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2-[4-(5-chloro-2-methoxyphenyl)-1H-pyrazol-1-yl]acetic acid
5-phenyl-N-[2-(pyrrolidine-1-sulfonyl)ethyl]-1H-pyrazole-3-carboxamide
2-(adamantan-1-yl)-4-hydroxy-N-[(3R)-piperidin-3-yl]pyrimidine-5-carboxamide
2,N4-dimethyl-N4-(quinolin-3-ylmethyl)pyrimidine-4,6-diamine
9-methoxy-7-(2-methoxyphenyl)-4-(2-methylpropyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-(3-methylbutyl)-8-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-(4-chlorophenyl)-N-methyl-N-[1-(pyridin-3-yl)propyl]butanamide
1-(3,5-dimethylphenyl)-4-(5-fluoro-1-methyl-1H-indole-2-carbonyl)piperazin-2-one
3-({5-[4-(2-phenylethyl)piperidine-1-carbonyl]pyridin-2-yl}amino)propan-1-ol
methyl 3-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-7-oxo-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-(4-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]methyl}phenyl)-6-propyl-3,4-dihydropyrimidin-4-one
3-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-2-(methylsulfanyl)pyridine
2-methyl-6-{[5-(oxolan-3-yl)-4-phenyl-1H-imidazol-1-yl]methyl}pyrimidin-4-ol
N-[(3S,4R)-4-propyl-1-(quinolin-2-ylmethyl)pyrrolidin-3-yl]acetamide
2-(methylsulfanyl)-N-({4-[(3-phenylpropyl)amino]quinazolin-2-yl}methyl)benzamide
4-hydroxy-N-[(1S)-1-(3-methoxyphenyl)ethyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
2-methyl-5-[4-(3-phenylpropyl)-1,4-diazepane-1-carbonyl]-1,4-dihydropyridin-4-one
1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethan-1-one
5-[2-(4-fluorophenoxy)ethyl]-2-methoxybenzamide
N-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-1-oxa-8-azaspiro[4.5]decan-3-amine
4-{[1-(furan-3-ylmethyl)piperidin-4-yl]oxy}-N-(pyridin-2-ylmethyl)benzamide
N-(6-methoxypyridin-3-yl)-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl][1-(2-fluorophenyl)propan-2-yl]amine
N-({5-methyl-2-[3-(propane-2-sulfonamido)phenyl]-1,3-oxazol-4-yl}methyl)-2-(propan-2-yl)oxane-4-carboxamide
3-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-1-{8-methyl-2,8-diazaspiro[4.5]decan-2-yl}propan-1-one
2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]-1-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}ethan-1-one
2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)-N-{[2-(trifluoromethyl)phenyl]methyl}acetamide
8-(3,5-dichloro-4-methylbenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
7-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
1-(2-aminoethyl)-N-benzyl-N-[(1R,2R)-2-hydroxycyclohexyl]-1H-1,2,3-triazole-4-carboxamide
4-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-1-{[2-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
N-(3-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-oxopropyl)methanesulfonamide
1-benzyl-4-[(3-cyclopropyl-1H-pyrazol-5-yl)methyl]piperazine
2-amino-N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-1,3-benzothiazole-5-carboxamide
3-{[4-(1,3-dimethyl-1H-pyrazol-5-yl)-4H-1,2,4-triazol-3-yl]methyl}pyridine
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-amine
(4aR,7aS)-1-(2-hydroxyethyl)-4-(5-methylthiophene-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(2-{7-[(4-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)oxolane-2-carboxamide
(3S,7S)-5-(1-methyl-6-oxo-1,6-dihydropyridazine-3-carbonyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
1-[3-(4-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}phenoxymethyl)piperidin-1-yl]-2-(thiophen-2-yl)ethan-1-one
5-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
(3S,4R)-1-(2-methanesulfonylethyl)-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
(1R,2R,6S,7S)-4-(4-propylbenzoyl)-10-oxa-4-azatricyclo[5.2.1.02,6]decane
2-[1-(2H-1,3-benzodioxol-5-yl)-3-cyclopropyl-1H-1,2,4-triazol-5-yl]-3,5-difluoropyridine
1-(2-{[(isoquinolin-5-ylmethyl)(methyl)amino]methyl}-5-methoxyphenoxy)-3-(pyrrolidin-1-yl)propan-2-ol
2-(2-methylpyrimidin-5-yl)-4-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)quinoline
(2R)-N-[1-(4-methoxyphenyl)-4-(propan-2-yloxy)-1H-indazol-3-yl]oxolane-2-carboxamide
ethyl 3-[(4-fluorophenyl)methyl]-1-{4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carbonyl}piperidine-3-carboxylate
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-2-(3-methyl-2-oxo-1,2,3,4-tetrahydroquinazolin-1-yl)acetamide
(6S)-6-{4-[(3-methylphenyl)methyl]piperazine-1-carbonyl}piperidin-2-one