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(1S,5R)-6-(5-methyl-1,2-oxazole-4-carbonyl)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
3-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-1-(1-oxo-2,3-dihydro-1H-inden-5-yl)urea
2-[(3-methylthiophen-2-yl)methyl]-2,8-diazaspiro[4.5]decane
N-[(1S,2R)-2-(cycloheptylamino)cyclobutyl]-4-(1H-1,2,4-triazol-1-yl)butanamide
methyl({4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl})(quinoxalin-6-ylmethyl)amine
1-(2-methoxyphenyl)-4-(2-oxoimidazolidine-4-carbonyl)piperazin-2-one
3-(hydroxymethyl)-1-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carbonyl]piperidin-3-ol
3-(2H-1,3-benzodioxol-5-yl)-N-methyl-N-[2-(1,2,4-oxadiazol-3-yl)ethyl]propanamide
9-methoxy-3-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-10-(pyrrolidine-1-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
(3R,4S)-1-[(5-methyl-2,1,3-benzothiadiazol-4-yl)sulfonyl]-4-phenylpyrrolidin-3-amine
(4aS,8aR)-1-(2-aminoethyl)-6-(5-phenylpentanoyl)-decahydro-1,6-naphthyridin-2-one
2-(adamantan-1-yl)-N-(2-methanesulfonylethyl)acetamide
9-(4-chloro-2-methylbenzoyl)-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
methyl 1-benzyl-5-[(2-ethylbutyl)amino]-3-(oxolane-2-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[2-(dimethylamino)ethyl]-3-(2-methylphenyl)-3-phenylpropanamide
(4aS,8aS)-2-[2-(morpholin-4-yl)pyrimidine-5-carbonyl]-decahydro-2,7-naphthyridin-4a-ol
(4S)-4-hydroxy-3,3,4-trimethyl-N-(2-phenylphenyl)piperidine-1-carboxamide
(3S,4R)-1-[(1-methyl-1H-indol-2-yl)methyl]-4-(3-methylthiophen-2-yl)piperidin-3-ol
4-(4-chlorophenyl)-N-[(3R,4R)-4-hydroxypiperidin-3-yl]butanamide
N-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
(3E)-1-(4-ethyl-3,3-dimethylpiperazin-1-yl)hex-3-en-1-one
3-[9-methoxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]-1H-pyrazol-5-amine
N,1-dimethyl-6-propyl-N-(1,3-thiazol-2-ylmethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-2-(trifluoromethyl)-1H-1,3-benzodiazole
(5-{[1-(3-chlorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}furan-2-yl)methanol
1-(4-ethylpiperazin-1-yl)-3-{1-[1-(4-methylpyridin-2-yl)propan-2-yl]piperidin-4-yl}propan-1-one
4-acetyl-N-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]benzamide
2-(dimethyl-1,2-oxazol-4-yl)-N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methylacetamide
3-[(1S)-2-hydroxy-1-phenylethyl]-1-{4-[(1-methylpiperidin-4-yl)oxy]phenyl}urea
2-(1-ethylpiperidin-4-yl)-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)acetamide
N-{[3-(3-methylbutyl)-3H-imidazo[4,5-b]pyridin-2-yl]methyl}-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
6-{[4-(1-benzyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]methyl}-2-methylpyrimidin-4-ol
N4-[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-5-methylpyrimidine-2,4-diamine
2-[(1-{2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}piperidin-4-yl)oxy]pyrimidine
5-(5-methyl-1H-indol-3-yl)thiophene-2-sulfonamide
2-[2-({4-[(2-methyl-1H-imidazol-1-yl)methyl]piperidin-1-yl}methyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]acetic acid
N,N-dimethyl-4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine-1-sulfonamide
2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
(3S,7S)-5-(thiophene-3-carbonyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
1-[2-(4-methanesulfonylpiperazin-1-yl)-2-oxoethyl]-3-methoxy-1,2-dihydropyridin-2-one
{2-[(2H-1,3-benzodioxol-4-ylmethyl)[(5-methylthiophen-2-yl)methyl]amino]ethyl}dimethylamine
3-(1-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl)-5-(propan-2-yl)-1,2-oxazole
(2E)-3-(3,4-dimethoxyphenyl)-1-{3-[5-(4-fluorophenyl)-2-methylpyrimidin-4-yl]piperidin-1-yl}prop-2-en-1-one
1-[1-(4-ethylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-(5-methyl-1H-pyrazol-1-yl)propan-1-one
1-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-phenylpiperidine
ethyl 1-(4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-3-(2-phenylethyl)piperidine-3-carboxylate
N-(1-hydroxybutan-2-yl)-3-methyl-N-[(5-methylthiophen-2-yl)methyl]furan-2-carboxamide
2-(2-{1-[2-(3,4-dimethylphenoxy)acetyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
N-cyclopropyl-1-(1-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}piperidin-4-yl)piperidine-3-carboxamide
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(1H-imidazol-2-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane