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ethyl 1-{2-[3-(2-chlorophenyl)-1-cyclopentyl-2,5-dioxopyrrolidin-3-yl]acetyl}piperidine-3-carboxylate
1-(3-oxo-1,3-dihydro-2-benzofuran-5-yl)-3-(propan-2-yl)-3-(2,2,2-trifluoroethyl)urea
N,2,8-trimethyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]quinoline-4-carboxamide
dimethyl({5-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]furan-2-yl}methyl)amine
N-(1-{1-[2-(3,4-difluorophenyl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopropanecarboxamide
1-[(2,3-difluorophenyl)methyl]-3-({[(5-fluoro-2-methylphenyl)methyl]amino}methyl)-3-hydroxypiperidin-2-one
1-{3-[5-(oxolan-3-yl)-4-phenyl-1H-imidazol-1-yl]propyl}pyrrolidin-2-one
1-[2-({[2-(adamantan-1-yl)-1,3-thiazol-4-yl]methyl}amino)ethyl]imidazolidin-2-one
N-ethyl-4-{4-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-1H-1,2,3-triazol-1-yl}piperidine-1-carboxamide
5-{[benzyl(methyl)amino]methyl}-N-[(5-chlorothiophen-2-yl)methyl]-1,2-oxazole-3-carboxamide
N'-{2-[methyl(phenyl)amino]propyl}ethanediamide
4-{3-[4-(furan-2-carbonyl)piperazine-1-carbonyl]piperidin-1-yl}-2-(2-methoxyethyl)-2,3-dihydro-1H-isoindole-1,3-dione
2-[2-fluoro-6-(propan-2-yloxy)phenyl]-2-[methyl(1,2-oxazol-3-ylmethyl)amino]acetic acid
{[(1-{[3-(4-chlorophenoxy)phenyl]methyl}piperidin-3-yl)methyl]sulfamoyl}dimethylamine
N4-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-5-ethyl-6-methylpyrimidine-2,4-diamine
4-(2-cyclopropyl-4-methylpyrimidine-5-carbonyl)-2-(trifluoromethyl)morpholine
[(3R,4R)-1-(3-chloro-5-fluorobenzoyl)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)pyrrolidin-3-yl]methanol
1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-3-phenylpyrrolidin-3-ol
N-cyclopropyl-1-{1-[3-(dimethylamino)benzoyl]piperidin-4-yl}piperidine-4-carboxamide
7-methyl-3-[3-(prop-2-en-1-yloxy)benzoyl]-3,7,11-triazaspiro[5.6]dodecan-12-one
{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]methylamine
(5S,9aS,9bS)-5-(3-hydroxy-4-methoxyphenyl)-2-[(2-methylphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
(3aR,6aR)-2-cyclopropanecarbonyl-5-[(2-ethylpyrimidin-5-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-4-[2-(2-phenylethyl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidine
N-[1-(dimethyl-1,3-thiazol-2-yl)propyl]-2-(methylamino)acetamide
3-[1-(pyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-1H-indazole
N-{[1-(morpholin-4-yl)cyclohexyl]methyl}-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
5-{1-[4-(2-methylpropyl)benzoyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-propylimidazolidine-2,4-dione
4-(3-fluorophenoxy)-1-(pyridin-3-ylmethyl)piperidine-4-carboxylic acid
5-(4-hydroxypiperidin-1-yl)-1-methyl-N-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-(but-2-yn-1-yl)-5-{1-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]piperidin-4-yl}-5-(3-phenylpropyl)imidazolidine-2,4-dione
[(3R,4S)-1-{[4-methoxy-2-methyl-5-(propan-2-yl)phenyl]methyl}-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
methyl 2-[1-(2-methoxyethyl)-2,4-dioxo-8-{[3-(trifluoromethyl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decan-3-yl]acetate
(3S,4R)-3-ethyl-1-(3-methoxypyrazin-2-yl)-4-methylpiperidin-4-ol
1-(4-chlorophenyl)-3-(furan-2-yl)-4-[2-(3-hydroxyazetidin-1-yl)-2-oxoethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{[4-(1H-1,3-benzodiazol-2-yl)cyclohexyl]methyl}-2-(2-oxo-1,2-dihydropyridin-1-yl)acetamide
N-[1-({benzyl[(4-methyl-1,3-thiazol-5-yl)methyl]carbamoyl}methyl)-1H-pyrazol-4-yl]thiophene-3-carboxamide
N-[(3R,4S)-1-(1,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-4-propylpyrrolidin-3-yl]methanesulfonamide
2-methyl-1-(1-{[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}azetidin-3-yl)piperidine
6-fluoro-N-methyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1H-1,3-benzodiazole-2-carboxamide
1-methyl-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
1-(3-chloro-2-fluorophenyl)-2-(1H-imidazol-4-yl)-1H-imidazole
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}quinoline-8-carboxamide
1-(azepan-1-yl)-3-(3-{[benzyl(methyl)amino]methyl}phenoxy)propan-2-ol
2-(3-fluoro-4-hydroxyphenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one
1-[(2-chloro-4-fluorophenyl)methyl]-N-[(3S)-2-oxoazepan-3-yl]-1H-1,2,3-triazole-4-carboxamide
1-{8-methylimidazo[1,2-a]pyridine-2-carbonyl}-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
3-(5-hydroxy-4,4-dimethylpentyl)-1-(2-methoxy-6-methylphenyl)urea
4-[3-(aminomethyl)phenyl]-N-(pyridin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
1-[1'-(2-methoxypyridine-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one