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3-({2-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]acetamido}methyl)-4-methylbenzoic acid
1-[(1R,5R)-6-[(5-chloro-2,4-dimethoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}quinoline-8-carboxamide
1-{2-[(2-chlorophenyl)methyl]morpholin-4-yl}-3-(pyrazin-2-yl)propan-1-one
2-chloro-4-({[(4,6-dimethylpyrimidin-2-yl)methyl]carbamoyl}amino)-N-propylbenzamide
5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-[3-(methylsulfanyl)propyl]pyridin-2-amine
N-[2-(4-methoxyphenyl)phenyl]-1-(1H-pyrazol-3-ylmethyl)piperidine-3-carboxamide
7-(3,4-dihydronaphthalen-2-yl)-4-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-cyclopentyl-8-[4-(ethylamino)pyrimidin-2-yl]-2,8-diazaspiro[5.5]undecan-3-one
3-(dimethylamino)-N-(2-methoxy-6-methylphenyl)pyrrolidine-1-carboxamide
3-(5-fluoro-1H-1,3-benzodiazol-2-yl)-1-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]propan-1-one
1-[(4-fluorophenyl)methyl]-4-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}piperazin-2-one
4-(3-phenylpropyl)-11-[(propan-2-yl)amino]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-(propan-2-yl)-5-(3,4,5-trimethoxyphenyl)-1,3-thiazole
1-[3-(3-fluoro-4-phenylbenzoyl)piperidin-1-yl]-2-(methylsulfanyl)ethan-1-one
{[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl}[2-(pyridin-3-yloxy)propyl]amine
1-cyclohexyl-3-(3-phenylpiperidine-1-carbonyl)-5-(pyrrolidine-1-carbonyl)-1,4-dihydropyridin-4-one
(3aS,6aR)-3-cyclopentyl-5-[(2-methoxyquinolin-3-yl)methyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
(4aS,8aR)-2-{[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-decahydroisoquinoline
5-(1-{3-chloro-6-methylpyrazolo[1,5-a]pyrimidine-2-carbonyl}pyrrolidin-2-yl)-3-(propan-2-yl)-1,2,4-oxadiazole
3-[2-(ethylsulfanyl)ethyl]-1-(2-fluoro-4-methylphenyl)urea
2-(2-methoxyethyl)-6-(thiomorpholine-4-carbonyl)-1,3-benzoxazole
1-(4-benzyl-6-hydroxy-1,4-diazepan-1-yl)-2-(2,5-dimethylphenyl)ethan-1-one
N-[2-(2-ethoxyphenoxy)ethyl]-4-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-methylbenzamide
8-(3-methoxypyrazin-2-yl)-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
methyl 4-[5-({methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)-1,2,4-oxadiazol-3-yl]benzoate
1-(4-tert-butylbenzoyl)-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
5-[(2-methoxyethyl)[(1-methyl-1H-pyrazol-4-yl)methyl]carbamoyl]-1H-imidazole-4-carboxylic acid
(1R,9S)-5-amino-3-(2,3-dihydro-1,4-benzodioxin-6-yl)-13-methyl-6,13-diazatricyclo[7.3.1.02,7]trideca-2,4,6-triene-4-carbonitrile
N-[(dimethyl-1,3-thiazol-5-yl)methyl]-3-(piperidin-3-yl)benzamide
5-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-1-(2-phenylethyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-benzyl-4-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]-1H-pyrazole
1-[4-(butan-2-yl)phenyl]-3-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]urea
N-[3-(1H-imidazol-1-yl)propyl]-2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
1-{2-methoxy-4-[({[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}amino)methyl]phenoxy}-3-(thiomorpholin-4-yl)propan-2-ol
methyl 5-[(cyclohex-3-en-1-ylmethyl)amino]-1-ethyl-3-(oxolane-3-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-methanesulfonyl-N-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]piperazine-1-carboxamide
7-fluoro-3-[({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amino)methyl]-1,2-dihydroquinolin-2-one
2-{4-[(4-fluoro-3-methoxyphenyl)methyl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
N-[1-(1,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
7-amino-4-(2,3-dihydro-1,4-benzodioxin-6-yl)-1,2,3,4-tetrahydro-1,8-naphthyridin-2-one
1-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-4-(pyrrolidine-1-sulfonyl)piperazine
2-(5-{4-[(pyridin-2-yl)amino]piperidine-1-carbonyl}-1H-pyrazol-3-yl)phenol
ethyl 2-{[3-({[3-(trifluoromethyl)phenyl]formamido}methyl)piperidine-1-carbonyl]amino}acetate
({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)[(1-ethyl-1H-imidazol-2-yl)methyl]methylamine
N,2,3,5-tetramethyl-N-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
4-[(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)carbamoyl]pyridin-1-ium-1-olate
4-(4-methyl-1H-pyrazol-1-yl)-1-[2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)ethyl]piperidine-4-carboxylic acid
1-[3-(5-benzyl-2-methylpyrimidin-4-yl)piperidin-1-yl]-2-(2-methoxyphenoxy)ethan-1-one
5-[2-(2-butyl-4-methyl-3-oxopiperazin-1-yl)-2-oxoethyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione