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1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazine
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
1-[(5-chlorofuran-2-yl)methyl]-4-{imidazo[1,2-b]pyridazin-6-yl}piperazine
[3-benzyl-1-(2,4-dimethylbenzoyl)piperidin-3-yl]methanol
N-[(1-cyclopentylpiperidin-3-yl)methyl]-N-[2-(piperidin-1-yl)ethyl]propanamide
(2R,3S,6R)-3-(3,5-difluorophenyl)-5-propyl-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(1'-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl)propan-1-one
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-[2-(4-methoxyphenyl)phenyl]pyrrolidine-2-carboxamide
4-{1-[3-(2-methylpropyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1,2-dihydrophthalazin-1-one
6-{[methyl(2-methylpropyl)amino]methyl}-2-oxo-N-(quinolin-3-ylmethyl)-1,2-dihydropyridine-3-carboxamide
{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}(methyl)(pyridin-3-ylmethyl)amine
5-(2-{4-[(6-chloropyridin-3-yl)methyl]piperazin-1-yl}-2-oxoethyl)-1,3-dimethylimidazolidine-2,4-dione
1-methyl-4-{4-[1-methyl-3-(2-methyl-1,3-thiazol-4-yl)-1H-1,2,4-triazol-5-yl]phenyl}piperazine
N-(4-fluorophenyl)-1-(4-phenyl-1H-imidazole-5-carbonyl)piperidin-3-amine
1-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine
1-(2-methoxyphenyl)-4-(2-propoxybenzoyl)piperazin-2-one
2-(4-{[1-(3-chlorophenyl)-1H-pyrazol-4-yl]methyl}-1-(2,2-dimethylpropyl)piperazin-2-yl)ethan-1-ol
(3S,4R)-4-(3-fluorophenyl)-1-{2-[(2-methoxyethyl)(methyl)amino]acetyl}pyrrolidine-3-carboxylic acid
3-[5-(2-phenylethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]benzonitrile
N-[(4-fluorophenyl)methyl]-4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}benzamide
N,N-dimethyl-2-[(4,4,4-trifluorobutanamido)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
N-(2-hydroxyethyl)-2-(pyridin-4-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]pyrimidine-5-carboxamide
9-oxo-N-(propan-2-yl)-8-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecane-2-carboxamide
2-({[2-(3-chlorophenyl)ethyl]amino}methyl)-4-(pyrazin-2-yl)phenol
N-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-[(3-fluorophenyl)methyl]-N-[(4-methoxyphenyl)methyl]-2-(pyrrolidin-3-yl)acetamide
1-[4-(1H-imidazol-1-yl)phenyl]-3-(5-oxo-1-propylpyrrolidin-3-yl)urea
N-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
4-ethyl-3-({1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(1r,4r)-4-[({5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]cyclohexane-1-carboxamide
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-2-(4-methyl-1,4-diazepan-1-yl)acetamide
methyl[(1-methyl-1H-imidazol-5-yl)methyl](quinolin-6-ylmethyl)amine
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
1-cyclopentyl-N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}piperidine-3-carboxamide
1-{6-[4-(2-methoxyphenoxy)piperidin-1-yl]pyridin-2-yl}ethan-1-ol
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-2-(phenylamino)pyrimidine-5-carboxamide
N,N-bis(1,3-oxazol-4-ylmethyl)-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanamide
(3S,4S)-1-(1H-imidazol-2-ylmethyl)-4-(4-methylpiperazin-1-yl)pyrrolidin-3-ol
N'-cyclopentyl-N-[1-(1-methyl-1H-imidazol-2-yl)butyl]butanediamide
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-cyclopropyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]acetamide
1-{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(2-methylphenoxy)piperidine
6-methyl-5-[5-(2-methyl-1,3-benzothiazol-5-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
4-{[3-(2-methylphenyl)piperidin-1-yl]methyl}-2-(propan-2-yl)pyrimidine
N-[(5-fluoro-2-methylphenyl)methyl]-4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
2-[5-cyclopropyl-4-(4-methylpiperazine-1-carbonyl)-1H-pyrazol-1-yl]-4-(thiophen-2-yl)pyrimidine
dimethyl({[(1R,5S,6S)-3-[1-methyl-5-(thiophen-2-yl)-1H-pyrazole-3-carbonyl]-3-azabicyclo[3.1.0]hexan-6-yl]methyl})amine
2-(2-hydroxyethyl)-8-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
4-methyl-2-({methyl[(3-phenyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenol
N-(1-{1-[(3-fluorophenyl)methyl]piperidin-4-yl}-2-phenylethyl)-N-methylthiophene-2-carboxamide
[(3R,4R)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}-1-[(1-methyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-yl]methanol