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1-[3-({[(5-methylthiophen-2-yl)methyl]amino}methyl)phenoxy]-3-(morpholin-4-yl)propan-2-ol
N-[2-(4-chlorophenyl)ethyl]-1-ethyl-N-(pyridin-4-ylmethyl)-1H-pyrazole-3-carboxamide
(1R,5R)-N,N-dimethyl-6-{[3-(4-methylphenyl)-1,2-oxazol-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-{[5-methyl-7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}furan-2-carboxamide
8-[(3-chloro-2-methylphenyl)carbamoyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)-3-(1-methyl-1H-pyrazol-4-yl)propanamide
2-amino-4-(2,3-dimethyl-1H-indol-7-yl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-(4-fluorophenoxymethyl)piperidine
5-cyclobutanecarbonyl-1'-[(2-methylphenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-3-(piperidine-1-carbonyl)pyrazine-2-carboxamide
2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}acetamide
5-ethyl-2-methyl-4-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}pyrimidine
(2R,3S,6R)-3-(2,3-difluorophenyl)-5-(1H-pyrazole-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-{2-[4-(4-methylpiperazine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}-2-(trifluoromethyl)benzamide
N-({1-[(2-aminopyridin-3-yl)methyl]piperidin-3-yl}methyl)thiophene-2-sulfonamide
3-{5-[(2-methyl-1,3-oxazol-4-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
3-methyl-5-{2-oxo-2-[4-(pyridin-4-yl)piperidin-1-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
5-[1-(2-hydroxybutyl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]-1,2-dihydropyridin-2-one
5-methoxy-2-({9-[(1-methylpiperidin-3-yl)methoxy]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}methyl)phenol
N-[(3R,4R)-3-hydroxy-1-[2-(3-methoxyphenoxy)ethyl]piperidin-4-yl]pyridine-2-carboxamide
3-{1-[2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)acetyl]piperidin-3-yl}benzoic acid
4-ethyl-3-{1-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(2-hydroxyethyl)-4-(4-methoxy-3,5-dimethylbenzoyl)piperazin-2-one
4-{[3-(3-phenoxyazetidine-1-carbonyl)-1,2-oxazol-5-yl]methyl}morpholine
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonan-7-yl]ethan-1-one
N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)acetamide
3-methyl-7-[4-(1H-pyrazol-3-yl)benzoyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-[2-(1H-imidazol-4-yl)ethyl]-4-{[(4-methylphenyl)amino]methyl}benzamide
2-(2,6-dimethoxypyridin-3-yl)-2-[methyl(quinolin-8-ylmethyl)amino]acetic acid
3-(morpholine-4-carbonyl)-N,N,1-tris(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-{[4-(2-methylphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-2-phenylacetamide
4-{4-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperazin-1-yl}butan-1-ol
4-[3-(2-methoxyethyl)piperidin-1-yl]-N,N,6-trimethylpyrimidin-2-amine
N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
4-{3-[(1R,5S,6S)-6-[(dimethylamino)methyl]-3-azabicyclo[3.1.0]hexane-3-carbonyl]phenyl}-2-methylbutan-2-ol
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-N-[(1S,2S)-1-amino-2,3-dihydro-1H-inden-2-yl]propanamide
methyl 2-[({1-[(2,3-difluorophenyl)methyl]-3-hydroxy-2-oxopiperidin-3-yl}methyl)amino]acetate
2-ethoxy-4-(1-methyl-4-phenyl-1H-imidazol-5-yl)phenol
8-{2-[(2R,6S)-2,6-dimethylpiperidin-1-yl]acetyl}-2-(3-methylbutyl)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
2-[(4-chlorophenyl)methyl]-8-[(5-methylfuran-2-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
3-(3-fluorophenyl)-N-[(3R,4R)-4-(4-methylpiperazin-1-yl)oxolan-3-yl]-1H-pyrazole-4-carboxamide
2-(4-chlorophenyl)-5-{1-[2-(4H-1,2,4-triazol-4-yl)ethyl]-1H-imidazol-2-yl}pyrimidine
4-(azepan-1-yl)-5-methyl-N-(pyridin-4-ylmethyl)thieno[2,3-d]pyrimidine-6-carboxamide
1-[(1S,5R)-3-methyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-[3-(trifluoromethyl)phenyl]ethan-1-one
3-{5-[(4-phenylphenyl)methyl]-1,3,4-oxadiazol-2-yl}-N-(pyridin-2-ylmethyl)propanamide
3-{5-[({1-[(2-fluorophenyl)methyl]piperidin-3-yl}amino)methyl]thiophen-3-yl}prop-2-yn-1-ol
methyl({[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl})(pyrimidin-4-ylmethyl)amine
1-[(4aR,8aS)-1-(5-methyl-1,3-diphenyl-1H-pyrazole-4-carbonyl)-decahydro-1,6-naphthyridin-6-yl]-2-methoxyethan-1-one
4-ethyl-5-methyl-6-[4-(pyrrolidine-1-sulfonyl)-1,4-diazepan-1-yl]pyrimidin-2-amine
N-[2-(dimethylamino)ethyl]-3-(3-methyl-1H-pyrazol-1-yl)-N-{[8-methyl-2-(3-methylphenyl)quinolin-3-yl]methyl}propanamide