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2-(4-carboxy-4-hydroxypiperidin-1-yl)-6-phenylpyridine-3-carboxylic acid
2,6-diamino-4-[5-(2-cyanophenyl)furan-2-yl]-5,6,7,8-tetrahydroquinoline-3-carbonitrile
[(1-cyclopentylpiperidin-3-yl)methyl][(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl][2-(piperidin-1-yl)ethyl]amine
3-({[(2,3-difluorophenyl)methyl]amino}methyl)-N,N-diethylpyridin-2-amine
(5S,9aS,9bS)-2-cyclopentyl-5-(3-methoxyphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-(1-benzyl-1H-pyrazol-4-yl)-2-[4-(1H-pyrazol-1-ylmethyl)piperidin-1-yl]acetic acid
4-[(1E)-3-[3-(2-hydroxyethyl)-4-(thiophen-2-ylmethyl)piperazin-1-yl]prop-1-en-1-yl]-2-methoxyphenol
7-[(1R,4S)-1,7,7-trimethyl-3-oxo-2-oxabicyclo[2.2.1]heptane-4-carbonyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
4-ethyl-1-[(5-methylthiophen-2-yl)methyl]-1,4-diazepan-5-one
N-benzyl-2-(1-ethylpiperidin-4-yl)-N-[(3-methylpyridin-2-yl)methyl]acetamide
4-[4-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]pyrimidin-2-amine
N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}acetamide
2-({3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}methyl)-3,4-dimethoxypyridine
2-(2-methyl-1H-indol-3-yl)-1-(7-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
5-({4-phenyl-5-[5-(1H-pyrazol-5-yl)furan-2-yl]-1H-imidazol-1-yl}methyl)-1H-1,2,3,4-tetrazole
1-ethyl-N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]-1H-pyrazole-4-carboxamide
4-(4-methoxyphenoxymethyl)-1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidine
2-[5-(methanesulfonylmethyl)pyridin-2-yl]-2,7-diazaspiro[4.5]decan-6-one
1-(3-chlorophenyl)-4-[1-(cyclopropylmethyl)piperidin-3-yl]piperazine
N-{[(2-fluoro-4-methylphenyl)carbamoyl]methyl}-2-(2-methyl-1H-indol-3-yl)acetamide
4-[2-(3,5-difluorophenyl)acetyl]-6-[(3-methoxyphenyl)methoxy]-1-(pyridin-2-ylmethyl)-1,4-diazepan-2-one
1-cyclopentyl-N-(1H-indol-4-ylmethyl)-6-oxopiperidine-3-carboxamide
2-amino-4-[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]-6-(1H-pyrrol-2-yl)pyridine-3-carbonitrile
methyl 7-oxo-3-(quinolin-5-ylmethyl)-9-[2-(thiophen-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-[(4aR,7aS)-6,6-dioxo-4-(1-phenylcyclopropanecarbonyl)-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-[2-(pyrrolidin-1-yl)benzoyl]piperidine
4-(4-methoxyphenoxy)-N-[(5-methyl-1,2-oxazol-3-yl)methyl]benzamide
methyl[(7-methyl-1H-1,3-benzodiazol-2-yl)methyl]{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}amine
5-[(4-fluorophenyl)methyl]-5-[1-(4-methylpentanoyl)piperidin-4-yl]-3-(oxolan-2-ylmethyl)imidazolidine-2,4-dione
5-cyclopropanecarbonyl-1'-(4-fluoro-2-methylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-methyl-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-2-propyl-1,3-thiazole-4-carboxamide
1-{1-[4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]-1,2,3,6-tetrahydropyridin-4-yl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
(4aR,8aS)-6-[(2-methoxynaphthalen-1-yl)methyl]-1-[3-(2-oxopyrrolidin-1-yl)propyl]-decahydro-1,6-naphthyridin-2-one
1-(2-{[3-(trifluoromethyl)phenyl]methyl}morpholine-4-carbonyl)cyclopropane-1-carboxamide
1-(benzenesulfonyl)-3-(4-methoxy-3,5-dimethylbenzoyl)piperidine
N-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamide
(1S,5R)-3-[2-(3,4-dichlorophenyl)acetyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-methanesulfonylpiperidine
2-{1-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-1H-1,2,3-triazol-4-yl}benzoic acid
N-({7-[1-(4-methoxyphenyl)cyclopentanecarbonyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)oxane-4-carboxamide
[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]({[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl})amine
N-{1-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
3-(1-ethyl-1H-imidazol-2-yl)-1-[(2,3,5,6-tetrafluoro-4-methoxyphenyl)methyl]piperidine
1-cyclobutyl-4'-(2,2-dimethylpropyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-[(2-ethyl-1,3-thiazol-4-yl)methyl]-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
1-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-2-(4-methyl-1H-pyrazol-1-yl)ethan-1-one
1-({3-[(2,4,6-trimethylpyridin-3-yl)carbamoyl]phenyl}methyl)piperidine-3-carboxamide
3-cyclopropyl-5-(2-fluoro-6-methoxyphenyl)-1-methyl-1H,4H-pyrazolo[3,4-d]imidazole
{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)(thiophen-3-ylmethyl)amine
{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}[1-(thiophen-2-yl)ethyl]amine