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2-(5-methylthiophen-2-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-methyl-8-{[5-(1H-pyrazol-5-yl)furan-2-yl]sulfonyl}-2,8-diazaspiro[4.5]decan-3-one
2-ethyl-4-{1-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-1H-imidazol-2-yl}pyrimidine
1-(2-chlorophenyl)-3-{1-[1-(2-hydroxypropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
2-amino-6-(2-fluorophenyl)-4-[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
(4aR,7aS)-1-methanesulfonyl-4-(4-methyl-1H-pyrrole-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
methyl (2R)-2-{[1-(4,7-dimethylquinazolin-2-yl)piperidin-4-yl]formamido}propanoate
2-methyl-3-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrazine
5-({4-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}methyl)quinoxaline
5-ethoxy-2-methyl-N-[(1-methylpyrrolidin-3-yl)methyl]-1-benzofuran-3-carboxamide
1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-3-(piperidin-1-ylmethyl)piperidine
3-cyclopentyl-N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)propanamide
3-(2-ethyl-1H-1,3-benzodiazol-6-yl)-1-methyl-1-[(1-phenylpyrrolidin-3-yl)methyl]urea
7-(1,3-benzothiazol-2-yl)-4-(pyrrolidine-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
ethyl 1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
(1R,5R)-6-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
1-[2-(dimethylamino)ethyl]-5-{2-[(5-methyl-1,3,4-oxadiazol-2-yl)amino]ethyl}pyrrolidin-2-one
5-methyl-5-phenyl-1-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}piperidin-2-one
(2S,4S)-4-{[(4-chlorophenyl)methyl]amino}-N-ethyl-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
N-{[2-(dimethylamino)-7-methoxyquinolin-3-yl]methyl}-N-(2-methoxyethyl)-3-phenyl-1H-pyrazole-5-carboxamide
(2E)-3-(2-chlorophenyl)-N-cyclopropyl-N-({3-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)prop-2-enamide
4-cyclobutaneamido-N-methyl-N-[3-(1H-pyrazol-1-yl)propyl]benzamide
3-(4-chloro-2-methylbenzoyl)-1-(1,4-dithiepan-6-yl)piperidine
6-[3-(4-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-2-methyl-2,3,4,5-tetrahydropyridazin-3-one
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-[1-(thiophen-2-ylmethyl)piperidin-3-yl]acetamide
2-butyl-8-(1-ethyl-1H-pyrazole-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
4-{1H-[1,2,3]triazolo[4,5-b]pyridin-6-yl}-1H-indole
1-{4-[2-(3-methoxyphenyl)-1-[methyl(pyridin-2-ylmethyl)amino]ethyl]piperidin-1-yl}-2-(methylsulfanyl)ethan-1-one
(3S,4S)-4-(dimethylamino)-1-[(2-fluoro-4,5-dimethoxyphenyl)methyl]pyrrolidin-3-ol
1-(3,5-dimethylfuran-2-carbonyl)-4-{4-[(3,3-dimethylpyrrolidin-1-yl)methyl]-1H-1,2,3-triazol-1-yl}piperidine
N-(1-phenylcyclopropyl)-5-[(quinolin-8-yloxy)methyl]-1,2-oxazole-3-carboxamide
6-methyl-2-(1-{6-methylpyrazolo[1,5-a]pyrimidine-3-carbonyl}pyrrolidin-2-yl)-1H-1,3-benzodiazole
1-{3-[2-(3-ethenylphenyl)-1H-imidazol-1-yl]propyl}piperidine-4-carboxamide
4-(1H-imidazol-1-yl)-1-[(5-methylthiophen-2-yl)sulfonyl]piperidine-4-carboxylic acid
N-ethyl-N'-(3-ethylphenyl)-N-(pyridin-4-ylmethyl)butanediamide
2-(thiomorpholin-4-yl)-2-[3-(trifluoromethoxy)phenyl]acetic acid
N-butyl-N-[(4-fluorophenyl)methyl]-2-(2-hydroxyphenyl)acetamide
2-(1,4-dimethylpiperazin-2-yl)-1-(3,3-diphenylpiperidin-1-yl)ethan-1-one
1-{1-[(3-cyanophenyl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
2-[4-(2,2-dimethylpropyl)-1-[(3-methoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
2-(2-methoxyethyl)-8-(7-methyl-1-benzofuran-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
1-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-[(1-methyl-1H-indol-3-yl)sulfanyl]ethan-1-one
3-(cyclopropylmethyl)-5-{[3-(2-fluorophenyl)pyrrolidin-1-yl]methyl}-1,2,4-oxadiazole
2-[2-(dimethylamino)ethyl]-9-(2-phenoxyacetyl)-2,9-diazaspiro[5.5]undecan-3-one
2-[(4-methoxyphenyl)methyl]-N-(prop-2-en-1-yl)-1,3-benzoxazole-6-carboxamide
1-(3,5-dimethylphenyl)-4-[2-(2-methoxyethoxy)acetyl]piperazin-2-one
methyl 4-{1-[(3-fluorophenyl)carbamoyl]-6-azaspiro[2.5]octan-6-yl}-4-oxobutanoate
N-(1-benzylpiperidin-4-yl)-1-[(4-methoxyphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
1-{4-[4-({[1-(morpholin-4-yl)cycloheptyl]methyl}amino)piperidin-1-yl]benzoyl}piperidin-3-ol
ethyl 4-{6-[(6-methyl-4-oxo-4H-chromen-3-yl)methyl]-6-azaspiro[2.5]octane-1-amido}piperidine-1-carboxylate