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(3S,4R)-1-[(3-cyclohexyl-1,2-oxazol-5-yl)methyl]-4-(3-fluorophenyl)pyrrolidine-3-carboxylic acid
3-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-1-[3-(2-methyl-1,3-thiazol-4-yl)phenyl]urea
7-methyl-3-{[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl}-3,7,11-triazaspiro[5.6]dodecan-12-one
(3S,5R)-1-(1-methyl-1H-pyrrole-2-carbonyl)-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxylic acid
2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-(2,2,2-trifluoroethyl)acetamide
4-[5-({[2-(2,5-dimethylphenoxy)ethyl](methyl)amino}methyl)thiophen-2-yl]-2-methylbut-3-yn-2-ol
N-[(2R,3R)-1'-[(2-hydroxy-6-methoxyphenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]thiophene-3-carboxamide
N-(cyclohexylmethyl)-5-[2-(hydroxymethyl)piperidine-1-carbonyl]-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
6-[1-(1-benzofuran-2-ylmethyl)piperidin-4-yl]-2-methylpyrimidin-4-ol
N-cyclopropyl-4-methoxy-2-({1-[(4-methylphenyl)methyl]piperidin-4-yl}oxy)benzamide
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(1-phenylcyclopropyl)acetamide
N-[(2-fluorophenyl)methyl]-4-(4-{[3-(pyridin-3-yloxy)propyl]amino}piperidin-1-yl)benzamide
1-{3-[ethyl(pyridin-4-ylmethyl)amino]piperidin-1-yl}-5-phenylpentan-1-one
(1-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)methanol
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-(1-benzylcyclopropyl)-1H-pyrazole-3-carboxamide
2-chloro-N-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]pyridine-4-carboxamide
1-[2-({[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}amino)ethyl]piperidin-2-one
7-(2,2-dimethylpropyl)-N-(2-methoxyphenyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
N-methyl-6-oxo-N-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}piperazine-2-carboxamide
methyl 4-(5-{[3-(benzyloxy)piperidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)benzoate
N,N-dimethyl-3-[2-oxo-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-8-yl]propanamide
6-{3-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}-9H-purine
(2S)-1-{4-[(4-fluorophenyl)methyl]piperidin-1-yl}-3-hydroxy-2-(methylamino)propan-1-one
4-{1-[4-(3-{[4-(furan-2-carbonyl)piperazin-1-yl]methyl}phenoxy)piperidin-1-yl]-1-oxopropan-2-yl}-1,2-dihydrophthalazin-1-one
5-tert-butyl-N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]-1,3,4-oxadiazol-2-amine
N-[3-(dimethylamino)propyl]-1-(3,4-dimethylbenzoyl)-N-methylpiperidin-3-amine
2-{2-[(4-aminoazepan-1-yl)methyl]-4-chlorophenoxy}acetic acid
5-[2-(aminomethyl)-5-methyl-2,3-dihydro-1-benzofuran-7-yl]-N-(2-methylpropyl)furan-2-carboxamide
2-chloro-4-{[1-cyclohexyl-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]methyl}phenol
N-[(3S,4R)-4-(5-methylfuran-2-yl)-1-[(2-phenyl-1,3-oxazol-4-yl)methyl]pyrrolidin-3-yl]acetamide
1-{4-[4-(2-aminopropan-2-yl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}-5-methylhexan-1-one
2-(5-acetylthiophen-3-yl)-N-(cyclohex-1-en-1-ylmethyl)acetamide
[(4-fluorophenyl)methyl](pyridin-4-ylmethyl){[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}amine
(4aR,7aS)-1-(pyridin-2-ylmethyl)-4-(1,3-thiazol-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-[2-(propan-2-yl)oxane-4-carbonyl]-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
2-cyclopropanecarbonyl-8-[2-(2-methylphenyl)acetyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-(3-methoxyphenoxy)-3-{[1-(1-methylcyclopropyl)ethyl]amino}propan-2-ol
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(1H-pyrazole-3-carbonyl)pyrrolidine-3-carboxylic acid
1-[(2,3-dimethyl-1H-indol-7-yl)methyl]-N,N-dimethylazepan-4-amine
N-{[6,7-dimethoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-(2-methoxyethyl)-4-phenylbenzamide
2,2-dimethylpropyl 7-methyl-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxylate
(4S)-1-(5-ethyl-1H-pyrrole-2-carbonyl)-3,3,4-trimethylpiperidin-4-ol
3-{2-[2-(3-methoxyphenyl)piperidin-1-yl]-2-oxoethyl}-1,3-diazinane-2,4-dione
N-(3-fluoro-4-methylphenyl)-2-[(5-oxo-1-propylpyrrolidin-3-yl)amino]acetamide
2-({6-[3-fluoro-5-(propan-2-yloxy)phenyl]pyrimidin-4-yl}amino)ethan-1-ol
(5-{2-[3-(4-fluorophenyl)oxolan-3-yl]-1H-imidazol-1-yl}-1H-1,3-benzodiazol-2-yl)methanol
1-phenyl-4-{[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}piperazin-2-one
N-[(2,6-difluoro-3-methoxyphenyl)methyl]-1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
N-[1-(2,6-dimethylphenoxy)propan-2-yl]-3-(1-methyl-1H-pyrazol-5-yl)propanamide
methyl 3-{[1-(cyclopropylmethyl)-5-(3,5-difluorobenzoyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]formamido}propanoate