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3-[2-oxo-2-(piperidin-1-yl)ethyl]-4-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-one
2-(1-cyclopentyl-4-propylpiperazin-2-yl)ethan-1-ol
methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}amine
2-(4-{[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl}-1-(3-methylbut-2-en-1-yl)piperazin-2-yl)ethan-1-ol
2-[2-(butan-2-yl)phenoxy]-1-[4-(pyrrolidin-1-yl)piperidin-1-yl]ethan-1-one
2-[2-(4-methoxybenzoyl)-1H-imidazol-1-yl]-N-(4-methyl-1-propyl-1H-pyrazol-5-yl)acetamide
2-{3-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]phenoxy}acetamide
2-chloro-N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-5-(1H-pyrazol-1-yl)benzamide
3-{1-[(3-cyanophenyl)methyl]piperidin-4-yl}propanamide
(3E)-N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}pent-3-enamide
3-({1-[(5-ethylpyridin-2-yl)methyl]pyrrolidin-3-yl}methyl)benzoic acid
3-{1-[3-(methylsulfanyl)propyl]piperidin-4-yl}-N-phenylpropanamide
(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)({[3-(prop-2-en-1-yl)-4-(prop-2-en-1-yloxy)phenyl]methyl})amine
3-phenyl-1-(1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carbonyl)piperidine
4-{1-[1-(4-ethyl-5-methylthiophene-3-carbonyl)piperidin-4-yl]ethyl}morpholine
N-{[1-(morpholin-4-yl)cycloheptyl]methyl}imidazo[1,2-a]pyrimidine-2-carboxamide
8-[(2E)-3-[4-(dimethylamino)phenyl]prop-2-en-1-yl]-3-ethyl-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}quinoxaline
4-(furan-3-yl)-6-methyl-2-oxo-N-[2-(4,5,6,7-tetrahydro-1H-indazol-3-yl)ethyl]-1,2,3,4-tetrahydropyrimidine-5-carboxamide
9-methoxy-3-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-N-(3-methylbutyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-(4-{4-[cyclohexyl(methyl)amino]piperidin-1-yl}phenyl)-N-[2-(2-methoxyphenyl)ethyl]acetamide
(3R,5R)-N-butyl-1-(pyridin-4-ylmethyl)-5-(pyrrolidin-1-ylmethyl)piperidine-3-carboxamide
4-benzyl-9-(cyclopropylmethyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-N-(trimethyl-1H-pyrazol-4-yl)piperidine-1-carboxamide
6-(4-ethylpiperazin-1-yl)-N-[3-(4-methoxyphenyl)propyl]pyridine-3-carboxamide
1-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine
N-{[3-(2-chlorophenyl)-1,2-oxazol-5-yl]methyl}-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
2-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-N-methylpyridine-4-carboxamide
{1-[({[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}(methyl)amino)methyl]cyclopropyl}methanol
4-{[1-(3-{3-methyl-3H-imidazo[4,5-b]pyridin-2-yl}propanoyl)pyrrolidin-3-yl]methyl}benzoic acid
8-(4-methylpent-3-en-1-yl)-2-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
5-fluoro-2-[1-(3-methoxy-5-methylthiophene-2-carbonyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-4-chloro-1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
N-(furan-2-ylmethyl)-N,1-dimethyl-5-({[1-(morpholin-4-yl)cyclohexyl]methyl}amino)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-[(4,5-dihydro-1H-imidazol-2-yl)amino]-N-[(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]propanamide
1-[(3-methyl-1-benzofuran-2-yl)methyl]-5-oxopyrrolidine-3-carboxylic acid
4,4-difluoro-N-{4-[(2-methoxyethyl)carbamoyl]phenyl}piperidine-1-carboxamide
ethyl 4-[(4-methoxyphenyl)methyl]-1-(4-methylbenzenesulfonyl)piperidine-4-carboxylate
2-methyl-4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]phenol
N-[(3R,4S)-1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-propylpyrrolidin-3-yl]pyrrolidine-1-sulfonamide
N-(3,4-dimethoxyphenyl)-3-(3-methylthiophene-2-carbonyl)piperidine-1-carboxamide
5-(4,4-difluoropiperidine-1-carbonyl)-1H-imidazole-4-carboxylic acid
3-({4-[5-(3-methoxyphenyl)-2-(pyridin-4-yl)pyrimidin-4-yl]piperidin-1-yl}methyl)-1-methyl-1H-indole
2-{[(4-methylpyridin-2-yl)methyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
5-methanesulfonyl-4-(piperidin-3-yl)-N-[3-(pyridin-2-yl)propyl]pyrimidin-2-amine
3-[5-(dimethylamino)-1-methyl-1H-1,2,4-triazol-3-yl]-5-[2-(piperidin-2-yl)ethyl]phenol
2-[(4aR,7aS)-4-[(5-chlorothiophen-2-yl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
1-{1-[(1-methyl-1H-indol-2-yl)methyl]piperidin-4-yl}piperidin-3-ol
4-(3,5-dimethoxyphenyl)-6-methyl-5-(3-oxopiperazine-1-carbonyl)-1,2,3,4-tetrahydropyrimidin-2-one
N-[(2R)-1-{3-hexyl-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl}-1-oxobutan-2-yl]acetamide