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2-{3-[({1-[(2-fluorophenyl)methyl]piperidin-3-yl}amino)methyl]phenoxy}ethan-1-ol
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-1-(2-phenylethyl)piperidin-4-amine
2-[4-(2H-1,3-benzodioxol-4-ylmethyl)-1-(1-methylpiperidin-4-yl)piperazin-2-yl]ethan-1-ol
1-{1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}-4-(2-methylphenyl)piperazine
6-[1-(6-ethyl-2-methylpyrimidin-4-yl)piperidin-4-yl]-2,3-dimethyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
(3E)-1-{4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pent-3-en-1-one
5-{[3-(3-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
1-[3-(3-fluoro-4-phenylbenzoyl)piperidin-1-yl]-2-(pyrimidin-2-ylsulfanyl)ethan-1-one
N-[1-(4-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine-1-carbonyl}phenyl)-1H-pyrazol-4-yl]pyridine-3-carboxamide
2-methyl-5-{3-[2-(propan-2-yloxy)phenyl]phenyl}-1,3,4-oxadiazole
1-(methoxymethyl)-N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}cyclobutane-1-carboxamide
3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}piperidine
({2-[2-(dimethylamino)ethoxy]-3-methoxyphenyl}methyl)(ethyl)[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amine
3-(2,5-dioxoimidazolidin-4-yl)-N-[2-(1H-indol-3-yl)ethyl]propanamide
4-{2-[1-tert-butyl-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]phenyl}morpholine
2-[4-(furan-3-ylmethyl)-6-hydroxy-1,4-diazepan-1-yl]-1,3-thiazole-4-carboxamide
1-(2,5-difluorobenzoyl)-4-(2-methylpropyl)-1,4-diazepan-5-one
{[5-(2-chlorophenyl)-1,2-oxazol-3-yl]methyl}[1-(1H-pyrazol-1-yl)propan-2-yl]amine
1-(oxan-4-yl)-4-{[4-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}piperazine
2-(4-methyl-1,3-oxazole-5-carbonyl)-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
{[6-(cyclohexylmethoxy)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amine
8-methyl-N-[(2-methylphenyl)methyl]-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
N-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)-2-methyl-2-phenoxypropanamide
2-(4-{2-[(dimethylamino)methyl]phenyl}phenoxy)propanamide
5-{[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-{1-[2-(dimethylamino)ethyl]-3-(3-fluorophenyl)-2,5-dioxopyrrolidin-3-yl}-N-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]acetamide
2-(dimethyl-1,3-thiazol-5-yl)-1-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}ethan-1-one
N-[1-(cyclopropylmethyl)-1H-pyrazol-5-yl]-2-[4-(9H-purin-6-yl)-1H-pyrazol-1-yl]acetamide
8-{[4-(furan-2-yl)phenyl]methyl}-1-(2-methoxyethyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-[1-(2,3-dimethylquinoxaline-6-carbonyl)piperidin-4-yl]-2-methylpyrimidin-4-ol
(3E)-N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)pent-3-enamide
(2R,6S)-2,6-dimethyl-4-(1-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}piperidin-4-yl)morpholine
2-phenyl-7-(quinoline-2-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-{[2-(methylsulfanyl)phenyl]methyl}-3-(4H-1,2,4-triazol-3-yl)piperidine
2-(cyclopropylmethyl)-9-(1,2,4-oxadiazol-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-[4-(morpholine-4-carbonyl)piperazin-1-yl]-5,6,7,8-tetrahydroquinazolin-2-amine
1-(carbamoylmethyl)-N-[(1-propyl-1H-imidazol-2-yl)methyl]piperidine-4-carboxamide
1-oxo-N-(5,6,7,8-tetrahydronaphthalen-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
(1-{1-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]piperidin-3-yl}piperidin-4-yl)methanol
1-[(4-fluorophenyl)methyl]-4-(morpholine-4-carbonyl)-2-(propan-2-yl)-1,4-diazepane
1,6-dimethyl-2-oxo-N-[1-(thiophen-2-ylmethyl)piperidin-3-yl]-1,2-dihydropyridine-3-carboxamide
N-{4-[2-(2,3-difluorophenyl)-1H-imidazol-1-yl]-2-methylphenyl}-2-(dimethylamino)acetamide
1-(3-fluoro-4-methylbenzoyl)-3-(3-methoxypropyl)piperidine
3-methyl-1-(4-methyl-2-oxo-2H-chromen-7-yl)-3-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)urea
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-{[(2-methoxyethyl)amino]methyl}piperidin-2-one
2-butyl-N-(2-methylprop-2-en-1-yl)-1,3-benzoxazole-5-carboxamide
2-({ethyl[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)-4-fluorophenol
2-(2-methoxy-4-methylphenoxymethyl)-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-1,3-oxazole-4-carboxamide
3-{5-[(2,5-dimethoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl}-1-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]propan-1-one
2-(5-{[2-(pyridin-2-yl)pyrrolidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)pyrazine