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N-{5-[2-(1H-imidazol-2-yl)-1H-imidazol-1-yl]-2-methoxyphenyl}methanesulfonamide
4-{2-[1-(1-methyl-1H-pyrazole-4-carbonyl)piperidin-2-yl]ethyl}morpholine
3-(morpholine-4-sulfonyl)-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]benzamide
3-{5-[methoxy(phenyl)methyl]-1,3,4-oxadiazol-2-yl}-N-methyl-N-(thiophen-2-ylmethyl)propanamide
(2R)-2-amino-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}-N-(pyridin-4-ylmethyl)propanamide
(4aR,7aS)-4-(2-ethoxybenzoyl)-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
N-{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-3-(pyrrolidin-1-yl)propanamide
2-(5-fluoro-2-methylphenyl)-N-[(5-oxopyrrolidin-2-yl)methyl]-N-(propan-2-yl)acetamide
N-cyclohexyl-N-[2-(dimethylamino)ethyl]-1-[(4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
N-[1-(7-{[4-(diethylamino)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]-2-methylbenzamide
2-(dimethyl-1,3-thiazol-5-yl)-1-[4-(2-phenoxyethyl)piperazin-1-yl]ethan-1-one
(5S,9aS,9bS)-5-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-(2,3-dihydro-1H-inden-2-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
[(3R,4R)-1-(2-chloro-6-fluoro-3-methylbenzoyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
(4aS,7aR)-1-[(3-hydroxyphenyl)methyl]-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-methyl-2-[3-oxo-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-9-yl]pyridine-3-carbonitrile
methyl({2-methylimidazo[1,2-a]pyridin-3-yl}methyl){[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
ethyl 4-[2-(dimethylamino)-2-(3-fluorophenyl)acetyl]piperazine-1-carboxylate
3-[(3-fluorophenyl)methyl]-N-[furan-2-yl(phenyl)methyl]-1,2-oxazole-5-carboxamide
3-(azocan-1-yl)-N-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-N-methylpropanamide
3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-[(4-methylphenyl)methyl]propanamide
5-({[1-(cyclopropylmethyl)-7-oxoazepan-4-yl]amino}methyl)-1,3-dimethyl-2,3-dihydro-1H-1,3-benzodiazol-2-one
3-[1-(6-ethyl-2-methylquinoline-4-carbonyl)piperidin-4-yl]-1,3-oxazolidin-2-one
3-cyclopropyl-N-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethyl)-1H-pyrazole-5-carboxamide
1-[5-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-1-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-4-phenylpiperazine
N-benzyl-1-(4,7-dimethylquinazolin-2-yl)-N-(2-hydroxyethyl)piperidine-3-carboxamide
3-(3-hydroxyquinoxalin-2-yl)-N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]propanamide
5-(oxolan-3-yl)-4-phenyl-1-[2-(thiophen-2-yl)ethyl]-1H-imidazole
3,5-difluoro-2-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyridine
N-({3-methyl-7-[4-(morpholin-4-yl)benzoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)thiophene-3-carboxamide
2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-1,3-oxazole-4-carboxylic acid
N-{[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)piperidin-3-yl]methyl}-1H-indazole-3-carboxamide
5-[4-(2,1-benzoxazole-3-carbonyl)piperazin-1-yl]-2-methyl-2,3-dihydropyridazin-3-one
2-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)-5-methoxyphenol
1-[(2,3-difluorophenyl)methyl]-4-[1-(1H-imidazole-5-carbonyl)pyrrolidin-3-yl]piperidine
[(4-ethyl-5-{1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
N-[3-(2-methoxyethoxy)phenyl]-4-(1H-pyrrole-2-carbonyl)piperazine-1-carboxamide
3-(cyclopropylsulfamoyl)-5-(4-methoxy-2-methylphenyl)benzoic acid
(3R,5S)-N-(2,3-dihydro-1H-inden-5-yl)-1-(2-phenylethyl)-5-(piperidine-1-carbonyl)piperidine-3-carboxamide
5-[({2,3-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1-methylpyrrolidin-2-one
5-[4-({2-oxo-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-3-yl}methyl)piperazin-1-yl]-2,3-dihydropyridazin-3-one
1-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-3-(naphthalene-1-carbonyl)piperidine
1-{4-[2-(3-methoxyphenyl)-1-[methyl(pyridin-2-ylmethyl)amino]ethyl]piperidin-1-yl}-2-(morpholin-4-yl)propan-1-one
3-chloro-N-cycloheptyl-4-[(1-methanesulfonylpiperidin-4-yl)oxy]benzamide
5-{[(5-fluoro-2-methylphenyl)methyl]amino}-N-(furan-2-ylmethyl)-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-chloro-N,6-dimethyl-N-[(3-methylpyridin-2-yl)methyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
3-(2-methyl-1H-indol-1-yl)-N-[2-(2-oxoimidazolidin-1-yl)ethyl]propanamide
methyl (2S,4S,5R)-2-ethyl-5-(4-fluorophenyl)-1-methyl-4-(piperidine-1-carbonyl)pyrrolidine-2-carboxylate
(1R,5S,6R)-3-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}-3-azabicyclo[3.1.0]hexane-6-carboxylic acid
methyl 3-[(1,2,5-thiadiazol-3-ylformamido)methyl]-5-[3-(trifluoromethyl)benzamido]benzoate
3-(1-{2-methyl-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidine-6-carbonyl}piperidin-3-yl)benzoic acid