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7-chloro-N-[(3-methoxyphenyl)methyl]-3,5-dimethyl-1-benzofuran-2-carboxamide
3-(2H-1,3-benzodioxol-5-ylmethyl)-3-cyclopentyl-1-(pyridin-3-yl)urea
3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]-N-[2-(1,3-thiazol-4-yl)ethyl]propanamide
1-{4-[7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decane-2-carbonyl]phenyl}ethan-1-one
3-(5-fluoro-1H-1,3-benzodiazol-2-yl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}propanamide
6-(4-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}piperazin-1-yl)pyridine-3-carboxamide
N-[4-fluoro-3-({[(2R)-1,1,1-trifluoro-3-methylbutan-2-yl]carbamoyl}amino)phenyl]acetamide
3-[(3-cyclopropyl-1H-1,2,4-triazol-5-yl)methyl]-1-methyl-1H-indole
1-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
methyl 8-[(2,6-difluorophenyl)methyl]-2-oxo-1-(prop-2-en-1-yloxy)-1,8-diazaspiro[4.5]decane-4-carboxylate
2-ethyl-4-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]-1,3-oxazole-5-carboxamide
2-{4-[1-(prop-2-ene-1-sulfonyl)pyrrolidin-3-yl]piperidin-1-yl}pyrimidine
(4aS,8aR)-6-[(2-methyl-1H-imidazol-4-yl)methyl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-3-(5-fluoro-2-methoxybenzoyl)piperidine
1-(6-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}pyridin-2-yl)ethan-1-ol
{3-[(2,4-difluorophenyl)methyl]-1-[(3-phenyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}methanol
1-methyl-N-{[8-(3-methylbutanoyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}-3-propyl-1H-pyrazole-5-carboxamide
2-methyl-6-({1-[4-(1H-pyrazol-1-yl)phenyl]piperidin-4-yl}amino)heptan-2-ol
ethyl 1-[6-(2-chlorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]piperidine-2-carboxylate
1-ethyl-3-methyl-4-({1-[4-(methylsulfanyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}methyl)-1H-pyrazole
N-ethyl-3-(pyrimidin-5-yl)benzamide
1-cyclopentyl-4-{[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}piperazine
N-benzyl-N-ethyl-4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
6-{[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methyl}quinoxaline
N-[(1-hydroxycyclohexyl)methyl]-2-[1-(3-methylphenyl)-5-oxo-3-propyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]acetamide
(4aS,7aR)-1-(1H-1,3-benzodiazol-2-ylmethyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1,3-dimethyl-5-{1-[3-(trifluoromethyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-1H-pyrazole
2-(4-{[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}-1-(3-methylbutyl)piperazin-2-yl)ethan-1-ol
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-2-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
(3S,4R)-1-[(4-acetyl-1-methyl-1H-pyrrol-2-yl)methyl]-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
(1S,5R)-3-{[2-(methylsulfanyl)phenyl]methyl}-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(3,4-difluorophenyl)-1-(quinoline-6-carbonyl)piperidin-3-amine
N-[3-(methylsulfanyl)propyl]-2-[2,6,6-trimethyl-4-oxo-1-(propan-2-yl)-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
8-methoxy-2-oxo-N-(pyridin-4-ylmethyl)-1,2,3,4-tetrahydroquinoline-4-carboxamide
({6-chloro-2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[1,2-a]pyridin-3-yl}methyl)(methyl)(1,2-oxazol-3-ylmethyl)amine
4-methyl-2-{2-[2-(pyridin-4-yl)-1H-imidazol-1-yl]ethyl}-6-(trifluoromethyl)pyrimidine
1-(morpholin-4-yl)-3-{1-[3-(1H-pyrazol-1-yl)propyl]piperidin-3-yl}propan-1-one
2-[3-({[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)-1H-indol-1-yl]acetamide
2-fluoro-N-[2-(pyridin-2-ylsulfanyl)ethyl]-5-sulfamoylbenzamide
8-[1-(hydroxymethyl)cyclopropanecarbonyl]-2-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[3-(1H-pyrazol-1-yl)phenyl]-1-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
3-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propanoic acid
methyl({[4-(5-methylpyridin-2-yl)piperidin-4-yl]methyl}){[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}amine
N-cycloheptyl-4-oxo-1-(propan-2-yl)-5-[4-(pyridin-4-ylmethyl)piperazine-1-carbonyl]-1,4-dihydropyridine-3-carboxamide
4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-11-{[(3-fluorophenyl)methyl]amino}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
4-[1-(propan-2-yl)piperidine-4-carbonyl]-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
N-(2-acetamidophenyl)-2-{[1-(3-hydroxyadamantan-1-yl)ethyl]amino}acetamide
1-[(3-fluorophenyl)methyl]-4-(5-{[(4-fluorophenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)piperidine
5-chloro-6-(3,5-dimethoxyphenyl)-2-methylpyrimidin-4-ol
1-[1-(2,2-dimethylpropyl)piperidin-3-yl]-N-(3-hydroxypropyl)-1H-1,2,3-triazole-4-carboxamide