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4-methyl-2-(propan-2-yl)-N-{1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl}-1,3-thiazole-5-carboxamide
1-{7-[(2,3-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-3-methoxypropan-1-one
(2S,4S)-N-ethyl-1-(oxan-4-yl)-4-[2-(pyridin-3-yl)acetamido]pyrrolidine-2-carboxamide
(2S,4R)-4-amino-1-[2-(7-fluoro-2-methyl-1H-indol-3-yl)acetyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-methyl-N-(2-phenoxyethyl)-2-(1H-pyrazol-4-yl)quinoline-4-carboxamide
N-(3,5-dimethoxyphenyl)-2-[(2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-yl)amino]acetamide
3-benzyl-N-(9H-fluoren-9-yl)-4,5-dihydro-1,2-oxazole-5-carboxamide
1-[4-hydroxy-3-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-5-oxopyrrolidine-3-carboxylic acid
3-ethyl-1-{[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl}piperidine-3-carboxylic acid
N-{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}-2-(4-methyl-1,2,5-oxadiazol-3-yl)acetamide
(2S)-2-{[6-(2-fluorophenyl)imidazo[2,1-b][1,3]thiazol-3-yl]formamido}-4-methylpentanamide
5-fluoro-N,N-dimethyl-2-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]pyrimidin-4-amine
2-(4-fluoro-1H-indol-1-yl)-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidine
3-hydroxy-1-(2-methoxyethyl)-3-{[methyl(quinolin-5-ylmethyl)amino]methyl}piperidin-2-one
5-cyclopropyl-N-(2,3-dihydro-1H-inden-2-yl)-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
methyl 2-{[(4-chlorophenyl)methyl]sulfamoyl}-6-[1-(methylsulfanyl)propan-2-yl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-(2-carboxyphenyl)-5-[(propan-2-yl)sulfamoyl]benzoic acid
6-[3-(3-methoxypropyl)piperidine-1-carbonyl]-1-methyl-1H-indole
ethyl 4-{[(furan-2-ylmethyl)[2-(morpholin-4-yl)ethyl]amino]methyl}-1H-pyrazole-3-carboxylate
2-[(4aS,7aR)-6,6-dioxo-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-2-oxoacetamide
2-({3-[(4-fluorophenyl)amino]piperidin-1-yl}methyl)-4-methoxyphenol
methyl 1-{2-[(1-methanesulfonylpiperidin-4-yl)oxy]benzoyl}piperidine-2-carboxylate
(3S,4S)-4-methyl-1-{[4-(methylsulfanyl)phenyl]methyl}piperidine-3,4-diol
3-[4-(2,3-dimethylphenyl)piperazine-1-carbonyl]-2-methyl-2,8-diazaspiro[4.5]decane
1-(1H-imidazol-2-ylmethyl)-4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidine
4-[(2R)-2-amino-3-phenylpropanoyl]-1-[(3-methoxyphenyl)methyl]piperazin-2-one
8-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-1-oxa-8-azaspiro[4.5]decane
N-tert-butyl-1-cyclohexyl-5-[4-(6-methylpyridin-2-yl)piperazine-1-carbonyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
N-{[(3S,4S)-1-[(4-ethynylphenyl)methyl]-3-hydroxypiperidin-4-yl]methyl}morpholine-4-carboxamide
1-[(4,5-dimethylfuran-2-yl)methyl]-N-[3-(1H-pyrazol-1-yl)phenyl]piperidine-3-carboxamide
4-ethyl-3-{[1-(5-hydroxypyrazine-2-carbonyl)piperidin-4-yl]methyl}-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(4-fluorophenyl)-1-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]piperidine
N-[(2R,3R)-1'-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]thiophene-2-carboxamide
2-methyl-8-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]-1,3,8-triazaspiro[4.5]dec-1-en-4-one
N-cyclohexyl-3-[4-(1-methyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]propanamide
ethyl 1-(2,2-dimethyloxane-4-carbonyl)-4-(3-phenylpropyl)piperidine-4-carboxylate
1-(1-benzothiophen-2-ylmethyl)-4-(2-methanesulfonylethyl)piperazine
3-(5-{[3-methyl-4-(propan-2-yl)piperazin-1-yl]methyl}thiophen-3-yl)prop-2-yn-1-ol
(1S,6R)-3-(2-{4-[(4-fluorophenyl)methyl]piperidin-1-yl}-2-oxoethyl)-3,9-diazabicyclo[4.2.1]nonan-4-one
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
1-[2-({[2-(1H-1,3-benzodiazol-2-yl)ethyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
4-(3-cyclopentyl-1-ethyl-1H-1,2,4-triazol-5-yl)pyridine
(3R,4S)-4-cyclopropyl-1-(3,5-dichloropyridin-2-yl)pyrrolidin-3-amine
N-[(1S,2S)-2-(benzyloxy)cyclohexyl]-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
6-{[(1R,5S,8S)-8-methoxy-3-azabicyclo[3.2.1]octan-3-yl]methyl}pyrazolo[1,5-a]pyrimidine-3-carboxylic acid
N-[3-(1H-imidazol-1-yl)propyl]-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
8-(furan-3-ylmethyl)-2-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
8-[4-(hydroxymethyl)benzoyl]-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
methyl 2-(1-{1-[(3-methoxyphenyl)methyl]-6-oxopiperidin-3-yl}-N-methylformamido)acetate