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3-{2-[4-(3-chlorophenoxy)piperidin-1-yl]-2-oxoethyl}-3-(3-fluorophenyl)-1-methylpyrrolidine-2,5-dione
1-(6-fluoro-4-methylquinazolin-2-yl)-N-[(2-fluorophenyl)methyl]azepan-4-amine
5-ethyl-3-(2-methylprop-2-en-1-yl)-5-{1-[(3-phenyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
1-({[2-(4,6-dimethylpyrimidin-2-yl)ethyl]carbamoyl}methyl)piperidine-4-carboxamide
(1-{2-[(6-ethyl-4-methylquinolin-2-yl)amino]ethyl}piperidin-3-yl)methanol
N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-6-{methyl[(3-methylpyridin-2-yl)methyl]amino}pyridine-3-carboxamide
5-methyl-N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
[(1-methyl-1H-imidazol-2-yl)methyl]({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)(oxolan-2-ylmethyl)amine
1-[4-(cyclopropylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]-3-methylbutan-1-ol
N-[(5-phenyl-4H-1,2,4-triazol-3-yl)methyl]-3-(2-phenylethyl)-1,2-oxazole-5-carboxamide
1-methyl-N-{[5-(methylcarbamoyl)furan-2-yl]methyl}-3-propyl-1H-pyrazole-5-carboxamide
N-cyclopropyl-3-[3-(1H-pyrazol-3-yl)phenyl]benzamide
2-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]amino}-N-[2-methyl-6-(propan-2-yl)phenyl]acetamide
4-(1H-imidazole-2-carbonyl)-1-[(4-methoxyphenyl)methyl]piperazin-2-one
3-fluoro-5-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
2-[3-(5-fluoro-2-methylphenyl)phenyl]ethan-1-amine
N-(1H-1,2,3-benzotriazol-5-yl)-4-(2-methoxyphenyl)-2-methylpiperazine-1-carboxamide
N-(oxolan-2-ylmethyl)-N-({4-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)pyridine-4-carboxamide
2-ethyl-4-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyridine
2-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-5-methylpyrazine
2-[2-(dimethylamino)ethyl]-9-(quinolin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-(4-chlorophenyl)-7-[(dimethylsulfamoyl)amino]-1,2,3,4-tetrahydroquinolin-2-one
N-methyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)pyridazine-3-carboxamide
(4aS,7aR)-1-(4-methoxy-2-methylbenzoyl)-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-benzyl-7-(3-chlorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
methyl 9-(2,3-dihydro-1H-inden-2-yloxy)-3-(3-fluorobenzoyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2-(methylsulfanyl)-1,3-thiazole-4-carboxamide
N-cyclopropyl-3-methyl-4-oxo-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-3,4-dihydroquinazoline-7-carboxamide
3-[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-[3-(oxolan-2-yl)propyl]propanamide
N-[2-(4-fluorophenyl)ethyl]-N-{[1-(2-hydroxyethyl)-1,2,5,6-tetrahydropyridin-3-yl]methyl}acetamide
N-(2,5-dimethoxyphenyl)-2-[2-(dimethylamino)ethyl]morpholine-4-carboxamide
2-cyclopropyl-8-{[2-(propylamino)pyrimidin-5-yl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}-N-(2,2,2-trifluoroethyl)piperidine-4-carboxamide
4-ethyl-2-methyl-N-[phenyl(pyridin-4-yl)methyl]-1,3-thiazole-5-carboxamide
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}(oxolan-2-ylmethyl)[(3-phenyl-1H-pyrazol-4-yl)methyl]amine
1-{3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}-3-(1H-pyrazol-1-yl)propan-1-one
N-[3-(4-fluorophenyl)phenyl]-1-[(4-methyl-1H-imidazol-5-yl)methyl]pyrrolidine-2-carboxamide
1-[6-(3-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-1,4-diazepan-5-one
N-ethyl-4-methyl-5-[2-(3-methyl-1H-1,2,4-triazol-5-yl)pyrrolidine-1-carbonyl]-1,3-thiazol-2-amine
8-[2-(benzyloxy)acetyl]-2-cyclopropyl-2,8-diazaspiro[5.5]undecan-3-one
2-[3-(pyridin-2-yl)azetidin-1-yl]-3-(pyrrolidin-1-yl)pyrazine
1-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidin-1-yl]-2-(1-methyl-1H-indol-3-yl)ethan-1-one
N-[3-(1,3-benzoxazol-2-yl)propyl]-2-(dimethylamino)-2-(4-fluorophenyl)acetamide
1-methyl-2-(5-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)-1H-1,3-benzodiazole
3-(1-{[2-(2-phenylethynyl)phenyl]methyl}piperidin-4-yl)-1-(pyrrolidin-1-yl)propan-1-one
N-{[5-(2-chlorophenyl)furan-2-yl]methyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
(1S,5R)-6-(4-methylpyridine-3-carbonyl)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
3-(3-fluorophenyl)-N-(oxolan-2-ylmethyl)-N-{[4-(pyridin-3-ylmethoxy)phenyl]methyl}benzamide
2-[1-benzyl-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]acetamide
2-[4-(quinolin-2-ylmethyl)piperazin-1-yl]pyridine-4-carboxamide