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1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-N-(6-phenoxypyridin-3-yl)piperidine-2-carboxamide
N-[1-(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)-2-phenylethyl]-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
N-(1-{7-benzyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)-2-methoxyacetamide
{[3-(3-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[3-(4-methyl-1,3-thiazol-5-yl)propyl]amine
5-{[4-(2-methoxyphenyl)piperidin-1-yl]methyl}-N-propylpyrimidin-2-amine
1-ethyl-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-1H-pyrazole-4-sulfonamide
methyl 2-hydroxy-5-{[4-(3-methylpyridin-2-yl)piperazin-1-yl]methyl}benzoate
2-({3-methyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl}sulfanyl)-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
N-methyl-1-(4,6,7-trimethylquinazolin-2-yl)piperidine-4-carboxamide
2-methyl-6-{1-[(1-phenyl-1H-pyrazol-5-yl)methyl]piperidin-4-yl}pyrimidin-4-ol
1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-3-(2-methylphenyl)pyrrolidin-3-ol
6-methyl-1-(2-methylphenyl)-4-[4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]piperazin-2-one
9-(2-fluorobenzoyl)-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecane
1-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-3-(1H-pyrazol-1-yl)propan-1-one
3-(3-fluorophenyl)-4-[2-(trimethyl-1H-pyrazol-1-yl)acetyl]piperazin-2-one
4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]-1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidine
N-(3-{2-[3-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}phenyl)acetamide
(3R,4S)-1-(3-chloro-1H-indole-2-carbonyl)-4-cyclopropylpyrrolidin-3-amine
N'-(2-fluoro-5-methylphenyl)-N-[2-(morpholin-4-yl)ethyl]butanediamide
2-[2-(1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)-1H-imidazol-1-yl]acetamide
N-(1,4-dioxan-2-ylmethyl)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
4-[5-(6-chloropyridazin-3-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl]morpholine
N,N-dimethyl-3-[1-(3-methylphenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]propanamide
N-benzyl-N-methyl-1-[1-(propan-2-yl)piperidin-4-yl]piperidin-3-amine
N-cycloheptyl-2-methyl-6-(piperidin-3-yl)pyrimidin-4-amine
1-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}-3-[3-(propan-2-yloxy)benzoyl]piperidine
2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)-1-{1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}ethan-1-one
5-(4-methylnaphthalen-1-yl)-1H-1,2,4-triazole
4-(2-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-oxoethyl)piperazin-2-one
1-[1'-(3-ethoxybenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-cyclobutanecarbonylpiperidine-4-carboxamide
{[3-(methylsulfanyl)phenyl]methyl}(oxolan-2-ylmethyl)(pyridin-4-ylmethyl)amine
N-[(3S)-2-oxoazepan-3-yl]-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
(5-{[3-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]methyl}furan-2-yl)methanol
6-methyl-4-[2-(4-methylpentyl)morpholine-4-carbonyl]-1,2-dihydroquinolin-2-one
2,6-dimethyl-3-[4-(pyridin-3-yl)piperazine-1-carbonyl]quinoline
2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-N-[6-(propan-2-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]acetamide
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-[(4-methyl-1H-imidazol-5-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
5-(5-chloro-2-methoxybenzoyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
2-chloro-N-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}benzamide
1-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine
N-({8-[(2,4,5-trimethoxyphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)furan-2-carboxamide
N-{[4-(aminomethyl)phenyl]methyl}-4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carboxamide
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(1,3-dihydroxypropan-2-yl)acetamide
3-amino-N-[1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]thiophene-2-carboxamide
1-(1-{[1-(cyclohexylmethyl)-2-cyclopropylmethanesulfonyl-1H-imidazol-5-yl]methyl}piperidin-3-yl)ethan-1-one
3-benzyl-8-(furan-3-ylmethyl)-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-1-(2-methylpropyl)-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
7-(oxan-4-yl)-2-(3-phenoxypropyl)-2,7-diazaspiro[4.5]decan-6-one
ethyl 5-[(3-hydroxyphenyl)methyl]-1-[3-(pyridin-3-yl)propyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate