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1-[4-(4-fluorophenyl)benzoyl]-4-[(4-methoxyphenyl)methyl]-1,4-diazepan-5-one
3-methyl-3-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}-1-[3-(sulfamoylmethyl)phenyl]urea
3-[(cycloheptylamino)methyl]-5,6,7-trimethoxy-N,N-dimethylquinolin-2-amine
N-[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1-methyl-1H-pyrazole-5-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-cyclopropyl-N'-(3,5-dimethylphenyl)propanediamide
6-{[benzyl(butyl)amino]methyl}-N-{[1-(morpholin-4-yl)cyclohexyl]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
N-{[7-(3,5-dimethylbenzoyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}oxolane-3-carboxamide
2-(1H-imidazol-1-yl)-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)acetamide
N-[1-(4-fluorophenyl)-2-hydroxyethyl]-2-(1-propylpiperidin-4-yl)acetamide
4-{3-[(4-fluorophenyl)methoxy]azetidine-1-carbonyl}-2-(thiophen-2-yl)-1,3-thiazole
[(3R,4R)-1-(5-chloro-3-fluoropyridin-2-yl)-4-[(4-ethylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
methyl (2S,4S)-1-[(4-methoxy-2,5-dimethylphenyl)methyl]-4-(quinoline-2-amido)pyrrolidine-2-carboxylate
{1-[(1-cycloheptanecarbonylpiperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}methanol
3-[2-(pyrrolidine-1-sulfonyl)ethyl]-1-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
6-[3-hydroxy-2-(thiophen-2-ylmethyl)propyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
2-{[(2S)-2-amino-4-(methylsulfanyl)butanamido]methyl}-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
2-{methyl[2-(1H-pyrazol-4-yl)ethyl]amino}-N-(pyrazin-2-yl)acetamide
2-[2-(dimethylamino)ethyl]-8-[5-(propan-2-yl)pyrimidin-4-yl]-2,8-diazaspiro[5.5]undecan-3-one
(3aS,6aS)-5-[(1-ethyl-1H-indol-6-yl)methyl]-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[5-(5-methyl-1,2-oxazol-4-yl)-3-(2-phenylethyl)-1H-1,2,4-triazol-1-yl]pyridine
4-(5-chloro-2-hydroxybenzoyl)-1-(2-methylphenyl)piperazin-2-one
6-{3-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-3-oxopropyl}-2,3-dihydropyridazin-3-one
ethyl 4-[(4-methoxyphenyl)methyl]piperidine-4-carboxylate
7-fluoro-4-[3-(2-methylphenoxy)azetidine-1-carbonyl]-1,2-dihydroquinolin-2-one
(2S,4R)-4-amino-N-methyl-1-[3-(trimethyl-1H-pyrazol-1-yl)propanoyl]pyrrolidine-2-carboxamide
4-[7-(5-chlorothiophene-2-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]morpholine
(3S,4R)-4-(3-methoxyphenyl)-1-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]pyrrolidine-3-carboxylic acid
4-(1H-1,3-benzodiazol-1-yl)-1-(2-methylpyrimidin-4-yl)piperidine-4-carboxylic acid
(4aS,7aR)-1-[(3-fluoro-2,4-dimethylphenyl)methyl]-4-(1H-imidazol-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{3-[3-(1H-1,3-benzodiazol-5-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}ethan-1-one
N,N-diethyl-5-methyl-3-(2-methylcyclohexyl)-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
1-[1-(5-chloropyridine-3-carbonyl)piperidin-4-yl]-3-phenylpropan-1-ol
(4-benzyl-1-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)-5-fluorophenyl]methyl}piperidin-4-yl)methanol
4-[(dimethylamino)methyl]-N-(2-hydroxy-2-phenylethyl)benzamide
2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)-1-[4-(5-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]ethan-1-one
3-(3-fluorophenyl)-4-[2-(propan-2-yl)-1,3-benzoxazole-5-carbonyl]piperazin-2-one
1-(cyclopropanesulfonyl)-N-[3-(4-fluorophenyl)phenyl]piperidine-3-carboxamide
[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]bis(1,3-oxazol-4-ylmethyl)amine
N-(1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-3-yl)-N-ethylacetamide
1-{[5-(morpholine-4-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}piperidin-3-ol
5-cyclopropanecarbonyl-1'-(2,3-difluorobenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-({4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridin-2-amine
2,5,7-trimethyl-4-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]quinoline
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-1-(pyrrolidin-1-yl)cyclopentane-1-carboxamide
N-[1-(1-{[3-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]-2-phenylacetamide
(1S,2R)-N1-[2-(1-ethyl-1H-1,3-benzodiazol-2-yl)ethyl]-N2-propylcyclohexane-1,2-dicarboxamide
N-[4-(3-methylphenyl)phenyl]-1-propylpiperidine-4-carboxamide
(2R,6S)-2,6-dimethyl-4-(5-{[4-(4-methyl-1,2,5-oxadiazol-3-yl)piperazin-1-yl]methyl}imidazo[2,1-b][1,3]thiazole-6-carbonyl)morpholine
N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-{methyl[(2-phenyl-1,3-thiazol-4-yl)methyl]amino}acetamide
ethyl 2-{1-[(4-methoxy-2-methylphenyl)carbamoyl]piperidin-2-yl}acetate