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3-{5-[(4-chlorophenyl)methyl]-1,3,4-thiadiazol-2-yl}-1-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]urea
(1R,5R)-6-(cyclopropylmethyl)-3-(4-fluorobenzenesulfonyl)-3,6-diazabicyclo[3.2.2]nonane
1-(2-chlorophenyl)-3-(ethoxymethyl)-5-(oxolan-3-yl)-1H-1,2,4-triazole
N-{2-[5-(2-chloro-3-hydroxy-4-methoxyphenyl)-4-phenyl-1H-imidazol-1-yl]ethyl}propanamide
1-[(5-phenylthiophen-2-yl)methyl]-3-(4H-1,2,4-triazol-3-yl)piperidine
2-{1-cyclopropyl-2,5-dioxo-3-[3-(trifluoromethyl)phenyl]pyrrolidin-3-yl}-N-methyl-N-(2-phenylethyl)acetamide
1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-4-(pyrrolidin-1-ylmethyl)piperidin-4-ol
2-(azepan-1-yl)-2-{1-[(4-methoxyphenyl)methyl]-1H-pyrazol-4-yl}acetic acid
2-[5-(4-methylquinolin-2-yl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
1-[(3,4-difluorophenyl)methyl]-3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
1-[2-(1H-imidazol-1-yl)ethyl]-4-phenyl-5-[5-(1H-pyrazol-5-yl)furan-2-yl]-1H-imidazole
4-{[3-(2-hydroxyethyl)-4-(3-methylbutyl)piperazin-1-yl]methyl}-2-methoxyphenol
5-(1-{[3-(benzyloxy)phenyl]methyl}piperidin-4-yl)-5-(3-methylbutyl)imidazolidine-2,4-dione
N-cyclopropyl-N-{[4-(methylsulfanyl)phenyl]methyl}-1-propanoylpyrrolidine-2-carboxamide
1-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]-4-(2-methyl-1H-imidazol-1-yl)butan-1-one
1-[5-(2,3-dihydro-1H-isoindole-2-carbonyl)-2-methylphenyl]imidazolidin-2-one
2-methyl-4-(thian-4-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-(3-acetylphenoxymethyl)-N-(3-hydroxy-2,2-dimethylpropyl)-1H-pyrazole-3-carboxamide
N-cycloheptyl-3-[(3S,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-(pyridin-4-ylmethyl)piperidin-3-yl]propanamide
2-(cyclohex-1-en-1-yl)-N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}acetamide
N-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)-3-(pyrazin-2-yl)propanamide
N-benzyl-5-[(3-ethoxypropyl)amino]-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[1-(4-fluorophenyl)propyl]-3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-4-[(2-methylpropanamido)methyl]benzamide
N,2-dimethyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-4-phenylpyrimidine-5-carboxamide
4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)-1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidine
1-(piperidin-1-yl)-3-[2-(thiomorpholin-4-ylmethyl)phenoxy]propan-2-ol
1-[(2,6-difluorophenyl)methyl]-3-(3-hydroxypropyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
4-(1-butyl-1H-imidazol-2-yl)-N-(2,5-dimethylphenyl)piperidine-1-carboxamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}benzamide
3-{2,3-dihydrospiro[indene-1,4'-piperidine]-1'-ylmethyl}-3-hydroxy-1-(2-methoxyethyl)piperidin-2-one
N,N-dimethyl-2-[(1S,5R)-6-[(6-methyl-4-oxo-1,4-dihydroquinolin-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
1-benzyl-4-(2-hydroxyacetyl)-1,4-diazepane-6-carboxylic acid
N-[1-(6-methoxynaphthalen-2-yl)ethyl]-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
1-ethyl-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-4-carboxamide
2-(morpholin-4-yl)-5-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)benzonitrile
N-ethyl-N-[(5-methylfuran-2-yl)methyl]-1-phenyl-1H-1,2,3-triazole-4-carboxamide
N-cyclopropyl-2-ethyl-N-{[2-(4-hydroxypiperidin-1-yl)-8-methylquinolin-3-yl]methyl}butanamide
N-{[2-(morpholin-4-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]oxolane-2-carboxamide
5-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-2-(pyridin-4-yl)pyrimidin-4-ol
N-[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl]-2-methyl-6-(1-methylpiperidin-3-yl)pyrimidin-4-amine
1-(4-methoxyphenyl)-N-[1-(pyrimidin-2-yl)piperidin-3-yl]cyclopropane-1-carboxamide
2-cyclopropyl-N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-4-methylpyrimidine-5-carboxamide
4-{[(2,3-dihydro-1H-inden-2-yl)(methyl)amino]methyl}benzonitrile
1-(3,5-dimethyladamantane-1-carbonyl)azetidin-3-ol
2-{3-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propane-1,3-diol
1-[(2,2-dimethyloxan-4-yl)methyl]-4-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]piperazine
3-({[(2-phenoxypyridin-3-yl)methyl]carbamoyl}methyl)-1,2,3-oxadiazol-3-ium-5-olate
3-{[(3R,4S)-1-acetyl-4-propylpyrrolidin-3-yl]sulfamoyl}benzoic acid
2-(3-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}phenoxy)acetamide