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3-[benzyl({[2-(ethylamino)pyrimidin-5-yl]methyl})amino]-2-methylpropan-1-ol
2-(6-hydroxypyrimidin-4-yl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)propanamide
N-benzyl-2-({3-methyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl}sulfanyl)-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}acetamide
1-{4-[6-amino-2-(butylsulfanyl)pyrimidin-4-yl]-1,4-diazepan-1-yl}ethan-1-one
[(5-ethylpyridin-2-yl)methyl](methyl)({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)amine
(2S,3R)-2-[({[(2-fluorophenyl)methyl]carbamoyl}methyl)amino]-3-hydroxybutanamide
2-[(4aS,8aR)-1-(4-hydroxybutyl)-2-oxo-decahydro-1,6-naphthyridin-6-yl]-1,3-thiazole-4-carboxamide
6-ethyl-2-methoxy-3-[({2-methylthieno[2,3-d]pyrimidin-4-yl}amino)methyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
dimethyl[(2-{[5-(morpholine-4-carbonyl)pyridin-2-yl]oxy}phenyl)methyl]amine
N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-2-(2-methyl-1H-indol-3-yl)acetamide
3-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-4,5,6,7-tetrahydro-1,2-benzoxazole
N-[(3R,4S)-4-cyclopropyl-1-[1-(piperidin-4-yl)-1H-1,2,3-triazole-4-carbonyl]pyrrolidin-3-yl]acetamide
3-(3-chloro-1H-1,2,4-triazol-5-yl)-1-(4-hydroxy-1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
1-cyclopropanecarbonyl-N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}piperidine-4-carboxamide
N-methyl-N-[4-(1-methyl-1H-1,2,4-triazol-5-yl)phenyl]methanesulfonamide
4-[4-fluoro-3-(hydroxymethyl)phenyl]benzamide
1-(2-methoxyethyl)-4-[3-(propan-2-yl)-1-(quinolin-8-yl)-1H-1,2,4-triazol-5-yl]pyrrolidin-2-one
N-{1-[1-(2-aminopyrimidin-4-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-phenylpropanamide
1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N-({1-[(3,5-dichlorophenyl)methyl]pyrrolidin-3-yl}methyl)-2-methoxyacetamide
1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-4-(2-methoxyphenyl)piperazine
5-[(7-{[4-(4-fluorophenyl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)methyl]-2-methoxyphenol
N-[(3-ethoxyphenyl)methyl]-N-(2-hydroxyethyl)-2-methyloxolane-2-carboxamide
N-[(5-fluoro-1H-indol-2-yl)methyl]-N-methyl-5-(phenoxymethyl)-1,2-oxazole-3-carboxamide
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-4-(1H-pyrazol-3-yl)benzamide
(3R,4S)-1-[4-methyl-2-(piperidin-1-yl)pyrimidine-5-carbonyl]-4-phenylpyrrolidin-3-amine
4-{[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-[3-(2-methyl-1H-imidazol-1-yl)-1-phenylpropyl]acetamide
3-(3-chloro-1,2-oxazol-5-yl)-1-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
2-(2-oxo-1,3-oxazolidin-3-yl)-N-[(1S,3S)-3-{[4-(pyridin-2-yl)pyrimidin-2-yl]amino}cyclopentyl]acetamide
4-(cyclopropylmethyl)-1-(5-ethylthiophene-3-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
4-[(2-ethoxyphenyl)methyl]-9-methoxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-methanesulfonyl-N-(pentan-3-yl)acetamide
1-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethan-1-one
3-{[(3aR,6aS)-5-methyl-octahydropyrrolo[3,4-c]pyrrol-2-yl]methyl}benzoic acid
N1-(4-ethyl-1,3-dimethyl-1H-pyrazol-5-yl)-4-(piperidin-1-yl)piperidine-1,4-dicarboxamide
methyl 3-[(2-methyl-1H-indol-3-yl)methyl]-9-[(1-methyl-5-oxopyrrolidin-3-yl)methoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-methyl-5-(4-methylpiperidin-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
6-(3-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-3-oxopropyl)-2,3-dihydropyridazin-3-one
4-{[6-(2,4-dimethylphenyl)pyridin-3-yl]methyl}morpholine
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[2-(4-methylphenyl)ethyl]piperidine-3-carboxamide
N-(1-ethyl-2-methyl-1H-indol-5-yl)-2-oxo-1-oxa-3,8-diazaspiro[4.6]undecane-8-carboxamide
2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}propanamide
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-2-(2-methyl-1,3-thiazol-4-yl)acetamide
1-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-5-(2-{[(2-fluorophenyl)methyl]amino}ethyl)pyrrolidin-2-one
4-{2-[(6-methoxypyrimidin-4-yl)oxy]hex-5-en-1-yl}morpholine
1-[(3,4-dimethoxypyridin-2-yl)methyl]-2-methyl-1,4-dihydroquinolin-4-one
2-(2-{6-oxa-9-azaspiro[4.5]decan-9-yl}-2-oxoethyl)-5-(piperidin-1-yl)-2,3-dihydropyridazin-3-one
(4aR,7aS)-1-[2-(4-hydroxypiperidin-1-yl)pyrimidin-4-yl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione