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(1R,5R)-3-(3-fluoro-4-methoxybenzenesulfonyl)-6-methyl-3,6-diazabicyclo[3.2.2]nonane
5-ethyl-2-methyl-4-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}pyrimidine
3-chloro-5-({3-[(2S,6S)-4-methyl-2,6-bis(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)pyridine
1-[2-(3-ethylpiperazin-1-yl)-2-oxoethyl]-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[(2-ethoxypyridin-3-yl)methyl]quinoxaline-6-carboxamide
N-[3,3-dimethyl-1-(pyridin-3-yl)butyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
1-[3-(3-fluorophenoxymethyl)piperidin-1-yl]-3-(methylsulfanyl)propan-1-one
1-({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)-1-methyl-3-propylurea
N-[2-(1-ethyl-1H-1,3-benzodiazol-2-yl)ethyl]-4,6-dimethyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
N-cyclopropyl-2-(4-fluorophenyl)-N-({3-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)acetamide
3-(1,3-diethyl-6-methyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)-1-[4-(1H-pyrazol-1-yl)butan-2-yl]urea
N-{[6,7-dimethoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-(2-methoxyethyl)furan-2-carboxamide
7-[2-(benzenesulfonyl)ethyl]-2-oxa-7-azaspiro[4.5]decane
2-(4-{1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-1-(furan-3-ylmethyl)piperazin-2-yl)ethan-1-ol
N-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]-3-(1H-pyrazol-1-yl)benzamide
3-{2-[4-(3,5-dimethylphenyl)-3-oxopiperazin-1-yl]-2-oxoethyl}-3-(2-fluorophenyl)-1-(2-methoxyethyl)pyrrolidine-2,5-dione
methyl (2S,4S)-4-cyclohexaneamido-1-[(4-ethylphenyl)methyl]pyrrolidine-2-carboxylate
3-[(1-{[4-(1H-imidazol-1-yl)phenyl]methyl}pyrrolidin-3-yl)methyl]benzamide
N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-3-(2-{[4-(methylsulfanyl)phenyl]methyl}-5-oxopyrrolidin-2-yl)propanamide
8-fluoro-N-[(1-hydroxycyclohexyl)methyl]-4-oxo-1,4-dihydroquinoline-2-carboxamide
1-[(3-fluorophenyl)methyl]-5-[4-(3-methoxypropyl)piperidine-1-carbonyl]piperidin-2-one
N-[(5-ethylpyridin-2-yl)methyl]-1-[2-(4-methoxyphenyl)ethyl]-N-methyl-6-oxopiperidine-3-carboxamide
6-[(3S,4R)-3-hydroxy-4-(hydroxymethyl)piperidine-1-carbonyl]-3,5-dimethyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
1-(2-{4-[1-(2,2-dimethylpropyl)pyrrolidin-3-yl]piperidin-1-yl}-2-oxoethyl)piperidin-2-one
(2S)-N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-1-methylpyrrolidine-2-carboxamide
1-[4-(piperidin-1-ylmethyl)benzoyl]-4-(pyridin-2-ylmethyl)piperazine
5-(4-acetyl-2-methoxyphenoxymethyl)-N-(2-methylprop-2-en-1-yl)-1,2-oxazole-3-carboxamide
4-(2-chloro-4-fluorobenzoyl)-1-[(4-methoxyphenyl)methyl]-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
3-phenyl-N-[4-(4-{[2-(pyridin-3-yl)ethyl]amino}piperidin-1-yl)phenyl]propanamide
N-(butan-2-yl)-6-methyl-4-oxo-N-(thiophen-3-ylmethyl)-1,4-dihydroquinoline-3-carboxamide
1-[3-({6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-5-methylthieno[2,3-d]pyrimidin-4-yl}amino)propyl]pyrrolidin-2-one
3-[2-(4-cyclopentyl-1,4-diazepan-1-yl)-2-oxoethyl]-4-(naphthalen-2-ylmethyl)piperazin-2-one
2-(1-ethyl-1H-pyrazole-4-carbonyl)-N-(pyridin-3-yl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
4-(5-acetylthiophene-2-carbonyl)-1-(4-methylphenyl)piperazin-2-one
3-(4-methylthiophen-2-yl)-5-(morpholine-4-sulfonyl)-N-[2-(piperidin-1-yl)ethyl]benzamide
(4aS,7aR)-4-(2-methoxyethyl)-N-[(2-methylphenyl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
2-(2-{[methyl({[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}phenoxy)propanoic acid
3-(6-methoxynaphthalene-2-carbonyl)-1-(1,3-thiazole-4-carbonyl)piperidine
3-(1H-1,3-benzodiazol-2-yl)-1,2,4,5,10,11-hexaazatricyclo[7.3.0.02,6]dodeca-3,5,7,9,11-pentaene
3-(oxolan-3-yl)-5-(3-phenoxypropyl)-1,2,4-oxadiazole
6-amino-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]pyridine-3-carboxamide
2-{4-[1-(2-fluorophenyl)-2,2-dimethylcyclopropanecarbonyl]piperazin-1-yl}pyridine-3-carbonitrile
N-[2-(2-ethylphenoxy)ethyl]-N-methyl-2-(pyridin-4-yl)pyrimidine-5-carboxamide
7-(1-benzothiophen-3-yl)-9-ethoxy-4-(pyridin-4-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-1-(2-phenylethyl)-1H-1,2,3-triazole-4-carboxamide
(3aS,6aR)-5-(4-methyl-1,3-thiazole-5-carbonyl)-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-(4-{4-[(oxan-4-yl)amino]piperidin-1-yl}phenyl)-3-phenylpropanamide
3-[ethyl({[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl})amino]-1λ6-thiolane-1,1-dione
4-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
1-(2-{1-[(2-cyclohexylpyrimidin-5-yl)methyl]piperidin-2-yl}ethyl)pyrrolidin-2-one