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2-[2-(4-fluorophenyl)morpholine-4-carbonyl]-3,5,7-trimethyl-1H-indole
2-ethyl-8-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
1-{1-[2-(4-methoxyphenoxymethyl)-1,3-oxazole-4-carbonyl]azetidin-3-yl}-2-methylpiperidine
2-{[4-(1,3-benzoxazol-2-yl)piperidin-1-yl]methyl}-6-methyl-4-(thiomorpholin-4-yl)quinazoline
4-[(diethylamino)methyl]-5-ethyl-N-[2-(1H-imidazol-4-yl)ethyl]furan-2-carboxamide
7-[(2,3-dimethoxyphenyl)methyl]-2-(1-methylpiperidin-4-yl)-2,7-diazaspiro[4.5]decan-6-one
1-{5-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl}pyrrolidin-3-amine
5-(2-cyclopentylacetamido)-1-methyl-2-(oxolan-2-yl)-N-(1-phenylcyclopropyl)-1H-1,3-benzodiazole-7-carboxamide
2-methyl-6-[1-(5-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)piperidin-4-yl]pyrimidin-4-ol
3-butyl-4-[2-(4-ethoxyphenyl)acetyl]-1-methylpiperazin-2-one
(3R,4S)-4-cyclopropyl-1-[2-(2-methoxy-4-methylphenoxy)ethyl]pyrrolidin-3-amine
4-{[3-(2-chlorophenoxy)azetidin-1-yl]methyl}-1H-imidazole
[(1-ethyl-1H-pyrazol-4-yl)methyl](2-methoxyethyl){[2-(3-methylphenyl)pyrimidin-5-yl]methyl}amine
5-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-4-{[(4-phenyloxan-4-yl)methyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
2-[4-(3-cyanopyrazin-2-yl)piperazin-1-yl]-N-(3-fluoro-2-methylphenyl)acetamide
6-methyl-5-(2,3,4-trimethoxyphenyl)pyridin-2-amine
3-{1-[(2-chlorophenyl)methyl]piperidin-3-yl}-1-(4-methylpiperazin-1-yl)propan-1-one
3-[5-(5-chlorothiophene-2-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
3-[5-({7-hydroxy-2-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl}methyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
5-(1H-indol-6-yl)isoquinoline
N-cyclopentyl-2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-[(2-chlorophenyl)methyl]-2-(dimethylamino)-N-methyl-2,3-dihydro-1H-indene-2-carboxamide
N-({5-[2-methyl-2-(morpholin-4-yl)propyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
1-benzyl-5-[(2,6-difluorophenyl)methyl]-N-methyl-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-{1-[(2E)-2-methylbut-2-enoyl]piperidin-4-yl}-5-(pyridin-3-yl)-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
1-(oxolane-2-carbonyl)-4-[1-(propan-2-yl)piperidine-4-carbonyl]piperazine
N-(4-{[methyl(oxolan-2-ylmethyl)carbamoyl]methyl}phenyl)cyclopropanecarboxamide
2-ethyl-8-({2-methyl-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidin-5-yl}methyl)-2,8-diazaspiro[5.5]undecan-3-one
4-{1-[(2,3-dichlorophenyl)methyl]piperidin-4-yl}-5-methylpyrimidine
methyl 2-[(butan-2-yl)sulfamoyl]-6-[(1-phenyl-1H-pyrazol-4-yl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-propyl-N-(pyridin-3-ylmethyl)-1,3-thiazole-4-carboxamide
4-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-1,3λ6,4-oxathiazinane-3,3-dione
2,6-difluoro-N-{[4-(2-methylphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}benzene-1-sulfonamide
methyl 2-[(5-{3-[(4-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)amino]acetate
1-(2-methoxyphenyl)-4-[1-oxo-1-(pyrrolidin-1-yl)propan-2-yl]piperazin-2-one
4-(4-fluorophenyl)-1-{5-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperidin-4-ol
ethyl 4-{1-[2-(2-chlorophenyl)ethyl]-2-(methoxymethyl)-6-methyl-4-oxo-1,4-dihydropyridine-3-carbonyl}piperazine-1-carboxylate
methyl 1-[(3S,5S)-5-{[(4-methoxyphenyl)methyl]carbamoyl}-1-[(2-methylphenyl)methyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
methyl 3-{[9-methoxy-7-(quinolin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]sulfonyl}thiophene-2-carboxylate
2-[4-({7-[cyclohexyl(hydroxy)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}methyl)phenoxy]ethan-1-ol
N-(3-phenyl-1,2,4-thiadiazol-5-yl)-2-(1,3-thiazol-2-yl)pyrrolidine-1-carboxamide
1-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}-3-(pyridin-4-yl)propan-1-one
(3aR,6aR)-2-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]-5-(propan-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-{[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
5-(2-methylphenyl)-4-{1-[(3-methylthiophen-2-yl)methyl]piperidin-3-yl}-2-(pyridin-4-yl)pyrimidine
2,6-dimethyl-5-{[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-3,4-dihydropyrimidin-4-one
1-{2-[4-(5-fluoro-2-methylbenzenesulfonyl)piperazin-1-yl]ethyl}-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
4-{[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}-1-propylpyrrolidin-2-one
1-(furan-3-carbonyl)-4-(3-methylphenoxy)piperidine-4-carboxylic acid
4-{3-[1-(dimethylamino)ethyl]phenyl}thiophene-2-carboxamide