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N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-(4-methyl-1,4-diazepan-1-yl)acetamide
N-methyl-N-[2-(2-methyl-1H-indol-1-yl)ethyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
5-{2-[2-(3,4-dichlorophenyl)morpholin-4-yl]-2-oxoethyl}-2-methyl-3,4-dihydropyrimidin-4-one
7-(3-chlorophenyl)-4-(piperidin-4-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-[1-(1H-indole-5-carbonyl)piperidin-3-yl]-N-[(5-methylfuran-2-yl)methyl]propanamide
3-(cyclopropylmethyl)-1-[2-(3-oxo-2,3-dihydro-1H-indazol-2-yl)acetyl]piperidine-3-carboxylic acid
1-{[3-(3-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-(pyridin-3-yl)piperidin-4-ol
3-butyl-1-methyl-4-(2,3,6-trimethylquinoline-4-carbonyl)piperazin-2-one
2-({4-[(2-cyanophenyl)methyl]piperazin-1-yl}methyl)pyridine-3-carboxylic acid
3-{2-[2-(2-methoxyphenyl)-1H-imidazol-1-yl]ethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[N-(3-methylphenyl)methanesulfonamido]-N-[3-(pyridin-3-yl)propyl]acetamide
[(4-{[1-(furan-2-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl](methyl)(naphthalen-1-ylmethyl)amine
2-({[(3R,4R)-4-(hydroxymethyl)-1-(7-methyl-1-benzofuran-2-carbonyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
N-ethyl-1-[(6-fluoroquinolin-2-yl)methyl]-N-(pyridin-4-ylmethyl)piperidin-3-amine
5-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1H,5H,6H,7H,8H-pyrido[3,2-f]indazol-7-one
4-[4-(3-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-6-methylpyrimidin-2-amine
6-({methyl[(5-methylfuran-2-yl)methyl]amino}methyl)-2-oxo-N-(quinolin-3-ylmethyl)-1,2-dihydropyridine-3-carboxamide
7-[(2,3-difluorophenyl)methyl]-2-(5-methyl-1H-pyrazole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl](methyl){[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}amine
N-[1-(cyclohexylmethyl)piperidin-3-yl]-3-methylbenzamide
3-{[1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1,2-dihydroquinolin-2-one
3-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-ylmethyl]benzonitrile
1-[(4-methoxyphenyl)methyl]-N-methyl-N-[4-(morpholin-4-yl)butyl]-1H-1,2,3-triazole-4-carboxamide
N-{[1-(morpholin-4-yl)cyclohexyl]methyl}-2,3-dihydro-1H-indene-1-carboxamide
1-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
N-ethyl-5-(1H-indol-1-ylmethyl)-N-(oxolan-2-ylmethyl)-1H-pyrazole-3-carboxamide
1-ethyl-4,6-dimethyl-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
N-(1H-1,2,3,4-tetrazol-5-ylmethyl)-5-[1-(3,3,3-trifluoropropyl)pyrrolidin-2-yl]thiophene-2-carboxamide
4-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-N,6-dimethylpyrimidin-2-amine
2-[1-(1-tert-butyl-1H-pyrrole-3-carbonyl)piperidin-4-yl]-4-methyl-1H-1,3-benzodiazole
[(3-methylthiophen-2-yl)methyl](oxolan-3-ylmethyl)(pyridin-2-ylmethyl)amine
2-chloro-N-{1-[1-(quinolin-4-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
N-[1-({[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl](methyl)carbamoyl}methyl)-1H-pyrazol-4-yl]-3-(2-methoxyphenyl)propanamide
8-methoxy-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-2-(pyridin-4-yl)quinoline-4-carboxamide
1-[(2-chloro-4-ethoxy-5-methoxyphenyl)methyl]piperidine-3-carbonitrile
5-methoxy-1,2-dimethyl-N-[(1-methylpiperidin-3-yl)methyl]-1H-indole-3-carboxamide
1-[1-(2-methylpropyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
3-cyano-N-{1-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}benzamide
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-6-methylpyridine-2-carboxamide
(4aS,7aR)-1-(1-ethyl-1H-pyrazole-3-carbonyl)-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidine-1-carbonyl]-N,N-dimethylpiperidine-1-carboxamide
N,5-dimethyl-N-[1-(2-phenylethyl)piperidin-3-yl]imidazo[1,2-a]pyridine-2-carboxamide
N-[(5-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]acetamide
{3-ethyl-1-[4-(morpholine-4-carbonyl)pyridin-2-yl]piperidin-3-yl}methanol
N-{[1-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetyl)piperidin-3-yl]methyl}naphthalene-1-carboxamide
3-methyl-N-(1-{1-[(4-phenylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)butanamide
2-methyl-6-{[3-(pyrrolidin-1-yl)pyrrolidin-1-yl]methyl}pyridine
3-(1-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-yl)-N-(2-methoxyethyl)propanamide
methyl 1-{[6-(azocane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}piperidine-2-carboxylate