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1-(3-methyl-1H-pyrazole-5-carbonyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
1-(dimethylamino)-2-(4-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)propan-2-ol
4-[(1E)-1-phenylprop-1-en-2-yl]-3-(pyridin-3-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
[3-(4-methyl-1,3-thiazol-5-yl)propyl]({[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl})amine
4-ethyl-3-[1-(1-ethyl-3,5-dimethyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(3-methoxybenzoyl)-4-(2-methylpyridin-4-yl)piperazine
1-[4-({3-[2-hydroxy-3-(piperidin-1-yl)propoxy]-4-methoxyphenyl}methyl)-1,4-diazepan-1-yl]ethan-1-one
4-[4-(2-chlorophenyl)-1H-1,2,3-triazol-1-yl]-1-(oxan-4-yl)piperidine
1-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}-3-[4-(trifluoromethyl)benzoyl]piperidine
1-[(3-{[1-(3-chlorobenzoyl)piperidin-4-yl]oxy}phenyl)methyl]-4-(pyridin-3-ylmethyl)piperazine
(2S,4R)-4-amino-N-ethyl-1-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)acetyl]pyrrolidine-2-carboxamide
3-(3-aminoazepan-1-yl)-1-(1,2,3,4-tetrahydroquinolin-1-yl)propan-1-one
5-{[3-(1-methylpiperidin-3-yl)propanamido]methyl}-1,2,4-oxadiazole-3-carboxamide
3-[(3R,4S)-1-(3,6-dimethylpyrazin-2-yl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
3-hydroxy-3-{[4-(hydroxymethyl)piperidin-1-yl]methyl}-1-[(3-methylphenyl)methyl]piperidin-2-one
4-methyl-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}piperidine-4-carboxamide
N-{1-[({2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethyl}carbamoyl)methyl]-1H-pyrazol-4-yl}thiophene-3-carboxamide
3-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidine-1-carbonyl]-2-methylpyridine
3-(2-ethyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-2-methyl-4-phenylpyridine
8-methoxy-5-(5-propylpyrimidin-2-yl)quinoline
N-(1-cyclopentyl-1H-pyrazol-5-yl)-3-cyclopropylpropanamide
1-methyl-5-{[(3-methyloxetan-3-yl)methyl]amino}-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
ethyl 4-[4-(2,2-dimethylpropyl)-3-(2-hydroxyethyl)piperazin-1-yl]piperidine-1-carboxylate
4-{2-[1-(2-aminopyridine-4-carbonyl)piperidin-2-yl]ethyl}phenol
3-[2-(3-methoxyphenyl)azetidin-1-yl]-N-(4-methylphenyl)-3-oxopropanamide
1-[(3-{[1-(naphthalene-1-sulfonyl)piperidin-4-yl]oxy}phenyl)methyl]-4-(pyridin-3-ylmethyl)piperazine
N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-1H-pyrazole-4-carboxamide
9-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
3-(5-tert-butyl-2-methoxyphenyl)-1-[3-(3-hydroxypiperidin-1-yl)propyl]urea
1-[2-(4-chlorophenyl)ethyl]-5-(1,4-oxazepane-4-carbonyl)piperidin-2-one
N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1-(thiophene-2-carbonyl)piperidine-2-carboxamide
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-3-(2-oxoimidazolidin-1-yl)benzamide
5-(2,6-dimethoxyphenyl)-3-methyl-1-phenyl-1H,4H-pyrazolo[3,4-d]imidazole
{[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}[2-(1H-imidazol-1-yl)ethyl]methylamine
3-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-6-(propan-2-yl)-1,2-dihydropyridin-2-one
2-(benzyloxy)-1-[(3R,5R)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidin-1-yl]ethan-1-one
2-(1H-imidazol-2-yl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]benzamide
N-[(2-ethoxyphenyl)methyl]-N-ethyl-2-(1H-1,2,4-triazol-1-yl)benzamide
2-{1-[(2-chloro-4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-ethyl-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
1-(2,2-dimethylpropyl)-4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
(1R,5R)-6-(cyclopropylmethyl)-3-[4-(morpholin-4-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
2-[(2-ethyl-6-methylpyridin-3-yl)oxy]-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]acetamide
(4aS,8aR)-1-(2-aminoethyl)-6-(2-fluorobenzoyl)-decahydro-1,6-naphthyridin-2-one
(2R,3R)-1'-(3-fluoropyridin-2-yl)-3-[(2-hydroxyethyl)(methyl)amino]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
3-{[(1R,3S,5S)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl]methyl}-7-(methylsulfanyl)-1,2-dihydroquinolin-2-one
8-[(2-ethyl-1,3-thiazol-4-yl)methyl]-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(3E)-N-[2-(dimethylamino)ethyl]-N-[(3-methylthiophen-2-yl)methyl]pent-3-enamide
1-(2,3-dihydro-1H-inden-2-yl)-4-[(furan-3-ylmethyl)amino]pyrrolidin-2-one
N-(3-methyl-1-phenyl-1H-pyrazol-5-yl)-2-(5-phenyl-2H-1,2,3,4-tetrazol-2-yl)acetamide
3-(2-methylpropyl)-1-phenyl-5-[3-(1H-1,2,4-triazol-1-yl)propyl]-1H-1,2,4-triazole