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N-ethyl-3-(2-methylpropanamido)-N-{[2-(prop-2-en-1-yloxy)phenyl]methyl}benzamide
5-(2-phenylphenyl)pyrimidin-2-amine
5-fluoro-2-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-ylmethyl}-3-methyl-1H-indole
1-benzyl-N5-ethyl-N3-methyl-4-oxo-N3-(2-phenylethyl)-1,4-dihydropyridine-3,5-dicarboxamide
(5S)-5-({[(1-ethyl-1H-indol-6-yl)methyl](pyridin-2-ylmethyl)amino}methyl)pyrrolidin-2-one
6-[5-(1-ethoxyethyl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-1-yl]-2-methyl-1,3-benzothiazole
2-[4-(cyclopropylamino)-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]-6-methylpyridine-3-carbonitrile
N-[2-(1-methylpiperidin-2-yl)ethyl]-6-(3-oxopiperazin-1-yl)pyridine-3-carboxamide
N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
1-(3-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}-3-oxopropyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-[(1S,2R)-2-[(1-methylpiperidin-4-yl)amino]cyclobutyl]-2,3-dihydro-1,4-benzodioxine-6-sulfonamide
2-(2,5-dimethylphenoxy)-N,N-bis(pyridin-3-ylmethyl)propanamide
1-(4-{[2-(hydroxymethyl)phenyl]methyl}piperazin-1-yl)-2-(oxan-2-ylmethoxy)ethan-1-one
(2S)-2-hydroxy-1-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-phenylethan-1-one
N-{[7-(6-methoxypyridazin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(3-methyl-1H-pyrazol-1-yl)acetamide
1-benzyl-5-acetamido-2-methyl-N-[(1-methyl-2,3-dihydro-1H-indol-5-yl)methyl]-1H-1,3-benzodiazole-7-carboxamide
2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-methyl-N-[3-(oxolan-2-yl)propyl]acetamide
N-benzyl-N-methyl-2-(4-methylpiperazin-1-yl)-6-(thiophen-2-yl)pyridine-3-carboxamide
1-benzyl-8-(oxan-4-yl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
8-{[5-(3-chlorophenyl)furan-2-yl]methyl}-1-(2-methoxyethyl)-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}-3,3-dimethylpiperazin-2-one
6-[3-(hydroxymethyl)-3-propylpiperidine-1-carbonyl]-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-[3-({ethyl[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]acetamide
1-[6-(3-chlorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-N,N-dimethylpyrrolidin-3-amine
3-amino-1-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}pyrrolidine-3-carboxylic acid
N-methyl-3-(2-methyl-1H-indol-1-yl)-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}propanamide
(1R,5R)-6-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-{1-[1-(2-cyclohexylethyl)-1H-1,2,3-triazole-4-carbonyl]pyrrolidin-2-yl}-6-methyl-1H-1,3-benzodiazole
1-benzoyl-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]piperidin-4-amine
1-(2,7-dimethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-5-phenylpentan-1-one
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-2-(methylamino)pyridine-3-carboxamide
5-methyl-3-[2-(1H-pyrazol-4-yl)ethyl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
2-(dimethylamino)-2-(3-methylphenyl)-1-[4-(1H-1,2,4-triazole-3-carbonyl)piperazin-1-yl]ethan-1-one
4-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]-1-[(3-fluorophenyl)methyl]piperazin-2-one
2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)-1-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}ethan-1-one
1-methyl-4-{2-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidine
8-[2-(3-fluoro-4-phenylphenyl)propanoyl]-2,8-diazaspiro[4.5]decan-3-one
2-ethyl-8-(7-fluoro-2-oxo-1,2-dihydroquinoline-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
1-{2-[(4-methoxyphenyl)sulfanyl]ethyl}-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
4-[2-(3-methoxyphenyl)acetyl]-5-methyl-1-(2-methylphenyl)piperazin-2-one
1-[3-(2-methoxyphenoxy)azetidin-1-yl]-2-[3-(methylsulfanyl)phenyl]ethan-1-one
N-(2,1,3-benzoxadiazol-5-ylmethyl)-6-(dimethylamino)-N-methylpyridine-3-carboxamide
2-[4-({[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amino)piperidin-1-yl]pyridine-3-carbonitrile
1-cyclohexyl-3-{[1-(1,3-dihydroxypropan-2-yl)pyrrolidin-3-yl]methyl}urea
7-chloro-3-{[(2,2-dimethyloxan-4-yl)amino]methyl}-1-(2-phenylethyl)-1,2-dihydroquinolin-2-one
4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]-1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperidine
2-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-4-[3-(3-methylpiperidine-1-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
1-[1-(1H-imidazol-4-ylmethyl)piperidin-4-yl]-3-methylbutan-1-ol
{[2-(3-methoxyphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}(methyl)(1,2-oxazol-5-ylmethyl)amine
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]acetamide