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6-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-N-ethyl-N-methylpyridine-3-carboxamide
1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-methanesulfonyl-1,4-diazepane
N-[2-(4-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-3-(2-oxopyrrolidin-1-yl)propanamide
3-methyl-2-(1-{4-[2-(1H-pyrazol-1-ylmethyl)phenyl]-1H-1,2,3-triazol-1-yl}ethyl)pyridine
3-chloro-6-{3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}pyridazine
N2,N2-dimethyl-N5-(oxan-4-yl)-5,6,7,8-tetrahydroquinazoline-2,5-diamine
3-(3-methoxyphenyl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1H-pyrazole-4-carboxamide
1-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-3-(2,6-dimethoxypyridin-3-yl)urea
3-({2-[(1S,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamido}methyl)-4-methylbenzoic acid
{[2-cyclopropylmethanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}[(4-fluorophenyl)methyl]methylamine
4-[(2,3-dimethoxyphenyl)methyl]-7-{[4-(pyridin-3-yloxy)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
[2-fluoro-5-(2-methyl-5-propylpyrimidin-4-yl)phenyl]methanol
2-(4-benzyl-2-oxopyrrolidin-1-yl)-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]acetamide
N-[(2R,3R)-2-methoxy-1'-(3-phenylpropyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]thiophene-3-carboxamide
N-(2-cyclopropylphenyl)-2-methyl-4-[(3-methylphenyl)methyl]-3-oxopiperazine-1-carboxamide
N-cyclopropyl-2-{4-[2-(pyridin-2-yl)-1H-imidazol-1-yl]phenyl}acetamide
1-(3-chlorobenzoyl)-4-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine
2-(morpholin-4-yl)-N-(5-oxo-1-phenylpyrrolidin-3-yl)benzamide
(1-{2-[4-(naphthalen-2-yl)-1H-1,2,3-triazol-1-yl]ethyl}piperidin-2-yl)methanol
3-fluoro-N-({7-[(3-fluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)benzamide
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-(propan-2-yl)piperidine-3-carboxamide
1-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}-4-(thiophene-2-carbonyl)piperazine
1-(3-{[({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]methyl}phenyl)ethan-1-one
1-[3-(2H-1,3-benzodioxol-5-yl)-2-methylpropyl]-3-[4-(propan-2-yl)-1H-pyrazol-5-yl]piperidine
6-(furan-3-yl)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
5-(thiophen-3-ylmethyl)-2-(3,4,5-trimethoxyphenyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
1-[2-(3-chlorophenyl)ethyl]-4-[(thian-4-yl)amino]pyrrolidin-2-one
4-{4-[3-(3-hydroxy-3-methylbut-1-yn-1-yl)benzoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-1-methylpiperidin-4-ol
N-[(1S,6R)-6-carbamoylcyclohex-3-en-1-yl]-3,5-dimethyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
2-(5-{[3-(pyridin-4-yl)azetidin-1-yl]sulfonyl}thiophen-2-yl)pyridine
(1-{[7-chloro-4-(morpholin-4-yl)quinazolin-2-yl]methyl}piperidin-4-yl)(thiophen-2-yl)methanol
1-methyl-N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-indole-4-carboxamide
4-(naphthalen-2-yloxy)-1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}piperidine-4-carboxylic acid
N-({1-[(5-ethylfuran-2-yl)methyl]piperidin-3-yl}methyl)-2,3-dimethoxybenzamide
1-methyl-3-[(2-methyl-5-oxopyrrolidin-1-yl)methyl]-1,2-dihydroquinolin-2-one
N-[2-(2,5-dimethylphenoxy)ethyl]-N-methyl-2-[methyl(pyridin-3-ylmethyl)amino]acetamide
(3E)-N-[4-methoxy-2-(2-methylpropanamido)phenyl]pent-3-enamide
1-[1-(2-amino-2-methylpropanoyl)piperidin-4-yl]-N-(2-phenylethyl)piperidine-3-carboxamide
N-(1-carbamoylcyclopentyl)-3-(4-hydroxyphenyl)-1H-pyrazole-5-carboxamide
N-(1H-1,3-benzodiazol-2-ylmethyl)-2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
(4aS,8aR)-6-(1H-imidazol-4-ylmethyl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
N-[2-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-5-propyl-1,2-oxazole-3-carboxamide
3-{2-[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidin-1-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
N-[2-(2,4-difluorophenyl)-1-{1-[(3-methylphenyl)methyl]piperidin-4-yl}ethyl]-N-methylfuran-2-carboxamide
N-[2-(7-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-1-(oxolan-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
11-(benzylamino)-4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
3-(2-chlorophenyl)-1-[4-(hydroxymethyl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-1-yl]propan-1-one
7-[(2,3-difluorophenyl)methyl]-2-(2-methylpyridine-3-carbonyl)-2,7-diazaspiro[4.5]decane
4-[2-(4-chlorophenyl)morpholin-4-yl]-N-cyclopentyl-4-oxobutanamide
(2R,3R,6R)-3-(4-methylphenyl)-5-(3-methylpyridine-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane