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1-[2-({[4-(furan-2-yl)phenyl]methyl}(methyl)amino)ethyl]piperidin-2-one
8-[(3,5-dimethoxyphenyl)methyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
N-cyclooctyl-4-oxo-4-[2-(pyridin-3-yl)piperidin-1-yl]butanamide
N-cyclopropyl-3-(3-hydroxy-3-methylbutyl)-N-[(4-hydroxyphenyl)methyl]benzamide
(3R)-1-{6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carbonyl}pyrrolidin-3-ol
[1-(4-{[2-(cyclohex-1-en-1-yl)ethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carbonyl)piperidin-2-yl]methanol
2-cyclohexyl-5-{[3-(2-methylpiperidin-1-yl)azetidin-1-yl]methyl}pyrimidine
1-{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-4-ethylpiperazine
(1R,5R)-6-(pyridin-2-ylmethyl)-3-(pyrrolidine-1-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
4-[3-(3,4-difluorophenyl)propanoyl]-1-(3-methoxyphenyl)piperazin-2-one
2-(4-ethyl-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]acetamide
4-{3-[(4-cyclopentyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}-2,6-dimethylpyrimidine
methyl({[4-(methylsulfanyl)phenyl]methyl})[3-(1H-pyrazol-1-yl)propyl]amine
(2R,3R)-3-[4-(3-methoxypropyl)piperidin-1-yl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
6-[(3aS,6aR)-3-[3-(morpholin-4-yl)propyl]-2-oxo-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-5-yl]pyridine-2-carbonitrile
N,N-bis(2-methoxyethyl)-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
2-{1-[(4-methanesulfonylphenyl)methyl]piperidin-2-yl}-1H-1,3-benzodiazole
N-{1-[1-(2,1,3-benzothiadiazol-5-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}pyridine-3-carboxamide
4-methoxy-N-[(5-methylpyrazin-2-yl)methyl]-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
N-({7-[(2,4-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)benzenesulfonamide
N-[(3S,4R)-1-(2-aminopyridine-4-carbonyl)-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
2-{4-[2,2-dimethyl-3-(pyrrolidin-1-yl)propyl]piperazin-1-yl}pyrazine
N,N,3,6-tetramethyl-2-[2-(pyridin-3-yl)pyrimidin-5-yl]quinoline-4-carboxamide
methyl 3-{[5-(3-chloro-2-fluorobenzoyl)-1-(cyclopropylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]formamido}propanoate
4-[4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]benzoic acid
methyl 4-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}piperazine-1-carboxylate
1-[2-chloro-5-(pyrrolidine-1-carbonyl)phenyl]-3-[(2-methyl-1,3-thiazol-4-yl)methyl]urea
N-[(2R,3R)-1'-[(3-ethoxy-4-hydroxyphenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
2-(2-methoxy-4-methylphenoxymethyl)-N,N-dimethyl-1,3-oxazole-4-carboxamide
N-{[(3S,4S)-3-hydroxy-1-[2-methyl-2-(1H-pyrrol-1-yl)propanoyl]piperidin-4-yl]methyl}pyrrolidine-1-carboxamide
N-cyclopentyl-N-{[4-(oxolan-3-yloxy)phenyl]methyl}quinoline-2-carboxamide
4-[(4-fluorophenyl)methyl]-1-(3-hydroxybenzoyl)-3-(propan-2-yl)-1,4-diazepan-5-one
4-{4-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]piperazin-1-yl}phenol
4-[(2,3-dimethoxyphenyl)methyl]-3-{2-[4-(2-methoxyethyl)piperazin-1-yl]-2-oxoethyl}piperazin-2-one
2-(2-hydroxyphenoxy)-N-{1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}acetamide
1-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}-4-(2-methylphenoxy)piperidine
4-[(7-fluoro-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
(3R,4R)-1-{[3-(2-hydroxyethoxy)phenyl]methyl}-3-methyl-4-(oxan-4-yl)piperidin-4-ol
2-(1H-indol-5-yl)-N,N-dimethylbenzamide
(3R,4R)-1-[(5-chloro-2,4-dimethoxyphenyl)methyl]-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
6-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]pyridine-2-carbonitrile
benzyl(methyl){[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
2-(5-{[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]methyl}furan-2-yl)benzonitrile
N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
7-[(3,4-difluorophenyl)methyl]-3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
N-{1-[1-(1-methoxypropan-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-4-phenylbutanamide
(1-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)(1-methyl-1H-imidazol-2-yl)methanol
1-(cyclopropylmethyl)-4-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)-2-(propan-2-yl)-1,4-diazepane
N-(cyclohex-1-en-1-ylmethyl)-6-(4-fluorophenyl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
5-phenyl-N-(pyridin-3-ylmethyl)-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-amine