyl]-3-{1-[2-(methylsulfanyl)acetyl]piperidin-4-yl}propanamide
1-{[3-(2-hydroxyethyl)-4-(3-methylbut-2-en-1-yl)piperazin-1-yl]methyl}naphthalen-2-ol
N-{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}-2,3-dihydro-1H-inden-1-amine
2-ethyl-N-[(5-methylfuran-2-yl)methyl]pyrimidine-5-carboxamide