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1-(furan-2-ylmethyl)-4-[4-(oxolan-2-ylmethyl)-5-[(2-phenylethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]piperidine
3-phenoxy-N-[1-({[2,2,2-trifluoro-1-(furan-2-yl)ethyl]carbamoyl}methyl)-1H-pyrazol-4-yl]propanamide
4-ethyl-1-methyl-3-[1-(5-propyl-1,2-oxazole-3-carbonyl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
5-chloro-2-(3-methyl-1,2,4-oxadiazol-5-yl)-3-phenyl-1H-indole
7-(3-chlorophenyl)-4-(pyridine-2-carbonyl)-9-(thiophen-3-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-{[4-(adamantan-2-yl)piperazin-1-yl]methyl}-4-(pyrimidin-2-yl)phenol
2-amino-4-(5-chloro-2,3-dimethoxyphenyl)-6-(1H-pyrrol-2-yl)pyridine-3-carbonitrile
[(3R,4R)-1-[1-(2-chlorophenyl)piperidin-4-yl]-4-[(dimethylamino)methyl]pyrrolidin-3-yl]methanol
4-{[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl]methyl}benzamide
4-({1-[(2,3-difluorophenyl)methyl]-3-hydroxy-2-oxopiperidin-3-yl}methyl)piperazin-2-one
2-({3-methyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl}sulfanyl)-N-(2-phenylethyl)acetamide
9-[(2R)-2-cyclohexyl-2-hydroxyacetyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-1-{4-[hydroxy(pyridin-2-yl)methyl]piperidin-1-yl}ethan-1-one
N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
6-[(2-fluorophenyl)methoxy]-1-(2-methylpropyl)-4-[1-(propan-2-yl)piperidin-4-yl]-1,4-diazepan-2-one
N-[(1-cyclopentylpiperidin-4-yl)methyl]-3-(propan-2-yl)-N-(pyridin-3-ylmethyl)-1H-pyrazole-5-carboxamide
(benzylsulfamoyl)(methyl)(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)amine
5-(1-benzofuran-2-ylmethyl)-3-[2-(methylsulfanyl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
1-(furan-2-ylmethyl)-N-[4-(3-methylphenyl)phenyl]piperidine-4-carboxamide
3-{3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1H-indole
2-amino-6-[4-(morpholin-4-ylmethyl)thiophen-2-yl]-4-(pyridin-4-yl)pyridine-3-carbonitrile
4-{[1-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}thiomorpholine
6-(2-chlorophenyl)-N-methyl-N-(1,2-oxazol-5-ylmethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-[(naphthalen-2-ylmethyl)amino]-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
(3S,4S)-3-(dimethylamino)-N-{4-[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]phenyl}-4-hydroxypyrrolidine-1-carboxamide
1-{6-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecan-4-yl]pyridin-3-yl}ethan-1-one
[(2-tert-butyl-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl)sulfamoyl]dimethylamine
2-amino-3-ethyl-N-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-3H-imidazo[4,5-b]pyridine-6-carboxamide
(3R,4S)-1-[2-(difluoromethoxy)benzoyl]-4-propylpyrrolidin-3-amine
1-(7-chloro-4-methylquinolin-2-yl)-3-(piperidin-1-ylmethyl)pyrrolidin-3-ol
1-[5-methyl-6-(4-methylpiperazine-1-carbonyl)thieno[2,3-d]pyrimidin-4-yl]azocane
3-(pyridin-3-yl)-N-[(7-{[2-(trifluoromethyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]propanamide
1-cyclopentyl-N3-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-4-oxo-N5-(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N-[4-(4-methoxyphenyl)butan-2-yl]-2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
{3-[(5-chlorofuran-2-yl)methyl]-9-(oxan-4-yl)-3,9-diazaspiro[5.5]undecan-1-yl}methanol
3-(3-methoxypropyl)-1-[3-(piperidin-4-ylmethyl)benzoyl]piperidine
N-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
N-[1-(1H-imidazol-1-yl)-3-methylbutan-2-yl]-6-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide
5-[1-(2-chlorobenzoyl)piperidin-4-yl]-3-[2-(dimethylamino)ethyl]-5-(3-methylbutyl)imidazolidine-2,4-dione
1-(carbamoylmethyl)-N-methyl-N-(quinolin-4-ylmethyl)piperidine-3-carboxamide
2-amino-7-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
4-{1-[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-4-yl}thiomorpholine
(1S,5R)-3-[(4-fluorophenyl)methyl]-6-(3-fluoropyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(2-{4-[5-(methoxymethyl)thiophene-2-amido]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]-5-methylpyrazine-2-carboxamide
3-{4-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]piperazin-1-yl}-1-azabicyclo[2.2.2]octane
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-3-(4-methyl-1,3-thiazol-5-yl)propanamide
5-methyl-N-{3-[(1-methylpiperidin-4-yl)oxy]propyl}pyrazolo[1,5-a]pyrimidin-7-amine
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-cyclopropyl-2-methyl-1-benzofuran-5-carboxamide
6-(4H-1,2,4-triazol-4-yl)-N-{2-[(trifluoromethyl)sulfanyl]ethyl}pyridine-3-carboxamide
ethyl 1-[6-(2-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]piperidine-4-carboxylate