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(1-{1-[(2-cyclohexylpyrimidin-5-yl)methyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methanol
7-(cyclopropylmethyl)-2-(1-methylpiperidin-4-yl)-2,7-diazaspiro[4.5]decane
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
(1S,5R)-3-[(6-methylpyridin-2-yl)methyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-6-[(3-hydroxypropyl)(methyl)amino]pyridine-3-carboxamide
2-(2,3-dihydro-1H-inden-1-yl)-N-methyl-N-(quinolin-2-ylmethyl)acetamide
5-{1-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]pyrrolidin-2-yl}thiophene-2-carboxamide
5-methyl-4-(1-methyl-1H-pyrazol-4-yl)-N-[(1-methylpyrrolidin-3-yl)methyl]pyrimidin-2-amine
1,4-dimethyl-9-{2-[(2-methylprop-2-en-1-yl)oxy]benzoyl}-1,4,9-triazaspiro[5.5]undecane
2-{2-methyl-6-[4-(pyrrolidin-1-yl)piperidin-1-yl]pyrimidin-4-yl}ethan-1-amine
2-butyl-N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-1,3-benzoxazole-5-carboxamide
6-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
3-{[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}piperidine
N-(1-carbamoylcyclopentyl)-4-methylpyrimidine-5-carboxamide
1-ethyl-4-[5-(2-fluoro-6-methoxyphenyl)-4-phenyl-1H-imidazol-1-yl]pyrrolidin-2-one
7-[4-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)benzoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-(4-chloro-2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}phenoxy)acetamide
[(3,5-dichloropyridin-4-yl)methyl](methyl)(1,2-oxazol-3-ylmethyl)amine
1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-4-(pyrrolidin-3-yl)piperazine
N-{[4-(2,3-dihydro-1H-inden-2-yloxy)phenyl]methyl}-N-[(3S)-2-oxoazepan-3-yl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
1-(3-methoxy-4-methylphenyl)-3-[2-(1-methylpyrrolidin-2-yl)ethyl]urea
3-(1-ethyl-1H-imidazol-2-yl)-1-[2-(4-methylphenoxy)ethanesulfonyl]piperidine
4-(1H-1,2,3,4-tetrazol-5-yl)-2-(4H-1,2,4-triazol-4-yl)phenol
N-[(3,4-difluorophenyl)methyl]-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
1-[(2,3-difluorophenyl)methyl]-4-(pyrrolidin-3-yl)piperidine
ethyl 4-{1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carbonyl}piperazine-1-carboxylate
6-(3-cyclopentylpropanoyl)-N-[(6-methylpyridin-2-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
1-[1'-(2,3-dihydro-1H-inden-2-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
1-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]-4-(4H-1,2,4-triazol-4-yl)piperidine
3-(1-methanesulfonylpiperidin-3-yl)-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
(3S,9aR)-3-[(1R)-1-(benzyloxy)ethyl]-8-{[1-(2-chlorophenyl)-1H-pyrazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
5-ethyl-2-(4-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-1-yl)pyrimidine
3-(2H-1,3-benzodioxol-5-yl)-5-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
(4aS,8aR)-6-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-1-propyl-decahydro-1,6-naphthyridin-2-one
(2R,3R,6R)-3-(4-fluorophenyl)-5-{imidazo[1,2-a]pyridine-3-carbonyl}-1,5-diazatricyclo[5.2.2.02,6]undecane
3-phenyl-1-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]piperazine
{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]methylamine
7-(2-hydroxyethyl)-2-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
1-[benzyl(methyl)amino]-3-(2-methoxy-5-{[(2-methoxyethyl)(methyl)amino]methyl}phenoxy)propan-2-ol
4-({[3-(1H-imidazol-1-yl)propyl](pyridin-3-ylmethyl)amino}methyl)benzoic acid
N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
9-methoxy-4-[(2-methoxyphenyl)methyl]-7-(6-methoxypyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
7-{[5-(3-chlorophenyl)furan-2-yl]methyl}-3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
2-({[6-(azocane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}(thiophen-2-ylmethyl)amino)ethan-1-ol
N-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-4-(pyridin-3-yl)pyrimidin-2-amine
ethyl 4-[({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)(2-methylpropyl)amino]piperidine-1-carboxylate
2,5-dimethyl-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
(3E)-1-[2-(ethoxymethyl)-4-(pyrrolidin-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]pent-3-en-1-one
3-(oxolan-3-yl)-5-[3-(pyrrolidin-1-yl)propyl]-1,2,4-oxadiazole
(3S,4R)-4-(3-methoxyphenyl)-1-[3-(2-methyl-1H-imidazol-1-yl)propanoyl]pyrrolidine-3-carboxylic acid