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3-fluoro-2-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine
N-[2-(2-methylpropanesulfonyl)ethyl]-3-(1H-pyrazol-1-yl)benzamide
methyl 4-[ethyl(1-hydroxypropan-2-yl)carbamoyl]benzoate
1-{1-[3-cyclopentyl-1-(2-fluorophenyl)-1H-1,2,4-triazol-5-yl]ethyl}-4-methylpiperazine
1-{3-[(2-methylprop-2-en-1-yl)oxy]benzoyl}-4-phenylpiperidin-4-ol
(3S,4R)-N,N-dimethyl-4-(4-methylphenyl)-1-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}pyrrolidin-3-amine
1-benzyl-8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]pent-4-enamide
2-[9-(2-hydroxyacetyl)-7-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl]acetamide
methyl (1R,3S,3aR,6aS)-5-methyl-4,6-dioxo-3-[1-(propan-2-yl)-2,3-dihydro-1H-indol-5-yl]-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
N-(carbamoylmethyl)-2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
(2R,3S,6R)-3-(3-methoxyphenyl)-5-(1,3-thiazol-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-4-(2-methoxyphenyl)-2-methylpiperazine
N-[3-(pyridin-2-yl)propyl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
2-{[2,5-dioxo-4-(piperidin-4-yl)-4-(pyridin-3-yl)imidazolidin-1-yl]methyl}benzonitrile
3-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]-1-phenylpropan-1-one
4-[3-(3-methoxyphenyl)propanoyl]-1-(4-methylphenyl)piperazin-2-one
N-{[1-(1H-imidazol-4-ylmethyl)piperidin-3-yl]methyl}-2-(2-methoxyphenoxy)acetamide
(1R,5R)-3-[3-(3-methoxyphenyl)benzoyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonane
4-[2-(3-methoxyphenyl)piperidine-1-carbonyl]-1-methyl-1H-indole
N-[2-(4-methoxyphenyl)ethyl]-3-[(3S,4R)-1-(2-methylpropyl)-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]propanamide
3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]propanamide
2-(dimethylamino)-N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-4-methylpyrimidine-5-carboxamide
2-{1-cyclopentyl-4-[(2,4-dimethoxy-3-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
[4-benzyl-1-(8-chloroquinolin-2-yl)piperidin-4-yl]methanol
N-(2-fluoro-4-methoxyphenyl)-4-(3-phenylpropyl)-1,4-diazepane-1-carboxamide
N,3-dimethyl-N-[1-(1,2-oxazol-3-yl)ethyl]-5-propyl-1-benzofuran-2-carboxamide
1-(4-acetylpiperazin-1-yl)-4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]butan-1-one
{[2-(3-chlorophenyl)-7-methylquinolin-3-yl]methyl}(1,3-thiazol-2-ylmethyl)amine
1-{3-[ethyl(pyridin-4-ylmethyl)amino]piperidin-1-yl}-4-(4-fluorophenyl)butane-1,4-dione
N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-2,3-dihydro-1H-indene-1-carboxamide
7-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
6-ethyl-5-methyl-N4-[1-(4-methyl-1H-imidazol-2-yl)propyl]pyrimidine-2,4-diamine
3-{2-oxo-2-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethyl}-1,3-oxazolidin-2-one
4-({[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]amino}methyl)-2,6-dimethylphenyl acetate
3-{1-[1-cyclohexyl-3-(cyclopropylmethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl]-N-methylformamido}-N-methylpropanamide
methyl 3-(quinoline-8-sulfonamido)-5-[(1,3-thiazol-5-ylformamido)methyl]benzoate
1-[(4S,4aS,8aS)-4-hydroxy-4-phenyl-decahydroquinolin-1-yl]-2-(2-ethyl-1H-imidazol-1-yl)ethan-1-one
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-N-methyl-6-oxo-1-(3-phenylpropyl)piperidine-3-carboxamide
7-[(1-cyclohexyl-1H-imidazol-5-yl)methyl]-2-oxa-7-azaspiro[4.5]decane
3-(3-chlorophenyl)-N-{[1-(methoxymethyl)cyclopropyl]methyl}-3-phenylpropanamide
2-{3-[(4-fluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}pyridine-3-carbonitrile
3-[ethyl({[2-(pyridin-2-yl)pyrimidin-5-yl]methyl})amino]-1λ6-thiolane-1,1-dione
3-(2-{3-[(dimethylamino)methyl]phenyl}-1H-imidazol-1-yl)-N,2-dimethylpropanamide
1-[(1-methyl-1H-imidazol-2-yl)methyl]-8-(6-methylpyridin-2-yl)-1,8-diazaspiro[4.5]decane
(2S,4R)-4-amino-1-[(2-methoxypyridin-3-yl)methyl]-N-methylpyrrolidine-2-carboxamide
4'-(3,3-dimethylbutyl)-1-(2,2-dimethylpropanoyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
3-(2-phenylethyl)-N-{[3-(trifluoromethoxy)phenyl]methyl}-1,2-oxazole-5-carboxamide
1-(methoxymethyl)-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]cyclobutane-1-carboxamide
N-[(2,6-difluorophenyl)methyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide